Compile Data Set for Download or QSAR
Report error Found 358 with Last Name = 'taglialatela-scafati' and Initial = 'o'
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataEC50:  200nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29078(cyclopropanolamide, 13a | racemic | cyclopropanola...)
Affinity DataEC50:  1.90E+3nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29079(cyclopropanolamide, 12a | racemic | cyclopropanola...)
Affinity DataEC50:  50nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataEC50:  3.65E+3nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29081(cyclopropanolamide, 13b | racemic | cyclopropanola...)
Affinity DataEC50:  3.70E+3nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29082(cyclopropanolamide, 12b | racemic | cyclopropanola...)
Affinity DataEC50:  60nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29083(Palmidrol | Impulsin | MimyX | Palmityoletanolamid...)
Affinity DataEC50: >1.00E+4nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29084(racemic | cyclopropanolamide, rac-10c)
Affinity DataEC50:  2.64E+4nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29085(cyclopropanolamide, rac-9c)
Affinity DataEC50:  40nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  20nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29078(cyclopropanolamide, 13a | racemic | cyclopropanola...)
Affinity DataEC50:  610nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29087(cyclopropanolamide, 14a)
Affinity DataEC50:  2.40E+3nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29088(cyclopropanolamide, 11a)
Affinity DataEC50:  47nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29079(cyclopropanolamide, 12a | racemic | cyclopropanola...)
Affinity DataEC50:  23nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29081(cyclopropanolamide, 13b | racemic | cyclopropanola...)
Affinity DataEC50:  150nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29091(cyclopropanolamide, 14b)
Affinity DataEC50:  180nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29082(cyclopropanolamide, 12b | racemic | cyclopropanola...)
Affinity DataEC50:  13nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29093(cyclopropanolamide, 11b)
Affinity DataEC50:  19nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  565nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB1 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluorescence as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  73nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB2 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  1.61E+4nMAssay Description:Agonist activity at recombinant rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  7.30E+3nMAssay Description:Agonist activity at recombinant rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at recombinant rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  75nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB1 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  4.78E+3nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB2 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  200nMAssay Description:Agonist activity at recombinant rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  6.20E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluorescence as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  180nMAssay Description:Agonist activity at recombinant rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  5.30E+3nMAssay Description:Agonist activity at recombinant rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456756(CHEMBL4214981)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456758(CHEMBL1631518)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456759(CHEMBL4215902)
Affinity DataEC50:  1.15E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456757(CHEMBL4209008)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456760(CHEMBL4205263)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456761(CHEMBL4213753)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456762(CHEMBL4215072)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456763(CHEMBL4210989)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456765(CHEMBL1915188)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456766(CHEMBL4209967)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456764(CHEMBL4218752)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456769(CHEMBL4211797)
Affinity DataEC50:  1.10E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM217379(CDDO-Me, 2)
Affinity DataEC50:  60nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456770(CHEMBL4208824)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456767(CHEMBL4211445)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456755(CHEMBL4212101)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50456768(CHEMBL4211885)
Affinity DataEC50:  2.45E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50463445(CHEMBL4238545)
Affinity DataEC50:  490nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 358 total ) | Next | Last >>
Jump to: