Affinity DataKi: 0.0910nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 0.980nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of recombinant human AChE expressed in HEK293 cells using varying levels of acetylthiocholine iodide as substrate by Lineweaver-burk plot ...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]8-OH DPAT from rat 5HT1A receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of recombinant human AChE expressed in HEK293 cells using varying levels of acetylthiocholine iodide as substrate by Lineweaver-burk plot ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of recombinant human AChE expressed in HEK293 cells using varying levels of acetylthiocholine iodide as substrate by Lineweaver-burk plot ...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Inhibition of recombinant human AChE expressed in HEK293 cells using varying levels of acetylthiocholine iodide as substrate by Lineweaver-burk plot ...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Inhibition of recombinant human AChE expressed in HEK293 cells using varying levels of acetylthiocholine iodide as substrate by Lineweaver-burk plot ...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Displacement of [3H]DTG from sigma2 receptor in rat liver membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Inhibition of recombinant human AChE expressed in HEK293 cells using varying levels of acetylthiocholine iodide as substrate by Lineweaver-burk plot ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of recombinant human AChE expressed in HEK293 cells using varying levels of acetylthiocholine iodide as substrate by Lineweaver-burk plot ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 62nMAssay Description:Inhibition of recombinant human AChE expressed in HEK293 cells using varying levels of acetylthiocholine iodide as substrate by Lineweaver-burk plot ...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Displacement of [3H]DOB from rat 5HT2A receptor expressed in mouse NIH/3T3 cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Consejo Superior de Investigaciones Cient�ficas (IQM-CSIC)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
