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TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50308541(7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3...)
Affinity DataKi:  0.0190nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50308541(7-Methoxy-2-oxo-8-pentyloxy-1,2-dihydroquinoline-3...)
Affinity DataKi:  0.0190nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50353091(CHEMBL1822944)
Affinity DataKi:  0.0200nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50353091(CHEMBL1822944)
Affinity DataKi:  0.0200nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073061(CHEMBL3410832)
Affinity DataKi:  0.0210nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073061(CHEMBL3410832)
Affinity DataKi:  0.0210nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073068(CHEMBL3410813)
Affinity DataKi:  0.0260nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073068(CHEMBL3410813)
Affinity DataKi:  0.0260nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50072968(CHEMBL3410818)
Affinity DataKi:  0.0530nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50072968(CHEMBL3410818)
Affinity DataKi:  0.0530nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50353090(CHEMBL1822943)
Affinity DataKi:  0.0849nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50353090(CHEMBL1822943)
Affinity DataKi:  0.0850nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073005(CHEMBL3410729)
Affinity DataKi:  0.0869nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073005(CHEMBL3410729)
Affinity DataKi:  0.0870nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073000(CHEMBL3410826)
Affinity DataKi:  0.0879nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073000(CHEMBL3410826)
Affinity DataKi:  0.0880nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50072967(CHEMBL3410817)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50072967(CHEMBL3410817)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073001(CHEMBL3410827)
Affinity DataKi:  0.110nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073001(CHEMBL3410827)
Affinity DataKi:  0.110nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Human)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50035105(1'-{4-[1-(4-fluorophenyl)-1H-3-indolyl]butyl}spiro...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity to sigma-2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50353092(CHEMBL1822945)
Affinity DataKi:  0.130nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50353092(CHEMBL1822945)
Affinity DataKi:  0.130nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50312599(CHEMBL1093735 | N-Cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50312599(CHEMBL1093735 | N-Cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cells pretreated for 10 mins measured after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073059(CHEMBL3410831)
Affinity DataKi:  0.180nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073059(CHEMBL3410831)
Affinity DataKi:  0.180nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50355892(CHEMBL1910035)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cells pretreated for 10 mins measured after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50312597(CHEMBL1093377 | N-Cyclohexyl-4-[(2,4-dichloropheny...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]p-Cl-DPDPE from rat delta opioid receptor expressed in rat C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50072992(CHEMBL3410819)
Affinity DataKi:  0.220nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50072992(CHEMBL3410819)
Affinity DataKi:  0.220nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50242582(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Human)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50216056((N-[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity to sigma-2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50072965(CHEMBL3410815)
Affinity DataKi:  0.330nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50072965(CHEMBL3410815)
Affinity DataKi:  0.330nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Human)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50048866(1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to sigma-2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562182(CHEMBL4744466)
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Human)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50248937(CHEMBL4062168 | US10981896, Compound 15)
Affinity DataKi:  0.390nMAssay Description:Inhibition of His6-tagged MELK catalytic domain (1 to 340 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells using Bcl-GL as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073066(CHEMBL3410811)
Affinity DataKi:  0.440nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50073066(CHEMBL3410811)
Affinity DataKi:  0.440nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Human)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50248946(CHEMBL1908392 | US10981896, Compound 16)
Affinity DataKi:  0.470nMAssay Description:Inhibition of His6-tagged MELK catalytic domain (1 to 340 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells using Bcl-GL as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50422834(CHEMBL204387)
Affinity DataKi:  0.480nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50422834(CHEMBL204387)
Affinity DataKi:  0.480nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Material Medica, Chinese Academy of Sciences

US Patent
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.5nM ΔG°:  -54.0kJ/mole IC50:  2.56nMT: 30°CAssay Description:Different concentrations (10^−5 M-10^−11 M) of the compound of the invention and corresponding isotope receptor ligand as well as recepto...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50427413(CHEMBL2326297)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]CP-55,940 from CB2 receptor (unknown origin) after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  0.600nMAssay Description:Antagonist activity at cloned human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  0.600nMAssay Description:Antagonist activity at rat spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Human)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50248938(CHEMBL4089284 | US10981896, Compound 21)
Affinity DataKi:  0.680nMAssay Description:Inhibition of His6-tagged MELK catalytic domain (1 to 340 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells using Bcl-GL as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]CP-55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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