Report error Found 434 with Last Name = 'spadari' and Initial = 's'
Affinity DataKi: 5nM IC50: 13nMAssay Description:Recombinant HSV TKs were assayed in reaction mixture containing substrate [3H-methyl]TdR and test compounds. After reaction was stopped, the radioact...More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
Affinity DataKi: 30nM ΔG°: -44.7kJ/mole IC50: 150nMpH: 7.5 T: 37°CAssay Description:Recombinant HSV TKs were assayed in reaction mixture containing substrate [3H-methyl]TdR and test compounds. After reaction was stopped, the radioact...More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity of the compound towards HSV-1 thymidine kinase was determinedMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V179DMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution Y181IMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 93nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution L1001More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution L1001More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution L1001More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution Y188LMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair