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Targetneuronal acetylcholine receptor subunit alpha-2(Western clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.00240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86042(NEP)
Affinity DataKi:  0.00310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.00380nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.00400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  0.00850nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.00920nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Western clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0130nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068612(2-(8-Bromo-benzo[1,2-b;4,5-b']difuran-4-yl)-1-meth...)
Affinity DataKi:  0.0200nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Western clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288406(1-(2-Acetylamino-3-phenyl-propionyl)-pyrrolidine-2...)
Affinity DataKi:  0.0400nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068612(2-(8-Bromo-benzo[1,2-b;4,5-b']difuran-4-yl)-1-meth...)
Affinity DataKi:  0.0400nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50451005(CHEMBL290376 | DuP-714)
Affinity DataKi:  0.0420nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
TargetCholinergic receptor, nicotinic alpha 1(clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288406(1-(2-Acetylamino-3-phenyl-propionyl)-pyrrolidine-2...)
Affinity DataKi:  0.0450nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185364(CHEMBL2371908 | CHEMBL415187 | Sub[-Tyr-Arg-Leu-Ar...)
Affinity DataKi:  0.0500nMAssay Description:Displacement of [125I]hPP from human NPY4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Western clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Western clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  0.0620nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(CHEMBL2110365 | GR-231118)
Affinity DataKi:  0.0700nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  0.0770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50099198(CHEMBL429531 | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly...)
Affinity DataKi:  0.0800nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50098525(2-(8-Bromo-benzo[1,2-b;4,5-b']difuran-4-yl)-1-meth...)
Affinity DataKi:  0.110nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289586(3-Methyl-2'-sulfamoyl-biphenyl-4-carboxylic acid [...)
Affinity DataKi:  0.110nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50361235(CHEMBL1934525)
Affinity DataKi:  0.170nMAssay Description:Displacement of N-[3H]-methylhistamine from histamine H3 receptor in rat cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50352357(CHEMBL558655)
Affinity DataKi:  0.182nMAssay Description:Displacement of N-[3H]methylhistamine from histamine H3 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068612(2-(8-Bromo-benzo[1,2-b;4,5-b']difuran-4-yl)-1-meth...)
Affinity DataKi:  0.190nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50361237(CHEMBL1934527)
Affinity DataKi:  0.200nMAssay Description:Displacement of N-[3H]-methylhistamine from histamine H3 receptor in rat cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50084682(1-[3-(4-Carbamimidoyl-phenyl)-2-(2-methyl-1,2,3,4-...)
Affinity DataKi:  0.210nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholinergic receptor nicotinic alpha 5 subunit(clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(CHEMBL429531 | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly...)
Affinity DataKi:  0.230nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068612(2-(8-Bromo-benzo[1,2-b;4,5-b']difuran-4-yl)-1-meth...)
Affinity DataKi:  0.230nMAssay Description:Antagonistic activity measured for 5-hydroxytryptamine 2A receptor using [3H]-MDL- 100,907 as radioligand in rat cortical homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068612(2-(8-Bromo-benzo[1,2-b;4,5-b']difuran-4-yl)-1-meth...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]MDL100907 from 5HT2A receptor in Sprague-Dawley rat brain by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50098526(2-(8-Bromo-benzo[1,2-b;4,5-b']difuran-4-yl)-1-meth...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50409214(CHEMBL2110365 | GR-231118)
Affinity DataKi:  0.260nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50098532(2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']d...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099197(CHEMBL411117 | Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  0.270nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50098530(1-Methyl-2-(8-trifluoromethyl-benzo[1,2-b;4,5-b']d...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2A receptor using [3H]-DOB as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50352358(CHEMBL558456)
Affinity DataKi:  0.295nMAssay Description:Displacement of N-[3H]methylhistamine from histamine H3 receptor in rat cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Human)
University of New Mexico Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKi:  0.300nMAssay Description:Displacement of E2-Alexa633 from GFP-tagged ERalpha expressed in COS7 cells by FACSMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50052337(2-(8-bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']d...)
Affinity DataKi:  0.300nMAssay Description:Agonistic activity at cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50052337(2-(8-bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']d...)
Affinity DataKi:  0.300nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50098525(2-(8-Bromo-benzo[1,2-b;4,5-b']difuran-4-yl)-1-meth...)
Affinity DataKi:  0.310nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2A receptor using [3H]-DOB as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50098536(1-Methyl-2-(8-trifluoromethyl-benzo[1,2-b;4,5-b']d...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2A receptor using [3H]-DOB as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50094092(CHEMBL336661 | N-(3-Bromo-2'-sulfamoyl-biphenyl-4-...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(clawed frog)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289591(2'-Diethylsulfamoyl-3-methyl-biphenyl-4-carboxylic...)
Affinity DataKi:  0.360nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEstrogen receptor beta(Human)
University of New Mexico Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKi:  0.380nMAssay Description:Displacement of E2-Alexa633 from GFP-tagged ERbeta expressed in COS7 cells by FACSMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50098530(1-Methyl-2-(8-trifluoromethyl-benzo[1,2-b;4,5-b']d...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50373621(CHEMBL403414)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125]PYY from human chimeric NPY Y5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289587(3-Methyl-biphenyl-4-carboxylic acid [(R)-4-guanidi...)
Affinity DataKi:  0.420nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
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