Found 218 with Last Name = 'vultaggio' and Initial = 's' TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Inhibitory activity against beta-glucosidase of sweet almondMore data for this Ligand-Target Pair
3D Structure (crystal)TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataKi: 4.30E+4nMAssay Description:Non-competitive inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using H3K4me1 peptide as substrate preincubated fo...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataKi: 4.84E+4nMAssay Description:Competitive inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using H3K4me1 peptide as substrate preincubated for 15...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.130nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.130nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.170nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.210nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.340nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.340nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 0.380nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.380nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using biotinylated H3K4me1 peptide as substrate preincubated for 2...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 6.70nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 7.80nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of human HDAC extracted from human HeLa cellsMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
