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TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316303(((2R,3S,4R,5R)-5-(2-amino-7-methyl-6-oxo-1H-purin-...)
Affinity DataKd:  45nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316302(((2R,3S,4R,5R)-5-(2-amino-7-methyl-6-oxo-1H-purin-...)
Affinity DataKd:  10nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316315(((2R,3S,4R,5R)-5-(2-Amino-7-(4-fluorobenzyl)-6-oxo...)
Affinity DataKd:  7.51E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in absence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316311(((2R,3S,4R,5R)-5-(2-Amino-7-(2-fluorobenzyl)-6-oxo...)
Affinity DataKd:  3.36E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in absence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316306(((2R,3S,4R,5R)-5-(2-Amino-7-(3-fluorobenzyl)-6-oxo...)
Affinity DataKd:  2.23E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in absence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316305(((2R,3S,4R,5R)-5-(2-amino-7-benzyl-6-oxo-1H-purin-...)
Affinity DataKd:  790nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in absence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316320(((2R,3S,4R,5R)-5-(2-Amino-7-(2-methylbenzyl)-6-oxo...)
Affinity DataKd:  6.91E+4nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316319(((2R,3S,4R,5R)-5-(2-Amino-7-(2,5-dichlorobenzyl)-6...)
Affinity DataKd:  1.73E+4nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316318(((2R,3S,4R,5R)-5-(2-Amino-7-(3-methylbenzyl)-6-oxo...)
Affinity DataKd:  1.58E+4nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316317(((2R,3S,4R,5R)-5-(2-Amino-7-(3-nitrobenzyl)-6-oxo-...)
Affinity DataKd:  1.44E+4nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316316(((2R,3S,4R,5R)-5-(2-Amino-7-(naphthalen-2-ylmethyl...)
Affinity DataKd:  9.05E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316315(((2R,3S,4R,5R)-5-(2-Amino-7-(4-fluorobenzyl)-6-oxo...)
Affinity DataKd:  8.22E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316313(((2R,3S,4R,5R)-5-(2-Amino-7-(3-methoxybenzyl)-6-ox...)
Affinity DataKd:  6.60E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316304(((2R,3S,4R,5R)-5-(2-amino-7-methyl-6-oxo-1H-purin-...)
Affinity DataKd:  7.50E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316305(((2R,3S,4R,5R)-5-(2-amino-7-benzyl-6-oxo-1H-purin-...)
Affinity DataKd:  1.32E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316306(((2R,3S,4R,5R)-5-(2-Amino-7-(3-fluorobenzyl)-6-oxo...)
Affinity DataKd:  1.59E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316307(((2R,3S,4R,5R)-5-(2-Amino-7-(4-chlorobenzyl)-6-oxo...)
Affinity DataKd:  1.99E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316308(((2R,3S,4R,5R)-5-(2-Amino-7-(3-chlorobenzyl)-6-oxo...)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316309(((2R,3S,4R,5R)-5-(2-Amino-7-(2-chlorobenzyl)-6-oxo...)
Affinity DataKd:  2.24E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316310(((2R,3S,4R,5R)-5-(2-Amino-7-(2-chloro-5-fluorobenz...)
Affinity DataKd:  3.10E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316311(((2R,3S,4R,5R)-5-(2-Amino-7-(2-fluorobenzyl)-6-oxo...)
Affinity DataKd:  4.39E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316312(((2R,3S,4R,5R)-5-(2-Amino-7-(4-carboxybenzyl)-6-ox...)
Affinity DataKd:  4.59E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50316314(((2R,3S,4R,5R)-5-(2-Amino-6-oxo-7-(3-(trifluoromet...)
Affinity DataKd:  7.56E+3nMAssay Description:Binding affinity to mouse eIF4E expressed in Escherichia coli by fluorescence time-synchronized titration method in presence of KKRYDREFLLGFQFIFAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410170(CHEMBL2079703)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370488(CHEMBL607618)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410173(CHEMBL2079719)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370490(CHEMBL610599)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410172(CHEMBL2079724)
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410171(CHEMBL2079700)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410174(CHEMBL2079702)
Affinity DataIC50: 8.50E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370482(CHEMBL610852)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370491(CHEMBL611110)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165117(2-amino-6-hydroxy-9-[(2R,4S,5R)-5-[(phosphinatooxy...)
Affinity DataIC50: 1.80E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370487(CHEMBL609052)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370481(CHEMBL611113)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370492(CHEMBL607905)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165142(disodium 2-amino-9-[(2R,4S,5R)-5-[({[(carboxylatom...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165127(2-Amino-9-((2R,4S,5R)-5-hydroxymethyl-3,4-diisopro...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165116(tetrasodium ({[(2R,3R,5R)-5-(2-amino-6-hydroxy-9H-...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165118(2-Amino-7-benzyl-9-((2R,4S,5R)-5-hydroxymethyl-3,4...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165119(2-Amino-9-((2R,4S,5R)-5-hydroxymethyl-3,4-diisopro...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410169(CHEMBL2021409)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370493(CHEMBL609636)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165141(disodium 2-amino-9-[(2R,4S,5R)-5-{[({[1-carboxylat...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165134(2-Amino-7-ethyl-9-((2R,4S,5R)-5-hydroxymethyl-3,4-...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370483(CHEMBL607903)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165122(disodium 2-amino-9-[(2R,4S,5R)-5-[({[(2-carboxylat...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370489(CHEMBL607902)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370484(CHEMBL611105)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEukaryotic translation initiation factor 4E(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165135(disodium 2-amino-9-[(2R,4S,5R)-5-[({[(1-carboxylat...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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