Compile Data Set for Download or QSAR
Report error Found 216 with Last Name = 'torisu' and Initial = 'k'
TargetProstaglandin D2 receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152512({1-[4-(7-Fluoro-4-methyl-3,4-dihydro-2H-benzo[1,4]...)
Affinity DataIC50: 0.810nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing human Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152515({2-Methyl-1-[4-(4-methyl-3,4-dihydro-2H-benzo[1,4]...)
Affinity DataIC50: 1.20nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing human Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50095207([6-(4-Benzhydryl-pyrazol-1-ylmethyl)-7,8-dihydro-n...)
Affinity DataIC50: 8nMAssay Description:Compound was tested for its binding affinity against Prostaglandin I2 receptor using conventional ligand assay by the displacement of [3H]-iloprost f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin D2 receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152510({2-Methyl-1-[4-(4-methyl-3,4-dihydro-2H-benzo[1,4]...)
Affinity DataIC50: 10nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing human Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284372({5-[2-(N',N'-Diphenyl-hydrazinocarbonyl)-ethyl]-5,...)
Affinity DataIC50: 10nMAssay Description:Compound was tested for prostacyclin (PGI-2) binding by displacement of [3H]iloprost from human platelets using conventional ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284377({5-[2-(4-Benzhydryl-pyrazol-1-yl)-ethyl]-5,6,7,8-t...)
Affinity DataIC50: 18nMAssay Description:Compound was tested for its binding affinity against Prostaglandin I2 receptor using conventional ligand assay by the displacement of [3H]-iloprost f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284370([6-(N',N'-Diphenyl-hydrazinocarbonylmethyl)-5,6,7,...)
Affinity DataIC50: 20nMAssay Description:Compound was tested for prostacyclin (PGI-2) binding by displacement of [3H]iloprost from human platelets using conventional ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM23954(CHEMBL494 | ILOPROST | 5-[(2E,3aS,4R,5R,6aS)-5-hyd...)
Affinity DataIC50: 27nMAssay Description:Prostaglandin I2 receptor binding by displacement of [3H]iloprost from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM23954(CHEMBL494 | ILOPROST | 5-[(2E,3aS,4R,5R,6aS)-5-hyd...)
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin D2 receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152508({1-[4-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethoxy)-b...)
Affinity DataIC50: 30nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing human Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152509({1-[4-(2,3-Dihydro-benzofuran-2-ylmethoxy)-benzoyl...)
Affinity DataIC50: 30nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing human Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152514({1-[4-(Chroman-2-ylmethoxy)-benzoyl]-2-methyl-1H-i...)
Affinity DataIC50: 30nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing human Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284378([6-(4-Benzhydryl-pyrazol-1-ylmethyl)-5,6,7,8-tetra...)
Affinity DataIC50: 40nMAssay Description:Compound was tested for its binding affinity against Prostaglandin I2 receptor using conventional ligand assay by the displacement of [3H]-iloprost f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152506({2-Methyl-1-[4-(2-phenoxy-ethoxy)-benzoyl]-1H-indo...)
Affinity DataIC50: 50nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing mouse Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152516({1-[4-(Benzo[1,3]dioxol-2-ylmethoxy)-benzoyl]-2-me...)
Affinity DataIC50: 50nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing human Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152513([2-Methyl-1-(4-phenethyloxy-benzoyl)-1H-indol-4-yl...)
Affinity DataIC50: 120nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing mouse Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284366((6-{2-[(E)-Benzhydryloxyimino]-butyl}-5,6,7,8-tetr...)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50095205([6-(2-Benzhydryloxyimino-pentyl)-5,6,7,8-tetrahydr...)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284371([5-(2-Benzhydrylideneaminooxy-ethyl)-5,6,7,8-tetra...)
Affinity DataIC50: 210nMAssay Description:Compound was tested for prostacyclin (PGI-2) binding by displacement of [3H]iloprost from human platelets using conventional ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284367(((S)-6-{2-[(E)-Benzhydryloxyimino]-propyl}-5,6,7,8...)
Affinity DataIC50: 220nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin D2 receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152506({2-Methyl-1-[4-(2-phenoxy-ethoxy)-benzoyl]-1H-indo...)
Affinity DataIC50: 250nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing human Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152518({1-[4-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethoxy)-b...)
Affinity DataIC50: 270nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing human Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152507([1-(4-Butoxy-benzoyl)-2-methyl-1H-indol-4-yl]-acet...)
Affinity DataIC50: 300nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing mouse Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284363(((R)-6-{2-[(E)-Benzhydryloxyimino]-propyl}-5,6,7,8...)
Affinity DataIC50: 380nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284374([5-(3-Benzhydryloxy-propyl)-5,6,7,8-tetrahydro-nap...)
