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TargetDelta-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545673(CHEMBL4634079)
Affinity DataKi: <0.169nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046866(CHEMBL3319256)
Affinity DataKi:  0.170nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046866(CHEMBL3319256)
Affinity DataKi:  0.170nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046866(CHEMBL3319256)
Affinity DataKi:  0.220nMAssay Description:Competitive inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells using p-tyramine as substrate by Dixon-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046950(CHEMBL3319244)
Affinity DataKi:  0.260nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046948(CHEMBL3319272)
Affinity DataKi:  0.270nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046878(CHEMBL3319247)
Affinity DataKi:  0.290nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50232425(CHEMBL4061639)
Affinity DataKi:  0.290nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046879(CHEMBL3317469)
Affinity DataKi:  0.300nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046949(CHEMBL3319273)
Affinity DataKi:  0.460nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50232429(CHEMBL4104691)
Affinity DataKi:  0.480nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50232429(CHEMBL4104691)
Affinity DataKi:  0.480nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50232429(CHEMBL4104691)
Affinity DataKi:  0.480nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36717(1,25(OH)2D3)
Affinity DataKi:  0.5nM ΔG°:  -49.3kJ/molepH: 7.5 T: 4°CAssay Description:VDR in vitro ligand-binding assay using human VDR constructed into a yeast expression plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545677(CHEMBL4645508)
Affinity DataKi: <0.510nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50513574(CHEMBL4539722)
Affinity DataKi:  0.570nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50513572(CHEMBL4466571)
Affinity DataKi:  0.570nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046949(CHEMBL3319273)
Affinity DataKi:  0.630nMAssay Description:Competitive inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells using p-tyramine as substrate by Dixon-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046865(CHEMBL3319257)
Affinity DataKi:  0.640nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50513575(CHEMBL4567537)
Affinity DataKi:  0.840nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001092(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001092(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Guinea pig)
D'Annunzio University of Chieti???Pescara

Curated by ChEMBL
LigandPNGBDBM50595851(CHEMBL5192735)
Affinity DataKi:  0.920nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50513573(CHEMBL4449231)
Affinity DataKi:  0.930nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545677(CHEMBL4645508)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bindin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Guinea pig)
D'Annunzio University of Chieti???Pescara

Curated by ChEMBL
LigandPNGBDBM50595850(CHEMBL5188021)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Guinea pig)
D'Annunzio University of Chieti???Pescara

Curated by ChEMBL
LigandPNGBDBM50595847(CHEMBL5199097)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50000335(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  1.80nMAssay Description:In Vitro evaluation for the binding affinity in homogenates of rat brain at Opioid receptor delta 1 by displacing [3H]- DSLETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Guinea pig)
D'Annunzio University of Chieti???Pescara

Curated by ChEMBL
LigandPNGBDBM50399881(CHEMBL2180639)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50398760(CHEMBL2179652)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Guinea pig)
D'Annunzio University of Chieti???Pescara

Curated by ChEMBL
LigandPNGBDBM50595846(CHEMBL5183917)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM19187((2S)-2-[({4-[(3-fluorophenyl)methoxy]phenyl}methyl...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545658(CHEMBL4644543)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bindin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50046871(CHEMBL3319254)
Affinity DataKi:  2.40nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rat)
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001090(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  2.5nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50362540(CHEMBL1941031)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]diprenorphine from human KOPR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50159165((2S,4aR,6aR,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]diprenorphine from human KOPR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Guinea pig)
D'Annunzio University of Chieti???Pescara

Curated by ChEMBL
LigandPNGBDBM50595852(CHEMBL5194818)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Guinea pig)
D'Annunzio University of Chieti???Pescara

Curated by ChEMBL
LigandPNGBDBM50595849(CHEMBL5169404)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545685(CHEMBL4646678)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bindin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545658(CHEMBL4644543)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545678(CHEMBL4636598)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Guinea pig)
D'Annunzio University of Chieti???Pescara

Curated by ChEMBL
LigandPNGBDBM50595853(CHEMBL5177451)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50232426(CHEMBL4089754)
Affinity DataKi:  3.60nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545652(CHEMBL4638667)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545683(CHEMBL4644731)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bindin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545690(CHEMBL4644964)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bindin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50545689(CHEMBL4646687)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bindin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Guinea pig)
D'Annunzio University of Chieti???Pescara

Curated by ChEMBL
LigandPNGBDBM50595848(CHEMBL5179970)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50362539(CHEMBL1941030)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]diprenorphine from human KOPR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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