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TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50259713(CHEMBL4095303)
Affinity DataEC50:  1.01E+4nMAssay Description:Partial agonist activity at human alpha4beta2 nAChR expressed in GH4CL cells by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50549595(CHEMBL4741357)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at wild type human alpha4beta2 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50357064(CHEMBL1917231)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at wild type human alpha4beta2 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50259713(CHEMBL4095303)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at wild type human alpha4beta2 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50549595(CHEMBL4741357)
Affinity DataEC50:  8.70E+3nMAssay Description:Partial agonist activity at human alpha3beta4 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50357064(CHEMBL1917231)
Affinity DataEC50:  1.70E+4nMAssay Description:Partial agonist activity at human alpha3beta4 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50549596(CHEMBL4785648)
Affinity DataEC50:  1.90E+4nMAssay Description:Partial agonist activity at human alpha3beta4 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50549595(CHEMBL4741357)
Affinity DataEC50:  5nMAssay Description:Partial agonist activity at human alpha4beta2 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50357064(CHEMBL1917231)
Affinity DataEC50:  300nMAssay Description:Partial agonist activity at human alpha4beta2 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50549596(CHEMBL4785648)
Affinity DataEC50:  1.40E+4nMAssay Description:Partial agonist activity at human alpha4beta2 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50259713(CHEMBL4095303)
Affinity DataEC50:  1.01E+4nMAssay Description:Partial agonist activity at human alpha4beta2 transfected in rat GH4-C1 cells at holding potential of -70 mV by whole cell patch clamp electrophysiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50600203(CHEMBL5183330)
Affinity DataEC50:  2.34E+3nMAssay Description:Partial agonist activity at high sensitivity isoform human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50357064(CHEMBL1917231)
Affinity DataEC50:  129nMAssay Description:Partial agonist activity at high sensitivity isoform human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50549596(CHEMBL4785648)
Affinity DataEC50:  799nMAssay Description:Partial agonist activity at high sensitivity isoform human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50600203(CHEMBL5183330)
Affinity DataEC50:  3.00E+3nMAssay Description:Partial agonist activity at low sensitivity isoform human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acety...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50357064(CHEMBL1917231)
Affinity DataEC50:  2.18E+4nMAssay Description:Partial agonist activity at low sensitivity isoform human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acety...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50549596(CHEMBL4785648)
Affinity DataEC50:  4.80E+3nMAssay Description:Partial agonist activity at low sensitivity isoform human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acety...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50549595(CHEMBL4741357)
Affinity DataEC50:  1.85E+4nMAssay Description:Partial agonist activity at low sensitivity isoform human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acety...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50357061(CHEMBL1917228)
Affinity DataKd:  0.300nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in Sprague-Dawley rat cerebral cortex by beta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187306(1-{[(2R)-3-(benzyloxy)-1-{1,1-dioxo-2H-spiro[1-ben...)
Affinity DataEC50:  5nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187307(1-{[(2R)-3-(benzyloxy)-1-oxo-1-{2H-spiro[1-benzoth...)
Affinity DataEC50:  10nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50370712(CHEMBL1793862)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187310(2-amino-N-((R)-1-((S)-3a-benzyl-2-ethyl-3-oxo-2,3,...)
Affinity DataEC50:  4nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187308(L-162970 | 1N-[1-benzyloxymethyl-2-oxo-2-spiro[2,3...)
Affinity DataEC50:  17nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187312(1-methyl-1-{[(2R)-1-oxo-5-phenyl-1-{2H-spiro[1-ben...)
Affinity DataEC50:  4.80nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187313(1-methyl-1-((R)-1-{2'-[(3-methyl-ureido)-methyl]-b...)
Affinity DataEC50:  1nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187314(1-methyl-1-{[(2R)-1-oxo-5-phenyl-1-{2H-spiro[1-ben...)
Affinity DataEC50:  2.70nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187315(1-{[(2R)-1-{1,1-dioxo-2H-spiro[1-benzothiophene-3,...)
Affinity DataEC50:  6nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187317(1-{[(2R)-1-{2,3-dihydrospiro[indene-1,4'-piperidin...)
Affinity DataEC50:  22nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187318(1-((R)-1-((S)-3a-benzyl-2-methyl-3-oxo-2,3,3a,4,6,...)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187316(1-{[(2R)-1-[(3R)-3-hydroxy-2,3-dihydrospiro[indene...)
Affinity DataEC50:  0.600nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187319(1-{[(2R)-1-{1,1-dioxo-2H-spiro[1-benzothiophene-3,...)
Affinity DataEC50:  1.10nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187320(1-{[(2R)-3-(benzyloxy)-1-oxo-1-{2H-spiro[1-benzofu...)
Affinity DataEC50:  8.5nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187322(1-{[(2R)-1-{2,3-dihydrospiro[indene-1,4'-piperidin...)
Affinity DataEC50:  10nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187321(2-amino-N-[(R)-2-((S)-3a-benzyl-3-oxo-2,3,3a,4,6,7...)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187323(5-amino-5-methyl-hex-2-enoic acid ((R)-1-{[2-(2-me...)
Affinity DataEC50:  18nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50066816((E)-5-Amino-5-methyl-hex-2-enoic acid methyl-{(R)-...)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187325(1-((R)-1-{2'-[(3-ethyl-ureido)-methyl]-biphenyl-4-...)
Affinity DataEC50:  6nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50370713(CHEMBL1162926)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187326((R,E)-2-methyl-6-(methyl(1-(methyl(2-(thiophen-2-y...)
Affinity DataEC50:  7.5nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50065107((R)-1-[(R)-2-(2-amino-2-methyl-propionylamino)-3-(...)
Affinity DataEC50:  1.60nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187327(1-{[(2R)-1-{1,1-dioxo-2H-spiro[1-benzothiophene-3,...)
Affinity DataEC50:  2.10nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50370714(CHEMBL1161827)
Affinity DataEC50:  2nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187329(5-amino-5-methyl-hex-2-enoic acid [(R)-1-({2-[2-(2...)
Affinity DataEC50:  5nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187330((R,E)-N,2-dimethyl-6-(methyl(1-(methyl(2-(thiophen...)
Affinity DataEC50:  0.800nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187332(1-{[(2R)-3-(1H-indol-3-yl)-1-oxo-1-{2H-spiro[1-ben...)
Affinity DataEC50:  5.60nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187331((R,E)-6-((1-((2-(2-hydroxyethoxy)phenethyl)(methyl...)
Affinity DataEC50:  5nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50370715(CHEMBL1161826)
Affinity DataEC50:  8.5nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187333(5-amino-5-methyl-hex-2-enoic acid {(R)-2-biphenyl-...)
Affinity DataEC50:  5nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50187335(1-methyl-1-{[(2R)-1-oxo-4-phenyl-1-{2H-spiro[1-ben...)
Affinity DataEC50:  57nMAssay Description:Activity at human GHS-R1a receptor in rat pituitary cells assessed as GH releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
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