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TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266433(CHEMBL445427 | N-(2-{5-Methoxy-2-[(2,3-dihydro-1H-...)
Affinity DataKi:  0.00100nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266405(CHEMBL457128 | N-(3-(3-methoxyphenyl)-3-(naphthale...)
Affinity DataKi:  0.110nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50240952((4-Methoxy-6,7-dihydro-5H-dibenzo[a,c]cyclohepten-...)
Affinity DataKi:  0.160nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50114704(CHEMBL33549 | N-(2-(5-methoxy-2-(3-methoxybenzyl)b...)
Affinity DataKi:  0.25nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50240440(4-P-PDOT | CHEMBL285718 | N-(4-Phenyl-1,2,3,4-tetr...)
Affinity DataKi:  0.460nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50086001(CHEMBL274438 | N-[2-(11-Methoxy-6,7-dihydro-5H-ben...)
Affinity DataKi:  0.5nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266354(CHEMBL514280 | N-(2-((1R,3R)-7-methoxy-3-phenyl-1,...)
Affinity DataKi:  0.900nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266430(CHEMBL514415 | N-(2-{5-Methoxy-2-[(2,3-dihydro-1H-...)
Affinity DataKi:  1.10nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50240952((4-Methoxy-6,7-dihydro-5H-dibenzo[a,c]cyclohepten-...)
Affinity DataKi:  1.40nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50241105((E)-N-[3-(3-methoxyphenyl)-3-phenyl-2-propenyl]ace...)
Affinity DataKi:  2.5nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266434(CHEMBL515856 | N-(2-{5-Methoxy-2-[(5-methoxy-2,3-d...)
Affinity DataKi:  5.80nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266434(CHEMBL515856 | N-(2-{5-Methoxy-2-[(5-methoxy-2,3-d...)
Affinity DataKi:  7.10nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50295871(CHEMBL552002 | N-[2-(5-Methoxy-2-{[(4-methoxypheny...)
Affinity DataKi:  8nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266431(CHEMBL457138 | N-(2-{5-Methoxy-2-[(2,3-dihydro-1H-...)
Affinity DataKi:  8nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50240442(CHEMBL33185 | N-((1-(4-chlorobenzyl)-4-methoxy-1H-...)
Affinity DataKi:  9nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50295871(CHEMBL552002 | N-[2-(5-Methoxy-2-{[(4-methoxypheny...)
Affinity DataKi:  9nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266408(CHEMBL508552 | N-(2-{5-Methoxy-2-[(2-methyl-2,3-di...)
Affinity DataKi:  14nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266432(CHEMBL457352 | N-(2-{5-Methoxy-2-[2,3-dihydro-1H-i...)
Affinity DataKi:  14.5nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266450(CHEMBL514427 | N-(2-{5-Methoxy-2-[(5-methyl-2,3-di...)
Affinity DataKi:  15nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266452(CHEMBL514904 | N-{2-[5-Methoxy-2-(pyrrolidin-1ylme...)
Affinity DataKi:  25nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266453(CHEMBL513933 | N-(2-{5-Methoxy-2-[(6-nitro-2,3-dih...)
Affinity DataKi:  26nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50114704(CHEMBL33549 | N-(2-(5-methoxy-2-(3-methoxybenzyl)b...)
Affinity DataKi:  27nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266451(CHEMBL457807 | N-(2-{2-[(5-Bromo-2,3-dihydro-1H-in...)
Affinity DataKi:  30nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266432(CHEMBL457352 | N-(2-{5-Methoxy-2-[2,3-dihydro-1H-i...)
Affinity DataKi:  38nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266431(CHEMBL457138 | N-(2-{5-Methoxy-2-[(2,3-dihydro-1H-...)
Affinity DataKi:  41nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266450(CHEMBL514427 | N-(2-{5-Methoxy-2-[(5-methyl-2,3-di...)
Affinity DataKi:  41nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50240440(4-P-PDOT | CHEMBL285718 | N-(4-Phenyl-1,2,3,4-tetr...)
Affinity DataKi:  59nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50295870(CHEMBL563847 | N-{2-(5-Methoxy-2-({[methyl[4-(trif...)
Affinity DataKi:  63nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266406(CHEMBL514413 | N-[2-(9-Methoxy-13a,14-dihydro-6H,1...)
Affinity DataKi:  65nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50086001(CHEMBL274438 | N-[2-(11-Methoxy-6,7-dihydro-5H-ben...)
Affinity DataKi:  66nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266451(CHEMBL457807 | N-(2-{2-[(5-Bromo-2,3-dihydro-1H-in...)
Affinity DataKi:  85nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266454(CHEMBL456505 | N-(2-{2-[(6-Amino-2,3-dihydro-1H-in...)
Affinity DataKi:  110nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50295870(CHEMBL563847 | N-{2-(5-Methoxy-2-({[methyl[4-(trif...)
Affinity DataKi:  111nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266430(CHEMBL514415 | N-(2-{5-Methoxy-2-[(2,3-dihydro-1H-...)
Affinity DataKi:  114nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266454(CHEMBL456505 | N-(2-{2-[(6-Amino-2,3-dihydro-1H-in...)
Affinity DataKi:  118nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266452(CHEMBL514904 | N-{2-[5-Methoxy-2-(pyrrolidin-1ylme...)
Affinity DataKi:  121nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266405(CHEMBL457128 | N-(3-(3-methoxyphenyl)-3-(naphthale...)
Affinity DataKi:  132nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266408(CHEMBL508552 | N-(2-{5-Methoxy-2-[(2-methyl-2,3-di...)
Affinity DataKi:  148nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50241105((E)-N-[3-(3-methoxyphenyl)-3-phenyl-2-propenyl]ace...)
Affinity DataKi:  230nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266453(CHEMBL513933 | N-(2-{5-Methoxy-2-[(6-nitro-2,3-dih...)
Affinity DataKi:  309nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266406(CHEMBL514413 | N-[2-(9-Methoxy-13a,14-dihydro-6H,1...)
Affinity DataKi:  320nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266407(CHEMBL515696 | N-[2-(2,9-Dimethoxy-13a,14-dihydro-...)
Affinity DataKi:  410nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266354(CHEMBL514280 | N-(2-((1R,3R)-7-methoxy-3-phenyl-1,...)
Affinity DataKi:  797nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50273283(CHEMBL455909 | N-[2-(13a,14-Dihydro-6H,13H-pyrazin...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50240442(CHEMBL33185 | N-((1-(4-chlorobenzyl)-4-methoxy-1H-...)
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266433(CHEMBL445427 | N-(2-{5-Methoxy-2-[(2,3-dihydro-1H-...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50273283(CHEMBL455909 | N-[2-(13a,14-Dihydro-6H,13H-pyrazin...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266407(CHEMBL515696 | N-[2-(2,9-Dimethoxy-13a,14-dihydro-...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAngiotensin-converting enzyme(Human)
Ranbaxy Laboratories

Curated by ChEMBL
LigandPNGBDBM50367254(ENALAPRILAT)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetMelatonin receptor type 1A(Human)
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50295869(CHEMBL556908 | N-[2-(8-Methoxy-2-methyl-1,2,3,4-te...)
Affinity DataIC50:  3.14nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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