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TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50322229(4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methy...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50050467(1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperi...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003068(CHEMBL3234537)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50050467(1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperi...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50322229(4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methy...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003066(CHEMBL3234536)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003074(CHEMBL3234544)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003068(CHEMBL3234537)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003063(CHEMBL3234237)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003065(CHEMBL3234522)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003073(CHEMBL3234543)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003066(CHEMBL3234536)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003071(CHEMBL3234541)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  244nMAssay Description:Binding affinity to sigma2 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003070(CHEMBL3234539)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003064(CHEMBL1503220)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003072(CHEMBL3234542)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003073(CHEMBL3234543)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003071(CHEMBL3234541)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003069(CHEMBL3234538)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003069(CHEMBL3234538)
Affinity DataKi:  880nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003063(CHEMBL3234237)
Affinity DataKi:  1.16E+3nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  1.22E+3nMAssay Description:Binding affinity to alpha2C receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003064(CHEMBL1503220)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  3.26E+3nMAssay Description:Binding affinity to alpha1D receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003070(CHEMBL3234539)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  3.41E+3nMAssay Description:Binding affinity to DAT receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H1 receptor(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  3.56E+3nMAssay Description:Binding affinity to H1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003074(CHEMBL3234544)
Affinity DataKi:  4.10E+3nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003065(CHEMBL3234522)
Affinity DataKi:  9.20E+3nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003072(CHEMBL3234542)
Affinity DataKi:  2.10E+4nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003075(CHEMBL3234545)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]methylspiperone from human D3 receptor expressed in HEK293 cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50003075(CHEMBL3234545)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]methylspiperone from human D2L receptor expressed in HEK cell membrane after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30026(triazolopyridazine, 18)
Affinity DataIC50:  1.5nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30024(triazolothiadiazine, 10)
Affinity DataIC50:  3nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30023(Racemic | cid_44142103 | triazolothiadiazine, 9)
Affinity DataIC50:  3.40nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30038(triazolothiadiazine, 32)
Affinity DataIC50:  3.80nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Heike firefly)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM50352641(CHEMBL1733803)
Affinity DataIC50:  5nMAssay Description:Inhibition of fire fly luciferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30021(triazolothiadiazine, 7)
Affinity DataIC50:  6.10nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30019(BMCL181297 Compound 5F | triazolothiadiazine, 5)
Affinity DataIC50:  6.70nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30048(triazolothiadiazine, 42)
Affinity DataIC50:  6.70nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30047(triazolothiadiazine, 41)
Affinity DataIC50:  7.10nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30025(triazolopyridazine, 17)
Affinity DataIC50:  7.30nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30043(triazolothiadiazine, 37)
Affinity DataIC50:  8.60nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30037(triazolothiadiazine, 31)
Affinity DataIC50:  9.80nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30022(triazolothiadiazine, 8)
Affinity DataIC50:  11nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30042(triazolothiadiazine, 36)
Affinity DataIC50:  11nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
National Human Genome Research Institute

LigandPNGBDBM30032(triazolothiadiazine, 26)
Affinity DataIC50:  11nMpH: 7.2 T: 22°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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