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TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21940(Ghrelin | US20240190875, Example Ghrelin)
Affinity DataEC50:  1.40nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21941(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  1.90nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21942(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  3nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21943(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  5.5nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21944(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  14.6nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21945(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  3.80nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21946(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  1nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21947(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  10.1nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21948(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  82.5nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21949(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  3.30nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21950(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  7.90nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21951(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  9.5nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM21952(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  45.3nMpH: 7.2 T: 2°CAssay Description:The functional FLIPR assay was developed from H4 glioma cells in which expression of the endogenous human GHS receptor was enhanced by RAGE-activatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM24657(1-methyl-4-phenyl-1H-imidazole | 4-phenylimidazole...)
Affinity DatapH: 6.5 T: 2°CAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM24658(1-benzyl-4-phenyl-1H-imidazole | 4-phenylimidazole...)
Affinity DatapH: 6.5 T: 2°CAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM24659(2-(4-phenyl-1H-imidazol-1-yl)ethan-1-amine | 4-phe...)
Affinity DatapH: 6.5 T: 2°CAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM24660(3-(4-phenyl-1H-imidazol-1-yl)propan-1-amine | 4-ph...)
Affinity DatapH: 6.5 T: 2°CAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM24661((4-phenyl-1H-imidazol-2-yl)methanol | 4-phenylimid...)
Affinity DatapH: 6.5 T: 2°CAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM24662(methyl[(4-phenyl-1H-imidazol-2-yl)methyl]amine | 4...)
Affinity DatapH: 6.5 T: 2°CAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM24682(5-phenyl-1,3-thiazole | 5-phenyl-1,3-thiazole, 34)
Affinity DatapH: 6.5 T: 2°CAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM16215(CHEMBL390066 | JMC514968 Compound 35 | 4-phenyl-1H...)
Affinity DatapH: 6.5 T: 2°CAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM12357(CHEMBL178516 | US8609708, 14 | 3-(1H-imidazol-4-yl...)
Affinity DataAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
Bryn Mawr College

LigandPNGBDBM24684(3-(furan-2-yl)pyridine | 3-furan-2-ylpyridine, 36)
Affinity DataAssay Description:The IC50 inhibition assays were performed in a 96-well microtiter plate format using purified recombinant IDO, which was added to the substrate, L-tr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50544056(CHEMBL4644327)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at LRH1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50544057(CHEMBL4637563)
Affinity DataEC50:  400nMAssay Description:Agonist activity at LRH1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546597(CHEMBL4750282)
Affinity DataKd:  1.28E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546597(CHEMBL4750282)
Affinity DataKd:  1.28E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546598(CHEMBL4749028)
Affinity DataKd:  9.47E+3nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546598(CHEMBL4749028)
Affinity DataKd:  9.47E+3nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546599(CHEMBL4745577)
Affinity DataKd:  5.72E+3nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546599(CHEMBL4745577)
Affinity DataKd:  5.72E+3nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546600(CHEMBL4751198)
Affinity DataKd:  1.19E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546600(CHEMBL4751198)
Affinity DataKd:  1.19E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546601(CHEMBL4747153)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546601(CHEMBL4747153)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546602(CHEMBL4749475)
Affinity DataKd:  9.17E+3nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546602(CHEMBL4749475)
Affinity DataKd:  9.17E+3nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546603(CHEMBL4797448)
Affinity DataKd:  3.36E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546603(CHEMBL4797448)
Affinity DataKd:  3.36E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546604(CHEMBL4745888)
Affinity DataKd:  2.49E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50546604(CHEMBL4745888)
Affinity DataKd:  2.49E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50370453(Lactose, anhydrous | LACTOSE)
Affinity DataKd:  3.79E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50370453(Lactose, anhydrous | LACTOSE)
Affinity DataKd:  3.79E+4nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50230648(CHEMBL3764379)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetGalectin-8(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50230648(CHEMBL3764379)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to N-terminal domain of human galectin-8 (8-154 residues) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50511467(CHEMBL4551205)
Affinity DataEC50:  100nMAssay Description:Agonist activity at LRH-1 (unknown origin) transfected in human HeLa cells measured after 24 hrs by Dual Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50605640(CHEMBL5198453)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at LRH-1 (unknown origin) transfected in human HeLa cells measured after 24 hrs by Dual Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataEC50:  43nMAssay Description:Agonist activity at LRH-1 (unknown origin) transfected in human HeLa cells measured after 24 hrs by Dual Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50511467(CHEMBL4551205)
Affinity DataKd:  2.10E+3nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50605640(CHEMBL5198453)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
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