Compile Data Set for Download or QSAR
Found 1503 with Last Name = 'sato' and Initial = 'h'
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Japan Energy Corporation

LigandPNGBDBM719((4R)-N-tert-butyl-3-[(2S,3S)-2-hydroxy-3-[(2R)-2-[...)
Affinity DataKi:  0.0880nM ΔG°:  -59.7kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002099(CHEMBL366965 | Dimethyl-[3-(2-methyl-6H-dibenzo[b,...)
Affinity DataKi:  0.130nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Japan Energy Corporation

LigandPNGBDBM718((4R)-3-[(2S,3S)-3-[(2-ethyl-3-hydroxyphenyl)formam...)
Affinity DataKi:  0.160nM ΔG°:  -58.2kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Japan Energy Corporation

LigandPNGBDBM717((4R)-N-[(2-chlorophenyl)methyl]-3-[(2S,3S)-2-hydro...)
Affinity DataKi:  0.290nM ΔG°:  -56.6kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002087(4-(1-Methyl-piperidin-4-ylidene)-4,9-dihydro-1-thi...)
Affinity DataKi:  0.310nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Japan Energy Corporation

LigandPNGBDBM580((4R)-3-[(2S,3S)-2-hydroxy-3-[(3-hydroxy-2-methylph...)
Affinity DataKi:  0.330nM ΔG°:  -56.3kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002083(2-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  0.480nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002102(2-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  0.630nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Japan Energy Corporation

LigandPNGBDBM579((4R)-N-tert-butyl-3-[(2S,3S)-2-hydroxy-3-[(2R)-2-[...)
Affinity DataKi:  0.740nM ΔG°:  -54.2kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002792(11-[2-(5-Benzylcarbamoyl-benzoimidazol-1-yl)-ethyl...)
Affinity DataKi:  0.910nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Japan Energy Corporation

LigandPNGBDBM712((4R)-N-tert-butyl-3-[(2S,3S)-3-[2-(2,6-dimethylphe...)
Affinity DataKi:  1.40nM ΔG°:  -52.6kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002778(11-[2-(5-Nitro-benzoimidazol-1-yl)-ethylidene]-6,1...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002784(11-[2-(5-Trifluoromethyl-benzoimidazol-1-yl)-ethyl...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Japan Energy Corporation

LigandPNGBDBM715((4R)-N-tert-butyl-3-[(2S,3S)-3-[(2-ethyl-3-hydroxy...)
Affinity DataKi:  2.24nM ΔG°:  -51.4kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002787(11-(2-[1,3]Dioxolo[4',5':4,5]benzo[1,2-d]imidazol-...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002785(11-[2-(5,6-Dimethyl-benzoimidazol-1-yl)-ethylidene...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002796(11-[2-(5-Methoxy-benzoimidazol-1-yl)-ethylidene]-6...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002808(11-[2-(5,6-Dimethoxy-benzoimidazol-1-yl)-ethyliden...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002814(11-[2-(4,5-Dimethyl-benzoimidazol-1-yl)-ethylidene...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002759(5-(2-Benzenesulfonylamino-ethylsulfanyl)-5,11-dihy...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity at TXA2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002759(5-(2-Benzenesulfonylamino-ethylsulfanyl)-5,11-dihy...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002783(11-[2-(4,6-Dimethyl-benzoimidazol-1-yl)-ethylidene...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50164606((2R)-3'-(5-bromothien-2-yl)-2'H-spiro[4-azabicyclo...)
Affinity DataKi:  4nMAssay Description:Inhibition of [125I]alpha-bungarotoxin binding to rat nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50190677((R)-3'-(3-bromobenzo[b]thiophen-5-yl)spiro[1-azabi...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50190686((R)-3'-(2,3-dimethylbenzo[b]thiophen-5-yl)spiro[1-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002820(11-[2-(2-Hydroxy-benzoimidazol-1-yl)-ethylidene]-6...)
Affinity DataKi:  4nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50190696((2S)-3'-(5-bromothien-2-yl)-2'H-spiro[4-azabicyclo...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002095(11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibe...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002103(3-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002085(CHEMBL304185 | [11-(4-Dimethylamino-butylidene)-6,...)
Affinity DataKi:  4.60nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002086(11-(3-Pyrrolidin-1-yl-propylidene)-6,11-dihydro-di...)
Affinity DataKi:  5nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002772(11-[2-(2-Hydroxy-benzoylamino)-ethylsulfanyl]-6,11...)
Affinity DataKi:  5.10nMAssay Description:Inhibition of the thromboxane A2 receptor assayed by binding to guinea pig platelets using [3H]-U-46,619 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002772(11-[2-(2-Hydroxy-benzoylamino)-ethylsulfanyl]-6,11...)
Affinity DataKi:  5.10nMAssay Description:Binding affinity at TXA2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Japan Energy Corporation