Affinity DataIC50: 460nMAssay Description:Compound was tested for prostacyclin (PGI-2) binding by displacement of [3H]iloprost from human platelets using conventional ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284355([5-(3-Benzhydryloxyimino-propyl)-5,6,7,8-tetrahydr...)
Affinity DataIC50: 600nMAssay Description:Prostaglandin I2 receptor binding by displacement of [3H]iloprost from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284355([5-(3-Benzhydryloxyimino-propyl)-5,6,7,8-tetrahydr...)
Affinity DataIC50: 600nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284360([6-(2-Benzhydryloxyimino-ethyl)-5,6,7,8-tetrahydro...)
Affinity DataIC50: 650nMAssay Description:Prostaglandin I2 receptor binding by displacement of [3H]iloprost from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284360([6-(2-Benzhydryloxyimino-ethyl)-5,6,7,8-tetrahydro...)
Affinity DataIC50: 650nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50150972(4-[1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indo...)
Affinity DataIC50: 910nMAssay Description:Inhibition of mouse Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50152511([1-(4-Benzyloxy-benzoyl)-2-methyl-1H-indol-4-yl]-a...)
Affinity DataIC50: 1.30E+3nMAssay Description:Effect on the increase in cAMP formation induced by PGD-2 in the presence of bovine serum albumin in CHO cells expressing mouse Prostaglandin D2 rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50101853((13E,15S)-11alpha,15-dihydroxy-9-oxoprost-13-en-1-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50150974(3-[1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indo...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of mouse Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50150973([1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indol-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of mouse Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284376({5-[2-(4-Benzhydryl-pyrazol-1-yl)-ethyl]-7,8-dihyd...)
Affinity DataIC50: 2.00E+3nMAssay Description:Compound was tested for its binding affinity against Prostaglandin I2 receptor using conventional ligand assay by the displacement of [3H]-iloprost f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284365((5-{3-[(E)-Benzhydryloxyimino]-hexyl}-5,6,7,8-tetr...)
Affinity DataIC50: 2.10E+3nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284363(((R)-6-{2-[(E)-Benzhydryloxyimino]-propyl}-5,6,7,8...)
Affinity DataIC50: 2.20E+3nMAssay Description:Displacement of [3H]iloprost from Prostaglandin I2 receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284368((6-Benzhydrylideneaminooxymethyl-5,6,7,8-tetrahydr...)
Affinity DataIC50: 2.40E+3nMAssay Description:Compound was tested for prostacyclin (PGI-2) binding by displacement of [3H]iloprost from human platelets using conventional ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50150968([1-(3-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indol-...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of mouse Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50150975([1-(4-Butoxy-benzoyl)-2,5-dimethyl-1H-indol-3-yl]-...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of mouse Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284353([6-((Z)-5,5-Diphenyl-pent-2-enyl)-5,6,7,8-tetrahyd...)
Affinity DataIC50: 3.00E+3nMAssay Description:Prostaglandin I2 receptor binding by displacement of [3H]iloprost from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50047491(Sodium; (E)-2-methyl-3-(4-pyridin-3-ylmethyl-pheny...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against Thromboxane A2 synthase in human platelet microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284358([6-((E)-5,5-Diphenyl-pent-2-enyl)-5,6,7,8-tetrahyd...)
Affinity DataIC50: 3.10E+3nMAssay Description:Prostaglandin I2 receptor binding by displacement of [3H]iloprost from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284357([3-(4-Benzhydryloxyimino-butyl)-phenoxy]-acetic ac...)
Affinity DataIC50: 3.90E+3nMAssay Description:Prostaglandin I2 receptor binding by displacement of [3H]iloprost from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50150966([1-(4-Butoxy-benzoyl)-2-methyl-1H-indol-3-yl]-acet...)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of mouse Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50150966([1-(4-Butoxy-benzoyl)-2-methyl-1H-indol-3-yl]-acet...)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of mouse Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50150967(1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indole-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of mouse Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284369([5-(4-Benzhydryloxy-butyl)-5,6,7,8-tetrahydro-naph...)
Affinity DataIC50: 4.20E+3nMAssay Description:Compound was tested for prostacyclin (PGI-2) binding by displacement of [3H]iloprost from human platelets using conventional ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin D2 receptor(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50150976(5-[1-(4-Butoxy-benzoyl)-5-methoxy-2-methyl-1H-indo...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of mouse Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284361([6-((E)-4-Hydroxy-5-phenyl-pent-2-enyl)-5,6,7,8-te...)
Affinity DataIC50: 4.90E+3nMAssay Description:Prostaglandin I2 receptor binding by displacement of [3H]iloprost from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Displayed 1 to 50 (of 216 total ) | Next | Last >>
Jump to: