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TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 50nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424306(CHEMBL2314485)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424312(CHEMBL2314488)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424313(CHEMBL2314487)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50006805(CHEMBL29097 | 3-(3-(tert-butylthio)-1-(4-chloroben...)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424307(CHEMBL2314484)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424308(CHEMBL2314483)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424314(CHEMBL2314486)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424304(CHEMBL2314489)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424305(CHEMBL2314492)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424311(CHEMBL2314480)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394654(CHEMBL188181)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424309(CHEMBL2314482)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424310(CHEMBL2314481)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424303(CHEMBL2314490)
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394652(CHEMBL2165236)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394653(CHEMBL2165235)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394655(CHEMBL2165237)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM26663((2S)-5,7-dihydroxy-8-(3-methylbut-2-en-1-yl)-2-phe...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin E synthase(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50424315(CHEMBL2314491)
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of mPGES1 (unknown origin) using PGH2 as substrate incubated for 30 mins prior to substrate addition by PGH2-coupled spectrophotometric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394656(CHEMBL2165240)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM21447(4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...)
Affinity DataKi: <1nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630076(CHEMBL5439741)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630094(CHEBI:66437 | Schweinfurthin G | SCHWEINFURTHIN G)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630093(CHEBI:66352 | Vedelianin | VEDELIANIN)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630092(CHEBI:66435 | Schweinfurthin E | SCHWEINFURTHIN E)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630083(CHEMBL5402401)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630095(CHEBI:66436 | Schweinfurthin F | SCHWEINFURTHIN F)
Affinity DataKi:  6nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630078(CHEMBL5418635)
Affinity DataKi:  16nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630089(CHEMBL5397075)
Affinity DataKi:  31nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630090(CHEMBL5401329)
Affinity DataKi:  37nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630088(CHEMBL5416867)
Affinity DataKi:  43nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630075(CHEMBL5414636)
Affinity DataKi:  46nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630080(CHEMBL5433096)
Affinity DataKi:  64nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630084(CHEMBL5394654)
Affinity DataKi:  119nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630087(CHEMBL5417439)
Affinity DataKi:  254nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630086(CHEBI:66438 | Schweinfurthin H | SCHWEINFURTHIN H)
Affinity DataKi:  401nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630081(CHEMBL5409120)
Affinity DataKi:  523nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630082(CHEMBL5433829)
Affinity DataKi:  829nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630085(CHEMBL5399392)
Affinity DataKi:  1.07E+3nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630091(Mappain | MAPPAIN)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630079(CHEMBL5396667)
Affinity DataKi:  3.22E+3nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630077(CHEMBL5397623)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022583(CHEMBL3298854)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of fluorescein-labeled BID from His-tagged MCL-1 (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022622(CHEMBL3299033)
Affinity DataKi:  5.90E+3nMAssay Description:Displacement of fluorescein-labeled BID from His-tagged MCL-1 (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022568(CHEMBL3298853)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022568(CHEMBL3298853)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of fluorescein-labeled BID from His-tagged MCL-1 (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022567(CHEMBL3298852)
Affinity DataKi:  1.40E+4nMAssay Description:Displacement of fluorescein-labeled BID from His-tagged MCL-1 (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022567(CHEMBL3298852)
Affinity DataKi:  1.92E+4nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022622(CHEMBL3299033)
Affinity DataKi:  1.94E+4nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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