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TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50111110(2N-(4-Benzamidinemethyl)-1-[2-aminosulfonamido-3,3...)
Affinity DataKi:  0.00300nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50111101((S)-1-((R)-2-Methanesulfonylamino-3,3-diphenyl-pro...)
Affinity DataKi:  0.00300nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131789(1-(2-sulfonamide-amino-3,3-diphenyl-propionyl)-pyr...)
Affinity DataKi:  0.00400nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50111105((S)-1-((R)-2-Methanesulfonylamino-3,3-diphenyl-pro...)
Affinity DataKi:  0.00500nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131790(1-(2-sulfonamideamino-3,3-diphenyl-propionyl)-pyrr...)
Affinity DataKi:  0.00800nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131795(1-(2-sulfonamideamino-3,3-diphenyl-propionyl)-pyrr...)
Affinity DataKi:  0.0100nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131778(3-(1-Benzhydryl-2-{2-[(5-carbamimidoyl-thiophen-2-...)
Affinity DataKi:  0.0100nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50111120(2N-(4-Benzamidinemethyl)-1-[2-Aminoaceticacid-3,3-...)
Affinity DataKi:  0.0130nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131780((1-Benzhydryl-2-{2-[(5-carbamimidoyl-thiophen-2-yl...)
Affinity DataKi:  0.0150nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131796((1-Benzhydryl-2-{2-[(5-carbamimidoyl-thiophen-2-yl...)
Affinity DataKi:  0.0150nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131791(1-(2-sulfonamideamino-3,3-diphenyl-propionyl)-pyrr...)
Affinity DataKi:  0.0150nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131792((1-Benzhydryl-2-{2-[(6-carbamimidoyl-pyridin-3-ylm...)
Affinity DataKi:  0.0170nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131798(1-(2-Methylamino-3,3-diphenyl-propionyl)-pyrrolidi...)
Affinity DataKi:  0.0200nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131782(1-(2-sulfonamide-amino-3,3-diphenyl-propionyl)-pyr...)
Affinity DataKi:  0.0200nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50111122(2N-(4-Benzamidinemethyl)-1-[2-Carbamicacidmethyles...)
Affinity DataKi:  0.0300nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131787((1-Benzhydryl-2-{2-[(5-carbamimidoyl-thiophen-3-yl...)
Affinity DataKi:  0.100nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131781(1-(2-sulfonamide-amino-3,3-diphenyl-propionyl)-pyr...)
Affinity DataKi:  0.120nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131797(1-(2-sulfonamide-amino-3,3-diphenyl-propionyl)-pyr...)
Affinity DataKi:  0.160nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131779((1-Benzhydryl-2-{2-[(4-carbamimidoyl-thiophen-2-yl...)
Affinity DataKi:  0.170nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131780((1-Benzhydryl-2-{2-[(5-carbamimidoyl-thiophen-2-yl...)
Affinity DataKi:  0.300nMAssay Description:In vitro inhibition constant (Ki) against human human trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131784(2-{4-[(Z)-amino(hydrazono)methyl]phenyl}-N-cyclope...)
Affinity DataKi:  0.400nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131783(1-(2-sulfonamide-amino-3,3-diphenyl-propionyl)-pyr...)
Affinity DataKi:  0.430nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131788((1-Benzhydryl-2-{2-[(5-carbamimidoyl-thiophen-3-yl...)
Affinity DataKi:  0.600nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131793((1-Benzhydryl-2-{2-[(4-carbamimidoyl-thiazol-2-ylm...)
Affinity DataKi:  0.640nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131777((1-Benzhydryl-2-{2-[(5-carbamimidoyl-furan-3-ylmet...)
Affinity DataKi:  1.40nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310131((2-hydroxy-4-(3-isobutyl-5-methylhexylidene)-5-oxo...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bovine)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131780((1-Benzhydryl-2-{2-[(5-carbamimidoyl-thiophen-2-yl...)
Affinity DataKi:  3nMAssay Description:In vitro inhibition constant (Ki) against human bovine trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310107((E)-(2-(hydroxymethyl)-4-(8-(nonyloxy)octylidene)-...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataKi:  4nMAssay Description:In vitro inhibition constant (Ki) against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310104((E)-(2-(hydroxymethyl)-4-(16-methoxyhexadecylidene...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310105((Z)-(2-(hydroxymethyl)-4-(16-methoxyhexadecylidene...)
Affinity DataKi:  5nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310120((E)-(2-(hydroxymethyl)-5-oxo-4-(16-oxohexadecylide...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310115((E)-(4-(16-hydroxyhexadecylidene)-2-(hydroxymethyl...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310124((E)-methyl 16-(5-(hydroxymethyl)-2-oxo-5-(pivaloyl...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310101((Z)-(2-(hydroxymethyl)-5-oxo-4-tetradecylidenetetr...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310112((E)-(2-(hydroxymethyl)-4-(4-(nonyloxy)butylidene)-...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310110((E)-(2-(hydroxymethyl)-4-(8-(isopentyloxy)octylide...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310100((E)-(2-(hydroxymethyl)-5-oxo-4-tetradecylidenetetr...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310125((E)-(4-(16-(formyloxy)hexadecylidene)-2-(hydroxyme...)
Affinity DataKi:  8nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310106((E)-(2-(hydroxymethyl)-5-oxo-4-(8-(pentyloxy)octyl...)
Affinity DataKi:  8.10nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310116((Z)-(4-(16-hydroxyhexadecylidene)-2-(hydroxymethyl...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310103((E)-(2-(hydroxymethyl)-4-(12-methoxydodecylidene)-...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310130((E)-(4-(16-acetamidohexadecylidene)-2-(hydroxymeth...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310126((E)-(4-(16-acetoxyhexadecylidene)-2-(hydroxymethyl...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310111((E)-(4-(8-(cyclopentyloxy)octylidene)-2-(hydroxyme...)
Affinity DataKi:  10nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310127((E)-16-(5-(hydroxymethyl)-2-oxo-5-(pivaloyloxymeth...)
Affinity DataKi:  11nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310121((Z)-(2-(hydroxymethyl)-5-oxo-4-(16-oxohexadecylide...)
Affinity DataKi:  11nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310114((E)-(4-(12-hydroxydodecylidene)-2-(hydroxymethyl)-...)
Affinity DataKi:  15nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50310128((E)-(4-(16-azidohexadecylidene)-2-(hydroxymethyl)-...)
Affinity DataKi:  16nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Human)
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50131780((1-Benzhydryl-2-{2-[(5-carbamimidoyl-thiophen-2-yl...)
Affinity DataKi:  22.5nMAssay Description:In vitro inhibition constant (Ki) against human Coagulation factor X was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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