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Report error Found 2296 with Last Name = 'xia' and Initial = 's'
TargetHemagglutinin(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Peking University

Curated by ChEMBL
LigandPNGBDBM50529725(CHEMBL4569515)
Affinity DataKd:  1.56E+4nMAssay Description:Binding affinity to recombinant Influenza A virus (A/California/04/2009 (H1N1)) hemagglutinin by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648167(CHEMBL5598046)
Affinity DataKd:  2.93E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase, H3 lysine-79 specific(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50460738(CHEMBL4225123)
Affinity DataKd:  4.78E+3nMAssay Description:Binding affinity to recombinant human His6-SUMO tagged DOT1L (1 to 416 residues) expressed in Escherichia coli BL21(DE3) by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648157(CHEMBL5598164)
Affinity DataKd:  2.03E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein ENL(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50617569(CHEMBL5418436)
Affinity DataKd:  30nMAssay Description:Binding affinity to C-terminal 6-His tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50583996(CHEMBL4554938 | US12318398, Compound XMU-MP-1)
Affinity DataKd:  22nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1)
Beijing Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50459313(CHEMBL4206744)
Affinity DataEC50:  3.63E+3nMAssay Description:Inhibition of HIV1 envelope glycoprotein-mediated cell-cell fusion between HL2/3 cells stably expressing HIV Gag, Env, Tat, Rev and Nef proteins and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247361(CHEMBL4077534)
Affinity DataEC50:  2.70E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human HEK293 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMed
TargetProtein ENL(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50576674(CHEMBL4850575)
Affinity DataKd:  1.41E+4nMAssay Description:Binding affinity to ENL YEATS domain (unknown origin) assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573836(CHEMBL4861375)
Affinity DataKd:  2.81E+3nMAssay Description:Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  120nMAssay Description:Binding affinity to BPTF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648174(CHEMBL5598541)
Affinity DataKd:  1.11E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase TAO2(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50583996(CHEMBL4554938 | US12318398, Compound XMU-MP-1)
Affinity DataKd:  100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50527569(CHEMBL4440098 | US11427593, Compound ZB-BD-216)
Affinity DataKd:  2.10nMAssay Description:Binding affinity to human partial length BRDT bromodomain 2 isoform b (K250 to E382 residues) expressed in bacterial expression system by bromoscan a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50617561(CHEMBL5438748)
Affinity DataKd:  17nMAssay Description:Binding affinity to C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648160(CHEMBL5590507)
Affinity DataKd:  370nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50605865(CHEMBL5202311)
Affinity DataKd:  9.25E+3nMAssay Description:Binding affinity to human recombinant VHL assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetAurora kinase B(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50583996(CHEMBL4554938 | US12318398, Compound XMU-MP-1)
Affinity DataKd:  40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247349(CHEMBL4072005)
Affinity DataEC50:  2.00E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human A549 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648173(CHEMBL5597324)
Affinity DataKd:  2.06E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50552663(CHEMBL4746871)
Affinity DataKd:  2.70E+3nMAssay Description:Binding affinity to recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells by SPR a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648154(CHEMBL5590641)
Affinity DataKd: >5.00E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAurora kinase A(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50583996(CHEMBL4554938 | US12318398, Compound XMU-MP-1)
Affinity DataKd:  13nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase 24(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50583996(CHEMBL4554938 | US12318398, Compound XMU-MP-1)
Affinity DataKd:  18nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50583996(CHEMBL4554938 | US12318398, Compound XMU-MP-1)
Affinity DataKd:  77nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648165(CHEMBL5596868)
Affinity DataKd:  1.31E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein ENL(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50617567(CHEMBL5395794)
Affinity DataKd:  119nMAssay Description:Binding affinity to 3xFLAG-HA-tagged wild-type human ENL YEATS domain assessed as dissociation constant by ITC titration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648163(CHEMBL5597013)
Affinity DataKd:  3.10E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648188(CHEMBL5597140)
Affinity DataKd:  87nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573851(CHEMBL4872422)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to human BPTF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648181(CHEMBL5597295)
Affinity DataKd:  140nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648180(CHEMBL5589996)
Affinity DataKd:  130nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648182(CHEMBL5596391)
Affinity DataKd:  270nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648172(CHEMBL5597735)
Affinity DataKd:  3.19E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648156(CHEMBL5596339)
Affinity DataKd:  1.22E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50583996(CHEMBL4554938 | US12318398, Compound XMU-MP-1)
Affinity DataKd:  11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648155(CHEMBL5598139)
Affinity DataKd:  920nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHemagglutinin(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Peking University

Curated by ChEMBL
LigandPNGBDBM50529726(CHEMBL4464620)
Affinity DataKd:  3.60E+4nMAssay Description:Binding affinity to recombinant Influenza A virus (A/California/04/2009 (H1N1)) hemagglutinin by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHemagglutinin(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
Peking University

Curated by ChEMBL
LigandPNGBDBM50605865(CHEMBL5202311)
Affinity DataKd:  3.18E+3nMAssay Description:Binding affinity to recombinant influenza A hemagglutinin assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648178(CHEMBL5596259)
Affinity DataKd:  3.93E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPhosphatidylinositol 5-phosphate 4-kinase type-2 gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50583996(CHEMBL4554938 | US12318398, Compound XMU-MP-1)
Affinity DataKd:  34nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50527569(CHEMBL4440098 | US11427593, Compound ZB-BD-216)
Affinity DataKd:  3nMAssay Description:Binding affinity to human partial length BRD4 bromodomain 1 long isoform (N44 to E168 residues) expressed in bacterial expression system by BROMOscan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  200nMAssay Description:Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247359(CHEMBL4062783)
Affinity DataEC50:  3.10E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human HEK293 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMed
LigandPNGBDBM50339886((S)-3-(1-(2-amino-6-(4-fluorophenyl)pyrimidin-4-yl...)
Affinity DataEC50:  100nMAssay Description:Inhibition of FAAH in rat RBL cell assessed as conversion of [3H]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50339871((S)-3-(1-(4-(5-chlorothiophen-2-yl)pyrimidin-2-yl)...)
Affinity DataEC50:  3nMAssay Description:Inhibition of FAAH in human T84 cell assessed as conversion of [3H]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM8465(CGS 27023 | CHEMBL514138 | hydroxamate analogue 1 ...)
Affinity DatapH: 7.5 T: 2°CAssay Description:The recombinant Agg-1 proteins pretreated with the various concentrations of the compound for 10 to 15 min. The reaction was initiated by addition of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2008
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50583996(CHEMBL4554938 | US12318398, Compound XMU-MP-1)
Affinity DataKd:  24nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
LigandPNGBDBM50339873((S)-3-(1-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-yl)...)
Affinity DataEC50:  80nMAssay Description:Inhibition of FAAH in rat RBL cell assessed as conversion of [3H]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50648168(CHEMBL5597112)
Affinity DataKd:  4.88E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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