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TargetAcetylcholinesterase(Electric eel)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50234829(CHEMBL4100760)
Affinity DataKi:  12nMAssay Description:Mixed-type inhibition of Electrophorus electricus AChE pretreated for 15 mins followed by varying levels of acetylthiocholine iodide substrate additi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDiphosphomevalonate decarboxylase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287714((3R)-3-(fluoromethyl)-3-hydroxy-5-{[(phosphonatoox...)
Affinity DataKi:  37nMAssay Description:Compound was evaluated for its inhibitory activity against Mevalonate 5-pyrophosphate decarboxylaseMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50067364(CHEMBL3401816)
Affinity DataKi:  63nMAssay Description:Inhibition of Mcl-1 (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50067458(CHEMBL3401801)
Affinity DataKi:  66nMAssay Description:Inhibition of Mcl-1 (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50067363(CHEMBL3401817)
Affinity DataKi:  74nMAssay Description:Inhibition of Mcl-1 (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067355(CHEMBL3401825)
Affinity DataKi:  80nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50067460(CHEMBL3401800)
Affinity DataKi:  86nMAssay Description:Inhibition of Mcl-1 (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50067354(CHEMBL3401826)
Affinity DataKi:  250nMAssay Description:Inhibition of Mcl-1 (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067363(CHEMBL3401817)
Affinity DataKi:  360nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetApoptosis regulator Bcl-2(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067458(CHEMBL3401801)
Affinity DataKi:  390nMAssay Description:Inhibition of Bcl-2 (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067469(CHEMBL3401796)
Affinity DataKi:  410nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067460(CHEMBL3401800)
Affinity DataKi:  420nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067451(CHEMBL3401804)
Affinity DataKi:  450nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067464(CHEMBL3401798)
Affinity DataKi:  460nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067461(CHEMBL3401799)
Affinity DataKi:  460nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067458(CHEMBL3401801)
Affinity DataKi:  470nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067454(CHEMBL3401802)
Affinity DataKi:  470nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetApoptosis regulator Bcl-2(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067364(CHEMBL3401816)
Affinity DataKi:  490nMAssay Description:Inhibition of Bcl-2 (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067450(CHEMBL3401805)
Affinity DataKi:  510nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067466(CHEMBL3401793)
Affinity DataKi:  520nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetApoptosis regulator Bcl-2(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067460(CHEMBL3401800)
Affinity DataKi:  540nMAssay Description:Inhibition of Bcl-2 (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067449(CHEMBL3401806)
Affinity DataKi:  540nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067452(CHEMBL3401803)
Affinity DataKi:  540nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKi:  620nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067475(CHEMBL3400166)
Affinity DataKi:  630nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetApoptosis regulator Bcl-2(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067354(CHEMBL3401826)
Affinity DataKi:  660nMAssay Description:Inhibition of Bcl-2 (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067371(CHEMBL3401809)
Affinity DataKi:  660nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067358(CHEMBL3401822)
Affinity DataKi:  680nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067365(CHEMBL3401815)
Affinity DataKi:  700nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067364(CHEMBL3401816)
Affinity DataKi:  710nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067354(CHEMBL3401826)
Affinity DataKi:  720nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067356(CHEMBL3401824)
Affinity DataKi:  720nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067465(CHEMBL3401794)
Affinity DataKi:  730nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDiphosphomevalonate decarboxylase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287713([methyl(2-{[(phosphonatooxy)phosphinato]oxy}ethyl)...)
Affinity DataKi:  750nMAssay Description:Compound was evaluated for its inhibitory activity against Mevalonate 5-pyrophosphate decarboxylaseMore data for this Ligand-Target Pair
In DepthDetails Article

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067357(CHEMBL3401823)
Affinity DataKi:  750nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067359(CHEMBL3401821)
Affinity DataKi:  750nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067369(CHEMBL3401811)
Affinity DataKi:  800nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067367(CHEMBL3401813)
Affinity DataKi:  850nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067368(CHEMBL3401812)
Affinity DataKi:  870nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067361(CHEMBL3401819)
Affinity DataKi:  900nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067468(CHEMBL3401797)
Affinity DataKi:  950nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067362(CHEMBL3401818)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067370(CHEMBL3401810)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067448(CHEMBL3401807)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067476(CHEMBL3401795)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067372(CHEMBL3401808)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067360(CHEMBL3401820)
Affinity DataKi:  5.60E+3nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-like protein 1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50067366(CHEMBL3401814)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of Bcl-XL (unknown origin) using 5-FAM-Bid-BH3 as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50482966(CHEMBL1270818)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK2/cyclin AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetCytochrome P450 2C9(Human)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50352206(CHEMBL1825089)
Affinity DataIC50:  1nMAssay Description:Inhibition of CYP2C9 using a fluorescent probe 7-methoxy-4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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