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TargetTyrosine-protein kinase Lyn(Human)
Osaka Prefecture University

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human LynMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Osaka Prefecture University

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
Osaka Prefecture University

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of FynMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50: 20nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Osaka Prefecture University

Curated by ChEMBL
LigandPNGBDBM4078(Elagic Acid | CHEMBL6246 | 6,7,13,14-tetrahydroxy-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of GST-fused human recombinant CK2alpha expressed in Escherichia coli HMS174 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetNeutrophil elastase(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50080264(FR-901277 | 1N-[21-benzyl-29-[(Z)-ethylidene]-13,1...)
Affinity DataIC50: 180nMAssay Description:Evaluated for the inhibition of Human Leukocyte Elastase (HLE) enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50488029((S)-METHYL-IMIDACLOPRID)
Affinity DataIC50: 190nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50488030((R,S)-METHYL-IMIDACLOPRID)
Affinity DataIC50: 210nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Osaka Prefecture University

Curated by ChEMBL
LigandPNGBDBM11319(IQA | 2-{8-oxo-1,9-diazatetracyclo[8.7.0.0^{2,7}.0...)
Affinity DataIC50: 390nMAssay Description:Inhibition of GST-fused human recombinant CK2alpha expressed in Escherichia coli HMS174 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Osaka Prefecture University

Curated by ChEMBL
LigandPNGBDBM7458(Naringenin, 18 | 5,7-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataIC50: 800nMAssay Description:Inhibition of GST-fused human recombinant CK2alpha expressed in Escherichia coli HMS174 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
Osaka Prefecture University

Curated by ChEMBL
LigandPNGBDBM11323(CHEMBL177820 | 4,5,6,7-tetrabromo-1H-1,2,3-benzotr...)
Affinity DataIC50: 900nMAssay Description:Inhibition of GST-fused human recombinant CK2alpha expressed in Escherichia coli HMS174 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50488028((R)-METHYL-IMIDACLOPRID)
Affinity DataIC50: 950nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50143314(CHEMBL298826 | (+)-Epibatidine | 2-(6-Chloro-pyrid...)
Affinity DataIC50: 1.34E+3nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Osaka Prefecture University

Curated by ChEMBL
LigandPNGBDBM11318(1,3,8-trihydroxy-6-methylanthra-9,10-quinone | CHE...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST-fused human recombinant CK2alpha expressed in Escherichia coli HMS174 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50143320(2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]hept...)
Affinity DataIC50: 2.79E+3nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataIC50: 1.19E+4nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Osaka Prefecture University

Curated by ChEMBL
LigandPNGBDBM11324(CHEMBL375530 | (2R,3R,4S,5R)-2-(5,6-dichloro-1H-1,...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of GST-fused human recombinant CK2alpha expressed in Escherichia coli HMS174 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM82068(Nicotine-D salicylate | CHEMBL9732 | Nicotine-L sa...)
Affinity DataIC50: 4.22E+5nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed