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TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM10882(6-ethoxy-1,3-benzothiazole-2-sulfonamide | Ethoxzo...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258299(1-({[5-(Aminosulfonyl)-3-(2,3,4,5,6-pentafluorophe...)
Affinity DataKi:  0.880nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM10887(Sulfamate 7 | [(1R,2S,6S,9R)-4,4,11,11-tetramethyl...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258298(1-({[5-(Aminosulfonyl)-3-(3-methoxyphenyl)-1H-indo...)
Affinity DataKi:  0.920nMAssay Description:Inhibition of human recombinant CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258299(1-({[5-(Aminosulfonyl)-3-(2,3,4,5,6-pentafluorophe...)
Affinity DataKi:  0.930nMAssay Description:Inhibition of human recombinant CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258299(1-({[5-(Aminosulfonyl)-3-(2,3,4,5,6-pentafluorophe...)
Affinity DataKi:  0.930nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant carbonic anhydrase Rv3273 by by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258681(1-({[5-(Aminosulfonyl)-3-(4-chlorophenyl)-1H-indol...)
Affinity DataKi:  0.960nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258678(1-({[5-(Aminosulfonyl)-3-(4-fluorophenyl)-1H-indol...)
Affinity DataKi:  0.960nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258716(2,4,6-trimethyl-1-(5-sulfamoyl-3-p-tolyl-1H-indole...)
Affinity DataKi:  0.970nMAssay Description:Inhibition of human recombinant CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258680(1-({[5-(Aminosulfonyl)-3-(3-chlorophenyl)-1H-indol...)
Affinity DataKi:  0.970nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258714(2,4,6-trimethyl-1-(5-sulfamoyl-3-o-tolyl-1H-indole...)
Affinity DataKi:  0.980nMAssay Description:Inhibition of human recombinant CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258679(1-(3-(2-bromophenyl)-5-sulfamoyl-1H-indole-2-carbo...)
Affinity DataKi:  1.01nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258715(1-({[5-(Aminosulfonyl)-3-(3-bromophenyl)-1H-indol-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human recombinant CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258298(1-({[5-(Aminosulfonyl)-3-(3-methoxyphenyl)-1H-indo...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 1(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258680(1-({[5-(Aminosulfonyl)-3-(3-chlorophenyl)-1H-indol...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of human recombinant CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-carbonic anhydrase 1(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258678(1-({[5-(Aminosulfonyl)-3-(4-fluorophenyl)-1H-indol...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant carbonic anhydrase Rv1284 by by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258716(2,4,6-trimethyl-1-(5-sulfamoyl-3-p-tolyl-1H-indole...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35733(sulfonamide deriv., 7a)
Affinity DataKi:  4.70nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetBeta-carbonic anhydrase 1(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258716(2,4,6-trimethyl-1-(5-sulfamoyl-3-p-tolyl-1H-indole...)
Affinity DataKi:  5.10nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant carbonic anhydrase Rv1284 by by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258681(1-({[5-(Aminosulfonyl)-3-(4-chlorophenyl)-1H-indol...)
Affinity DataKi:  5.20nMAssay Description:Inhibition of human recombinant CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35738(sulfonamide deriv., 7f)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35736(sulfonamide deriv., 7d)
Affinity DataKi:  5.40nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35735(sulfonamide deriv., 7c)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
Istanbul University

LigandPNGBDBM35738(sulfonamide deriv., 7f)
Affinity DataKi:  5.90nM ΔG°:  -47.0kJ/moleT: 2°CAssay Description:An SX.18MV-R Applied Photophysics (Oxford, UK) stopped-flow instrument has been used to assay the catalytic/inhibition of various CA isozymes. Phenol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258634(1-({[5-(Aminosulfonyl)-3-(3-methylphenyl)-1H-indol...)
Affinity DataKi:  6nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
Istanbul University

