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TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50382166(CHEMBL2023825)
Affinity DataIC50: 0.270nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50382169(CHEMBL2023824)
Affinity DataIC50: 2.90nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50401861(CHEMBL2204672)
Affinity DataIC50: 2.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50382165(CHEMBL2023823)
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50401862(CHEMBL2204668)
Affinity DataIC50: 5.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50401857(CHEMBL2204679)
Affinity DataIC50: 12.3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50382168(CHEMBL2023827)
Affinity DataIC50: 12.4nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50401859(CHEMBL2204677)
Affinity DataIC50: 36.1nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50401858(CHEMBL2204678)
Affinity DataIC50: 42nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50401860(CHEMBL2204675)
Affinity DataIC50: 48.1nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50382167(CHEMBL2023826)
Affinity DataIC50: 63.3nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50382164(CHEMBL2023828)
Affinity DataIC50: 100nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50078575(CHEMBL3414957)
Affinity DataIC50: 135nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human Jurkat cell membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423058(CHEMBL244471)
Affinity DataIC50: 282nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423056(CHEMBL243002)
Affinity DataIC50: 1.18E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423059(CHEMBL244472)
Affinity DataIC50: 1.41E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423057(CHEMBL242573)
Affinity DataIC50: 1.51E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423062(CHEMBL242786)
Affinity DataIC50: 1.59E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423063(CHEMBL396501)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423061(CHEMBL243003)
Affinity DataIC50: 2.04E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423055(CHEMBL244957)
Affinity DataIC50: 2.19E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM85065(CAS_117946-91-5 | NSC_122162 | Luzindole)
Affinity DataIC50: 2.46E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423064(CHEMBL244263)
Affinity DataIC50: 4.68E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423060(CHEMBL241928)
Affinity DataIC50: 5.13E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50423065(CHEMBL242806)
Affinity DataIC50: 6.17E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50034220(n-hexadecylphosphocholine | CHEMBL125 | hexadecyl ...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051809(Hexadecyl[2-(N-Methylmorpholinio)ethyl]phosphate |...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051810((N-methylpiperidino)ethanol 2-(hexadecyloxy)ethyl ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50411361(CHEMBL396991)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051808((N-methylmorpholino)ethanol dodecyl phosphonate | ...)
Affinity DataIC50: 2.90E+5nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051815((N-methylpiperidino)ethanol 2-(tetradecyloxy)ethyl...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051811((N-methylmorpholino)ethanol 2-(tetradecycloxy)ethy...)
Affinity DataIC50: 3.80E+5nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051816(hexadecyl 2-(1-methylpiperidinium-1-yl)ethyl phosp...)
Affinity DataIC50: 4.60E+5nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051813((N-methylpiperidino)ethanol tetradecyl phosphonate...)
Affinity DataIC50: 4.90E+5nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051806((N-methylmorpholino)ethanol dodecyl phosphonate | ...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051814((N-methylmorpholino)ethanol 2-(dodecyloxy)ethyl ph...)
Affinity DataIC50: 6.10E+5nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051807((N-methylmorpholino)ethanol 2-(hexadecyloxy)ethyl ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051806((N-methylmorpholino)ethanol dodecyl phosphonate | ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051810((N-methylpiperidino)ethanol 2-(hexadecyloxy)ethyl ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50034220(n-hexadecylphosphocholine | CHEMBL125 | hexadecyl ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051812((N-methylpiperidino)ethanol dodecyl phosphonate | ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051811((N-methylmorpholino)ethanol 2-(tetradecycloxy)ethy...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051814((N-methylmorpholino)ethanol 2-(dodecyloxy)ethyl ph...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051808((N-methylmorpholino)ethanol dodecyl phosphonate | ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetM-phase inducer phosphatase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051807((N-methylmorpholino)ethanol 2-(hexadecyloxy)ethyl ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 25 (Cdc25) phosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051815((N-methylpiperidino)ethanol 2-(tetradecyloxy)ethyl...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051812((N-methylpiperidino)ethanol dodecyl phosphonate | ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051809(Hexadecyl[2-(N-Methylmorpholinio)ethyl]phosphate |...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051813((N-methylpiperidino)ethanol tetradecyl phosphonate...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50051816(hexadecyl 2-(1-methylpiperidinium-1-yl)ethyl phosp...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Cell division cycle 2 (cdc2) kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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