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TargetVasopressin V2 receptor(Human)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1b receptor(Human)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.590nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Human)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.780nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Rat)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Rat)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi:  1.33nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Rat)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  1.45nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139906(CHEMBL414991 | DPhe-His-Leu-Leu-Arg-Glu-Val-Leu-Gl...)
Affinity DataKi:  2nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139920(Ac-(Glu-Aib-Glu-Lys)-Leu-Arg-Lys-Leu-Cha-Asp-Ile-I...)
Affinity DataKi:  3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139907(Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Cha-Asp-Ile-I...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139905(Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Phe-Asp-Ile-I...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  6.36nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Human)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  9.42nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Human)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139915(Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Nle-Asp-Ile-I...)
Affinity DataKi:  36.7nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139909(Ac-(Glu-Ala-Lys-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi:  44.8nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139901(Ac-(Glu-Ala-His-Lys)-Leu-Lys-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi:  45.1nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139904(Ac-(Glu-Ala-Leu-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi:  48.9nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139908(Ac-(Glu-Ala-His-Lys)-Asn-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi:  50nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139910(Ac-(Glu-Ala-His-Lys)-Leu-Ala-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi:  70.9nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139913(Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Phe-Asp-Ile-I...)
Affinity DataKi:  81nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139914(Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi:  130nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  150nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Rat)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi:  325nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Rat)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  524nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139912(Ac-(Glu-Ala-Phe-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139911(Ac-(Glu-Dap-His-Lys)-Asn-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139902(Ac-(Glu-Ala-His-Lys)-Asp-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139900(Ac-(Glu-Asp-His-Lys)-Asn-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139903(Ac-(Glu-Ala-His-Lys)-Dab-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139919(Ac-(Glu-Ala-His-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139916(Ac-(Glu-Ala-His-Lys)-Gln-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139918(Ac-(Glu-Ala-His-Lys)-Leu-Gly-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50139917(Ac-(Glu-Ala-Asp-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-I...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at human CRF1 receptor (CRFR1) on HeLA cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1b receptor(Human)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106478(CHEMBL443591 | FGGFTGARKCARKC)
Affinity DataIC50:  0.122nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  0.177nMAssay Description:Inhibition of human MMP-9 by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106477(CHEMBL265801 | FGGFTGARKSARKLADE | Phe-GGFTGARKSAR...)
Affinity DataIC50:  0.286nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106479(CHEMBL384755 | FGGFTGARKSARK | H-FGGFTGARKSARK-NH2...)
Affinity DataIC50:  0.353nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  0.422nMAssay Description:Inhibition of human MMP-2 by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106471(CHEMBL406718 | FGGFTGARKCARKC)
Affinity DataIC50:  0.471nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106480(CHEMBL437915 | FGGFTGARKSARKL)
Affinity DataIC50:  0.520nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289727(4-Hydroxy-piperidine-1-carboxylic acid ((S)-1-{[(S...)
Affinity DataIC50:  0.680nMAssay Description:In vitro renin inhibitory effect was evaluated for plasma renin activity (PRA) of human plasma, Expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106469(CHEMBL269029 | FGGFTCARKCARK | cyclo[Cys6,Cys10]N/...)
Affinity DataIC50:  0.833nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106470(CHEMBL442113 | FGGFTCARKCARK)
Affinity DataIC50:  3.03nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106476(CHEMBL435511 | FGGFTGCRKSCRK)
Affinity DataIC50:  3.04nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50549085(CHEMBL4752810)
Affinity DataIC50:  4nMAssay Description:Inhibition of histidine-tagged Pseudomonas aeruginosa LpxC (1-303) expressed in Escherichia coli BL21 (DE3) using UDP-3-O-(R-3-hydroxydecanoyl)-N-ace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50549082(CHEMBL4763699)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of histidine-tagged Pseudomonas aeruginosa LpxC (1-303) expressed in Escherichia coli BL21 (DE3) using UDP-3-O-(R-3-hydroxydecanoyl)-N-ace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50549081(CHEMBL4779477)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of histidine-tagged Pseudomonas aeruginosa LpxC (1-303) expressed in Escherichia coli BL21 (DE3) using UDP-3-O-(R-3-hydroxydecanoyl)-N-ace...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106468(CHEMBL424934 | FGGFTGCRKSARKC)
Affinity DataIC50:  4.97nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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