LigandPNGBDBM35742(sulfonamide deriv., 8)
Affinity DataKi:  6.10nM ΔG°:  -46.9kJ/moleT: 2°CAssay Description:An SX.18MV-R Applied Photophysics (Oxford, UK) stopped-flow instrument has been used to assay the catalytic/inhibition of various CA isozymes. Phenol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35742(sulfonamide deriv., 8)
Affinity DataKi:  6.10nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35726(sulfonamide deriv., 5a)
Affinity DataKi:  6.20nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258635(1-({[5-(Aminosulfonyl)-3-(4-methylphenyl)-1H-indol...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258587(1-(([5-(Aminosulfonyl)-3-phenyl-1H-indol-2-yl]carb...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of human recombinant CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258637(1-(3-(3-chlorophenyl)-5-sulfamoyl-1H-indole-2-carb...)
Affinity DataKi:  6.60nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
Istanbul University

LigandPNGBDBM35733(sulfonamide deriv., 7a)
Affinity DataKi:  6.70nM ΔG°:  -46.7kJ/moleT: 2°CAssay Description:An SX.18MV-R Applied Photophysics (Oxford, UK) stopped-flow instrument has been used to assay the catalytic/inhibition of various CA isozymes. Phenol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258636(1-(3-(2-chlorophenyl)-5-sulfamoyl-1H-indole-2-carb...)
Affinity DataKi:  6.70nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
Istanbul University

LigandPNGBDBM35739(sulfonamide deriv., 7g)
Affinity DataKi:  6.80nM ΔG°:  -46.6kJ/moleT: 2°CAssay Description:An SX.18MV-R Applied Photophysics (Oxford, UK) stopped-flow instrument has been used to assay the catalytic/inhibition of various CA isozymes. Phenol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
Istanbul University

LigandPNGBDBM35739(sulfonamide deriv., 7g)
Affinity DataKi:  6.80nM ΔG°:  -46.6kJ/moleT: 2°CAssay Description:An SX.18MV-R Applied Photophysics (Oxford, UK) stopped-flow instrument has been used to assay the catalytic/inhibition of various CA isozymes. Phenol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258714(2,4,6-trimethyl-1-(5-sulfamoyl-3-o-tolyl-1H-indole...)
Affinity DataKi:  6.80nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35734(sulfonamide deriv., 7b)
Affinity DataKi:  6.80nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
Istanbul University

LigandPNGBDBM35727(sulfonamide deriv., 5b)
Affinity DataKi:  6.90nM ΔG°:  -46.6kJ/moleT: 2°CAssay Description:An SX.18MV-R Applied Photophysics (Oxford, UK) stopped-flow instrument has been used to assay the catalytic/inhibition of various CA isozymes. Phenol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258588(1-(3-(2-fluorophenyl)-5-sulfamoyl-1H-indole-2-carb...)
Affinity DataKi:  6.90nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35737(sulfonamide deriv., 7e)
Affinity DataKi:  6.90nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35732(sulfonamide deriv., 6)
Affinity DataKi:  6.90nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35728(sulfonamide deriv., 5c)
Affinity DataKi:  6.90nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM25918(BMC173212 Compound 2n | 2-(hydrazinecarbonyl)-3-(2...)
Affinity DataKi:  7nM ΔG°:  -46.5kJ/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2008
Entry Details Article
PubMed
TargetCarbonic anhydrase 14(Human)
Istanbul University

LigandPNGBDBM25916(BMC173212 Compound 2l | 3-(4-bromophenyl)-2-(hydra...)
Affinity DataKi:  7nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2008
Entry Details Article
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
Istanbul University

LigandPNGBDBM35726(sulfonamide deriv., 5a)
Affinity DataKi:  7nM ΔG°:  -46.5kJ/moleT: 2°CAssay Description:An SX.18MV-R Applied Photophysics (Oxford, UK) stopped-flow instrument has been used to assay the catalytic/inhibition of various CA isozymes. Phenol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35727(sulfonamide deriv., 5b)
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
Istanbul University

LigandPNGBDBM35738(sulfonamide deriv., 7f)
Affinity DataKi:  7.10nM ΔG°:  -46.5kJ/moleT: 2°CAssay Description:An SX.18MV-R Applied Photophysics (Oxford, UK) stopped-flow instrument has been used to assay the catalytic/inhibition of various CA isozymes. Phenol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM35730(cid_694792 | sulfonamide deriv., 5e)
Affinity DataKi:  7.10nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM25904(BMC173212 Compound 1 | 2-(hydrazinecarbonyl)-3-phe...)
Affinity DataKi:  7.20nM ΔG°:  -46.5kJ/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2008
Entry Details Article
PubMed
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