Compile Data Set for Download or QSAR
Found 80 with Last Name = 'sato' and Initial = 'r'
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50245727(CHEMBL4063321)
Affinity DataKi:  121nMAssay Description:Mixed-type inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259790(CHEMBL4101395)
Affinity DataKi:  940nMAssay Description:Mixed-type inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075089(CHEMBL133420 | Sodium; [2-(4-chloro-benzenesulfony...)
Affinity DataIC50:  2.20nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075088(CHEMBL336846 | Sodium; {2-[(4-chloro-benzenesulfon...)
Affinity DataIC50:  3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  10nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075086(CHEMBL341221 | Sodium; [2-(benzenesulfonylamino-me...)
Affinity DataIC50:  13nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075091(CHEMBL131894 | Sodium; 3-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  15nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075077(CHEMBL131497 | Sodium; {2-[(naphthalene-2-sulfonyl...)
Affinity DataIC50:  22nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075082(CHEMBL264516 | Sodium; 2-[(4-chloro-benzenesulfony...)
Affinity DataIC50:  26nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075094(CHEMBL132659 | Sodium; {2-[2-(4-chloro-benzenesulf...)
Affinity DataIC50:  32nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075093(CHEMBL130377 | Sodium; 5-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  36nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50002805((daltroban){4-[2-(4-Chloro-benzenesulfonylamino)-e...)
Affinity DataIC50:  37nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075079(CHEMBL334501 | Sodium; 4-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  39nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  48nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 20...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50245727(CHEMBL4063321)
Affinity DataIC50:  55nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259791(CHEMBL4083406)
Affinity DataIC50:  59nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259788(CHEMBL4071948)
Affinity DataIC50:  65nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075096(CHEMBL336352 | Sodium; 2-[2-(4-chloro-benzenesulfo...)
Affinity DataIC50:  66nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259785(CHEMBL4069806)
Affinity DataIC50:  72nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075076(CHEMBL335043 | Sodium; {2-[(thiophene-2-sulfonylam...)
Affinity DataIC50:  85nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075092(CHEMBL339994 | Sodium; 2-[3-(4-chloro-benzenesulfo...)
Affinity DataIC50:  85nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259789(CHEMBL4091190)
Affinity DataIC50:  115nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075085(CHEMBL131036 | Sodium; {2-[(4-chloro-benzenesulfon...)
Affinity DataIC50:  141nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259783(CHEMBL4104730)
Affinity DataIC50:  151nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075091(CHEMBL131894 | Sodium; 3-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  160nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259794(CHEMBL4096091)
Affinity DataIC50:  180nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259779(CHEMBL4067102)
Affinity DataIC50:  197nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259792(CHEMBL4093669)
Affinity DataIC50:  216nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075090(CHEMBL422441 | Sodium; {2-[(naphthalene-1-sulfonyl...)
Affinity DataIC50:  295nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075085(CHEMBL131036 | Sodium; {2-[(4-chloro-benzenesulfon...)
Affinity DataIC50:  320nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075088(CHEMBL336846 | Sodium; {2-[(4-chloro-benzenesulfon...)
Affinity DataIC50:  360nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075089(CHEMBL133420 | Sodium; [2-(4-chloro-benzenesulfony...)
Affinity DataIC50:  360nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50002805((daltroban){4-[2-(4-Chloro-benzenesulfonylamino)-e...)
Affinity DataIC50:  460nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075081(CHEMBL130045 | Sodium; 2-[4-(4-chloro-benzenesulfo...)
Affinity DataIC50: >479nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075084(CHEMBL130170 | Sodium; {2-[3-(4-chloro-benzenesulf...)
Affinity DataIC50:  513nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259790(CHEMBL4101395)
Affinity DataIC50:  521nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 20...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259785(CHEMBL4069806)
Affinity DataIC50:  621nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 20...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259793(CHEMBL4072968)
Affinity DataIC50:  721nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259789(CHEMBL4091190)
Affinity DataIC50:  737nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 20...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259796(CHEMBL4098929)
Affinity DataIC50:  747nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259796(CHEMBL4098929)
Affinity DataIC50:  768nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 20...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075077(CHEMBL131497 | Sodium; {2-[(naphthalene-2-sulfonyl...)
Affinity DataIC50:  950nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075095(CHEMBL131336 | Sodium; {2-[4-(4-chloro-benzenesulf...)
Affinity DataIC50:  977nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259795(CHEMBL4080503)
Affinity DataIC50:  983nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 20...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075086(CHEMBL341221 | Sodium; [2-(benzenesulfonylamino-me...)
Affinity DataIC50:  1.02E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50259788(CHEMBL4071948)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured after 20...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075080(CHEMBL130460 | Sodium; [2-(cyclohexanesulfonylamin...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075082(CHEMBL264516 | Sodium; 2-[(4-chloro-benzenesulfony...)
Affinity DataIC50:  1.32E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075079(CHEMBL334501 | Sodium; 4-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  1.34E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075083(CHEMBL340073 | Sodium; {2-[(pentane-1-sulfonylamin...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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