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TargetCholecystokinin receptor type A(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM81962(S-L-365,260)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCholecystokinin receptor type A(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM81962(S-L-365,260)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50449787(CHEMBL2062154 | PD-134308)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50449787(CHEMBL2062154 | PD-134308)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472889(CHEMBL415240)
Affinity DataKi:  0.178nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472889(CHEMBL415240)
Affinity DataKi:  0.178nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50345941(9-(2-Methyl-allylamino)-3-p-tolyl-3H-pyrido[3',2':...)
Affinity DataKi:  0.200nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224406(9-(4-chlorophenyl)-2,3-dihydro-3(R)-methyl-1H-pyri...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]9-Dimethylamino-3-(4-methoxy-phenyl)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one from mGluR1 in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472863(CHEMBL333979)
Affinity DataKi:  0.209nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472863(CHEMBL333979)
Affinity DataKi:  0.209nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472878(CHEMBL331872)
Affinity DataKi:  0.224nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472878(CHEMBL331872)
Affinity DataKi:  0.224nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472863(CHEMBL333979)
Affinity DataKi:  0.251nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472863(CHEMBL333979)
Affinity DataKi:  0.251nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472898(CHEMBL332902)
Affinity DataKi:  0.288nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472898(CHEMBL332902)
Affinity DataKi:  0.288nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472855(CHEMBL331468)
Affinity DataKi:  0.295nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472855(CHEMBL331468)
Affinity DataKi:  0.295nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224407(2,3-dihydro-9-(4-methoxyphenyl)-3(R)-methyl-1H-pyr...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]9-Dimethylamino-3-(4-methoxy-phenyl)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one from mGluR1 in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472870(CHEMBL331975)
Affinity DataKi:  0.302nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472870(CHEMBL331975)
Affinity DataKi:  0.302nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472884(CHEMBL121021)
Affinity DataKi:  0.331nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472884(CHEMBL121021)
Affinity DataKi:  0.331nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50449787(CHEMBL2062154 | PD-134308)
Affinity DataKi:  0.355nMAssay Description:Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50449787(CHEMBL2062154 | PD-134308)
Affinity DataKi:  0.355nMAssay Description:Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472854(CHEMBL330977)
Affinity DataKi:  0.372nMAssay Description:Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472854(CHEMBL330977)
Affinity DataKi:  0.372nMAssay Description:Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224391(9-(4-chlorophenyl)-2,3-dihydro-1H-pyrimido[4'',5''...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]9-Dimethylamino-3-(4-methoxy-phenyl)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one from mGluR1 in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50345942(3-(4-Methoxy-phenyl)-9-(2-methyl-allylamino)-3H-py...)
Affinity DataKi:  0.400nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50364723(CHEMBL1951662)
Affinity DataKi:  0.400nMAssay Description:Antagonist activity at rat metabotropic glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472887(CHEMBL330773)
Affinity DataKi:  0.490nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472887(CHEMBL330773)
Affinity DataKi:  0.490nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224395(2,3-dihydro-9-(4-methylphenyl)-1H-pyrimido[4'',5''...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]9-Dimethylamino-3-(4-methoxy-phenyl)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one from mGluR1 in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224392(9-(4-chlorophenyl)-2,3-dihydro-2(S)-methyl-1H-pyri...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]9-Dimethylamino-3-(4-methoxy-phenyl)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one from mGluR1 in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472864(CHEMBL402702)
Affinity DataKi:  0.562nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472864(CHEMBL402702)
Affinity DataKi:  0.562nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472853(CHEMBL331244)
Affinity DataKi:  0.575nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472853(CHEMBL331244)
Affinity DataKi:  0.575nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224400(2,3-dihydro-3(R)-methyl-9-(4-methylphenyl)-1H-pyri...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]9-Dimethylamino-3-(4-methoxy-phenyl)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one from mGluR1 in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50345947(3-(4-Chloro-phenyl)-9-prop-2-ynylamino-3H-pyrido[3...)
Affinity DataKi:  0.600nMAssay Description:Antagonist activity at rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472876(CHEMBL332568)
Affinity DataKi:  0.603nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472876(CHEMBL332568)
Affinity DataKi:  0.603nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472885(CHEMBL118622)
Affinity DataKi:  0.646nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472885(CHEMBL118622)
Affinity DataKi:  0.646nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472871(CHEMBL118954)
Affinity DataKi:  0.661nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472871(CHEMBL118954)
Affinity DataKi:  0.661nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472848(CHEMBL420728)
Affinity DataKi:  0.676nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50472848(CHEMBL420728)
Affinity DataKi:  0.676nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

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