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TargetOxytocin receptor(Mouse)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  62nMAssay Description:Agonist activity at mouse OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506302(CHEMBL4546106)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553319(CHEMBL4796966)
Affinity DataEC50:  10nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077136(CHEMBL3416749)
Affinity DataKd:  61nMAssay Description:Binding affinity to V1aR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553345(CHEMBL4759930)
Affinity DataEC50:  21nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553354(CHEMBL4741725)
Affinity DataEC50:  15nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553314(CHEMBL4741249)
Affinity DataEC50:  9.00E+3nMAssay Description:Activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human V2 receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546625(CHEMBL4757910)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546625(CHEMBL4757910)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553310(CHEMBL4792908)
Affinity DataEC50:  7.80nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553356(CHEMBL4780405)
Affinity DataEC50:  5.20nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553313(CHEMBL4778891)
Affinity DataEC50:  830nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins in presence of 10% FB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553309(CHEMBL4745870)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553325(CHEMBL4756860)
Affinity DataEC50:  1.60E+3nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553380(CHEMBL4746732)
Affinity DataEC50:  23nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546641(CHEMBL4789614)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546641(CHEMBL4789614)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50139178(CHEMBL3763342)
Affinity DataEC50:  61nMAssay Description:Agonist activity at recombinant human OTR expressed in CHO-DUKX-A2 cells assessed as stimulation of intracellular calcium concentration by calcium 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546626(CHEMBL4800389)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546626(CHEMBL4800389)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553353(CHEMBL4743065)
Affinity DataEC50:  840nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553341(CHEMBL4788527)
Affinity DataEC50:  12nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553373(CHEMBL4753962)
Affinity DataEC50:  630nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546628(CHEMBL4748622)
Affinity DataEC50:  0.650nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546628(CHEMBL4748622)
Affinity DataEC50:  0.650nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetNeuropeptide FF receptor 2(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553307(CHEMBL4756913)
Affinity DataEC50:  920nMAssay Description:Activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553334(CHEMBL4787106)
Affinity DataEC50:  920nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546654(CHEMBL4756925)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50546654(CHEMBL4756925)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human NPY2R expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation incubated for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50139178(CHEMBL3763342)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human V1a receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553327(CHEMBL4760120)
Affinity DataEC50:  16nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506306(CHEMBL4460622)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553311(CHEMBL4751018)
Affinity DataEC50:  310nMAssay Description:Activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077134(CHEMBL3416751)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1bR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  2.70E+4nMAssay Description:Agonist activity at human V1b receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50077137(CHEMBL3416754)
Affinity DataKd:  1.90nMAssay Description:Binding affinity to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077137(CHEMBL3416754)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to V1bR (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506296(CHEMBL4537162)
Affinity DataEC50:  193nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553314(CHEMBL4741249)
Affinity DataEC50:  8.20nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553346(CHEMBL4782739)
Affinity DataEC50:  7.30nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553308(CHEMBL4742191)
Affinity DataEC50:  9.10nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins in presence of 10% FB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553309(CHEMBL4745870)
Affinity DataEC50:  470nMAssay Description:Activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50506296(CHEMBL4537162)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in CHOK1 cells assessed as increase in cAMP level measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553359(CHEMBL4777620)
Affinity DataEC50:  720nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553371(CHEMBL4783313)
Affinity DataEC50:  40nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553317(CHEMBL4741546)
Affinity DataEC50:  33nMAssay Description:Activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Calibr At Scripps Research

Curated by ChEMBL
LigandPNGBDBM50553310(CHEMBL4792908)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
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