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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118378(CHEMBL3612622)
Affinity DataIC50: 0.123nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118375(CHEMBL3612511)
Affinity DataIC50: 0.166nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118344(CHEMBL3612513)
Affinity DataIC50: 0.177nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118334(CHEMBL3612507)
Affinity DataIC50: 0.212nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118376(CHEMBL3612512)
Affinity DataIC50: 0.374nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM25036(CHEMBL393525 | N'-[(1E)-{6-bromoimidazo[1,2-a]pyri...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118224(CHEMBL3612503)
Affinity DataIC50: 0.762nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118372(CHEMBL3612508)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118377(CHEMBL3612515)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM25036(CHEMBL393525 | N'-[(1E)-{6-bromoimidazo[1,2-a]pyri...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant human CDK9/cyclin-T1 using H-YSPTSPSYSPTSPSYSPTSPS-KKKK-OH as substrate after 90 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118345(CHEMBL3612514)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27633(N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino]ethyl]ph...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27634(N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino]ethyl]ph...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118236(CHEMBL3612504)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27628(5-bromo-N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino]...)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27627(N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino]ethyl]ph...)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27637(N-{3-[(1S)-1-[(5-bromopyridin-3-yl)amino]ethyl]phe...)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM25036(CHEMBL393525 | N'-[(1E)-{6-bromoimidazo[1,2-a]pyri...)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118241(CHEMBL3612505)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27631(3-chloro-N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino...)
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27632(N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino]ethyl]ph...)
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27630(N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino]ethyl]ph...)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118259(CHEMBL3612506)
Affinity DataIC50: 10nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118373(CHEMBL3612509)
Affinity DataIC50: 10nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27639(N-{3-[(1S)-1-{[6-(4-hydroxy-3-methoxyphenyl)pyrazi...)
Affinity DataIC50: 11nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27626(N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino]ethyl]ph...)
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118374(CHEMBL3612510)
Affinity DataIC50: 15nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118370(CHEMBL3612501)
Affinity DataIC50: 21nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27619(N-[3-(1-{[6-(4-hydroxy-3-methoxyphenyl)pyrazin-2-y...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118212(CHEMBL3612498)
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human CDK9/cyclin-T1 using H-YSPTSPSYSPTSPSYSPTSPS-KKKK-OH as substrate after 90 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50041659((S)-3-[(S)-2-[2-tert-Butoxycarbonylamino-3-(1H-ind...)
Affinity DataIC50: 28nMAssay Description:In vitro binding for half maximal inhibition of [125I]- Bolton-Hunter-CCK-8 in guinea pig pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118370(CHEMBL3612501)
Affinity DataIC50: 29nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118346(CHEMBL3612482)
Affinity DataIC50: 32nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118212(CHEMBL3612498)
Affinity DataIC50: 33nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50520948(CHEMBL4443524)
Affinity DataIC50: 38nMAssay Description:Inhibition of hERG expressed in CHO cells Qpatch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27625(N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino]ethyl]ph...)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27629(N-{3-[(1S)-1-[(6-chloropyrazin-2-yl)amino]ethyl]ph...)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed in 384 well Optiplates (Packard) using an Alphascreen Protein Tyrosine Kinase kit. Inhibitors were added to the mixtures...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118334(CHEMBL3612507)
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant human CDK9/cyclin-T1 using H-YSPTSPSYSPTSPSYSPTSPS-KKKK-OH as substrate after 90 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118370(CHEMBL3612501)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant human CDK9/cyclin-T1 using H-YSPTSPSYSPTSPSYSPTSPS-KKKK-OH as substrate after 90 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118371(CHEMBL3612502)
Affinity DataIC50: 81nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118357(CHEMBL3612489)
Affinity DataIC50: 90nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118346(CHEMBL3612482)
Affinity DataIC50: 96nMAssay Description:Inhibition of recombinant human CDK9/cyclin-T1 using H-YSPTSPSYSPTSPSYSPTSPS-KKKK-OH as substrate after 90 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118371(CHEMBL3612502)
Affinity DataIC50: 97nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118352(CHEMBL3612485)
Affinity DataIC50: 154nMAssay Description:Inhibition of FLT3 (unknown origin) using biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2 as substrate after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118378(CHEMBL3612622)
Affinity DataIC50: 164nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118371(CHEMBL3612502)
Affinity DataIC50: 174nMAssay Description:Inhibition of recombinant human CDK9/cyclin-T1 using H-YSPTSPSYSPTSPSYSPTSPS-KKKK-OH as substrate after 90 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118345(CHEMBL3612514)
Affinity DataIC50: 194nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118334(CHEMBL3612507)
Affinity DataIC50: 198nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118357(CHEMBL3612489)
Affinity DataIC50: 201nMAssay Description:Inhibition of recombinant human CDK9/cyclin-T1 using H-YSPTSPSYSPTSPSYSPTSPS-KKKK-OH as substrate after 90 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50118344(CHEMBL3612513)
Affinity DataIC50: 203nMAssay Description:Inhibition of recombinant human CDK9/cyclin-T1 using H-YSPTSPSYSPTSPSYSPTSPS-KKKK-OH as substrate after 90 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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