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LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataIC50: 3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataIC50: 3.30nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 uM in LLCPKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataKi:  4nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50: 9.5nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 uM in LLCPKI cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50: 9.5nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50002692(1-((2R,4S,5S)-4-Azido-5-hydroxymethyl-tetrahydro-f...)
Affinity DataEC50:  10nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataIC50: 10nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044905((10,13-Dimethyl-17-octyl-2,3,4,7,8,9,10,11,12,13,1...)
Affinity DataEC50:  20nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044913(Heptadeca-9,12-dienoic acid 5-(5-methyl-2,4-dioxo-...)
Affinity DataEC50:  20nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataEC50:  33nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044911(Heptadeca-9,12,15-trienoic acid 5-(5-methyl-2,4-di...)
Affinity DataEC50:  40nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044910(Phosphoric acid bis-[5-(5-methyl-2,4-dioxo-3,4-dih...)
Affinity DataEC50:  50nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50013111(2',3'-didehydro-3'-deoxythymidine | 1-(5-Hydroxyme...)
Affinity DataEC50:  50nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044906(Phosphoric acid 8-(10,13-dimethyl-3-vinyloxy-2,3,4...)
Affinity DataEC50:  50nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044907(Hexadecanoic acid 5-(5-methyl-2,4-dioxo-3,4-dihydr...)
Affinity DataEC50:  80nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152981((2S,4R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  100nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataKi:  100nMAssay Description:Displacement of ATP from protein kinase C (PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
LigandPNGBDBM50228839(CHEMBL415414)
Affinity DataKi:  170nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152975((2S,4R)-4-Methoxy-2-(2-pyridin-2-yl-ethylthiocarba...)
Affinity DataEC50:  200nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044908(Phosphoric acid hexadecyl ester 5-(5-methyl-2,4-di...)
Affinity DataEC50:  200nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152972((2S,4R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  230nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50228839(CHEMBL415414)
Affinity DataIC50: 300nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataIC50: 300nMAssay Description:Inhibition of protein kinase C (PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152972((2S,4R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  430nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152975((2S,4R)-4-Methoxy-2-(2-pyridin-2-yl-ethylthiocarba...)
Affinity DataEC50:  470nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152981((2S,4R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  480nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152976((3S,5R)-4-Methoxy-pyrrolidine-1,2-dicarboxylic aci...)
Affinity DataEC50:  570nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152979((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  640nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152973((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  810nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataEC50:  850nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152979((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  890nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152977((3S,5R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  1.10E+3nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50228846(CHEMBL265876)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
LigandPNGBDBM50228847(CHEMBL407100)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
LigandPNGBDBM50228838(CHEMBL428973)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152980((3S,5R)-2-([1,4'']Bipiperidinyl-1''-carbonyl)-4-me...)
Affinity DataEC50:  1.20E+3nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152978((3S,5R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  1.30E+3nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152976((3S,5R)-4-Methoxy-pyrrolidine-1,2-dicarboxylic aci...)
Affinity DataEC50:  1.50E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152973((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  1.80E+3nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152982((2S,4R)-4-Methoxy-pyrrolidine-1,2-dicarboxylic aci...)
Affinity DataEC50:  1.80E+3nMAssay Description:Effective concentration for human Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50228841(CHEMBL351282)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
LigandPNGBDBM50011236(Isoquinoline-5-sulfonic acid (2-amino-ethyl)-amide...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152980((3S,5R)-2-([1,4'']Bipiperidinyl-1''-carbonyl)-4-me...)
Affinity DataEC50:  2.20E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152977((3S,5R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  2.30E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152978((3S,5R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  2.80E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50216682(cid_3542 | 1-(5-Isoquinolinesulfonyl)-2-methylpipe...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
LigandPNGBDBM50216682(cid_3542 | 1-(5-Isoquinolinesulfonyl)-2-methylpipe...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
LigandPNGBDBM15203(Isoquinoline-5-sulfonic acid piperazin-1 ylamide |...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
LigandPNGBDBM50216682(cid_3542 | 1-(5-Isoquinolinesulfonyl)-2-methylpipe...)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of ATP from protein kinase C (PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
LigandPNGBDBM50216682(cid_3542 | 1-(5-Isoquinolinesulfonyl)-2-methylpipe...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of protein kinase C (PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2019
Entry Details Article
PubMed
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