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TargetGlucagon-like peptide 1 receptor(Rat)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50604669(CHEMBL5208485)
Affinity DataEC50:  0.00800nMAssay Description:Positive allosteric modulator activity at GLP-1R in rat INS1 beta-cells assessed potentiation of GLP-1(7-36)NH2 induced insulin secretion incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205313(d[Leu4]AVP | CHEMBL265859)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50604669(CHEMBL5208485)
Affinity DataEC50:  0.100nMAssay Description:Positive allosteric modulator activity at human GLP-1R expressed in HEK293 cells assessed as potentiation of GLP-1(7-36)NH2 induced cAMP accumulation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205305(d[Arg4]AVP | CHEMBL375324)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205309(d[Leu4,Lys8]VP | CHEMBL412972)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205296(d[Arg4,Dab8]VP | CHEMBL385739)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205305(d[Arg4]AVP | CHEMBL375324)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145126((2S)-2-{[(2R)-1-{[(4S,7R,10S,13R,16S)-13-benzyl-7-...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205297(d[Leu4,Dab8]VP | CHEMBL412973)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Rat)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50604669(CHEMBL5208485)
Affinity DataEC50:  0.25nMAssay Description:Positive allosteric modulator activity at GLP-1R in rat INS1 beta-cells assessed potentiation of GLP-1(7-36)NH2 induced insulin secretion incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205300(d[Val4]AVP | CHEMBL221436)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205301(d[Leu4,Orn8]VP | CHEMBL375188)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205304(dVDAVP | CHEMBL435323)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145118(d[Val4]AVP | CHEMBL412353)
Affinity DataKi:  0.290nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205300(d[Val4]AVP | CHEMBL221436)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145112((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.370nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205303(d[Leu4,Dap8]VP | CHEMBL373968)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50370387(CHEMBL1790575)
Affinity DataKi:  0.420nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145124((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-10-but...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205306(d[Orn4,Lys8]VP | CHEMBL375323)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205311(d[Orn4]AVP | CHEMBL375096)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145107((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-10-(3-aminopropy...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145117((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205292(d[Arg4,Orn8]VP | CHEMBL385068)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205298(d[Arg4,Lys8]VP | CHEMBL375325)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145108((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.780nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205307(d[Cha4,Dab8]VP | CHEMBL412742)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205310(d[Orn4,Orn8]VP | CHEMBL219272)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetOxytocin receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]AVP from rat OT receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145111((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  1nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145109((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145118(d[Val4]AVP | CHEMBL412353)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against human vasopressin V2 receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetOxytocin receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]AVP from rat OT receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145123(d[Cha4]AVP | CHEMBL410573)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50594511(CHEMBL5182278)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to LPA2 receptor (unknown origin) by free solution assay-compensated interferometric reader (FSA-CIR) techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205312(d[Cha4]AVP | CHEMBL265858)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145111((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against human vasopressin V2 receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145129((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7,10-b...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against human vasopressin V1a receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145129((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7,10-b...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205296(d[Arg4,Dab8]VP | CHEMBL385739)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145122((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-10-(4-aminobutyl...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205293(d[Cha4,Lys8]VP | CHEMBL221485)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145115((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  2nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145109((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity against human vasopressin V2 receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Medical College of Ohio

Curated by ChEMBL
LigandPNGBDBM50145111((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity against human vasopressin V1a receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205295(d[Cha4,Orn8]VP | CHEMBL263090)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205292(d[Arg4,Orn8]VP | CHEMBL385068)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
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