LigandPNGBDBM714((4R)-N-tert-butyl-3-[(2S,3S)-2-hydroxy-3-[(3-hydro...)
Affinity DataKi:  5.14nM ΔG°:  -49.2kJ/molepH: 6.0 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Substrates and cleavage fragments...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002093(CHEMBL65699 | [11-(3-Dimethylamino-propylidene)-6,...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002757(11-[2-(Thiophene-2-sulfonylamino)-ethylsulfanyl]-6...)
Affinity DataKi:  5.70nMAssay Description:Compound was tested for its binding affinity at Thromboxane A2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig platelets ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002757(11-[2-(Thiophene-2-sulfonylamino)-ethylsulfanyl]-6...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity at TXA2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002097(11-(4-Dimethylamino-butylidene)-6,11-dihydro-diben...)
Affinity DataKi:  5.80nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002782(11-[2-(5-Chloro-benzoimidazol-1-yl)-ethylidene]-6,...)
Affinity DataKi:  6nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002770(11-[2-(3-Benzyl-thioureido)-ethylsulfanyl]-6,11-di...)
Affinity DataKi:  6.10nMAssay Description:Inhibition of the thromboxane A2 receptor assayed by binding to guinea pig platelets using [3H]-U-46,619 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002818(11-{2-[5-(Hydroxy-phenyl-methyl)-benzoimidazol-1-y...)
Affinity DataKi:  6.10nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002801(11-[2-(5,7-Dimethoxy-benzoimidazol-1-yl)-ethyliden...)
Affinity DataKi:  6.10nMAssay Description:Binding affinity at TXA2/PGH2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002770(11-[2-(3-Benzyl-thioureido)-ethylsulfanyl]-6,11-di...)
Affinity DataKi:  6.10nMAssay Description:Inhibition of the thromboxane A2 receptor assayed by binding to guinea pig platelets using [3H]-U-46,619 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002098(11-(4-Dimethylamino-butylidene)-6,11-dihydro-diben...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002751(11-[2-(2-Phenyl-ethenesulfonylamino)-ethylsulfanyl...)
Affinity DataKi:  6.5nMAssay Description:Binding affinity at TXA2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002751(11-[2-(2-Phenyl-ethenesulfonylamino)-ethylsulfanyl...)
Affinity DataKi:  6.5nMAssay Description:Compound was tested for its binding affinity at Thromboxane A2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig platelets ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002751(11-[2-(2-Phenyl-ethenesulfonylamino)-ethylsulfanyl...)
Affinity DataKi:  6.5nMAssay Description:Compound was tested for its binding affinity at Thromboxane A2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002758(11-(2-Benzenesulfonylamino-ethylsulfanyl)-9-bromo-...)
Affinity DataKi:  6.80nMAssay Description:Inhibition of the thromboxane A2 receptor assayed by binding to guinea pig platelets using [3H]-U-46,619 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50002758(11-(2-Benzenesulfonylamino-ethylsulfanyl)-9-bromo-...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity at TXA2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50040108(11-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-ethylsulfa...)
Affinity DataKi:  6.90nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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