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TargetVasopressin V1b receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85096(CAS_105077 | NSC_105077 | d(CH2)5Tyr(Me)AVP)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)
Affinity DataKi:  0.380nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM35709(YM-35278)
Affinity DataKi:  0.400nM ΔG°:  -53.3kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50013775((oxytocin-OT) cyclo[Cys-Tyr-Ile-Gln-Asn-Cys]-Pro-L...)
Affinity DataKi:  0.890nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  1.09nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85096(CAS_105077 | NSC_105077 | d(CH2)5Tyr(Me)AVP)
Affinity DataKi:  1.79nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85094(CAS_62357-86-2 | NSC_64759 | dDAVP)
Affinity DataKi:  1.93nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)
Affinity DataKi:  3.04nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  3.23nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35683(5H-1-benzazepin-5-ylidene acetamide, 1k)
Affinity DataKi:  3.40nM ΔG°:  -48.0kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35673(5H-1-benzazepin-5-ylidene acetamide, 1a | BMC16952...)
Affinity DataKi:  4.80nM ΔG°:  -47.2kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35673(5H-1-benzazepin-5-ylidene acetamide, 1a | BMC16952...)
Affinity DataKi:  4.80nM ΔG°:  -47.2kJ/mole EC50:  1.80nMpH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35677(5H-1-benzazepin-5-ylidene acetamide, 1e)
Affinity DataKi:  5.60nM ΔG°:  -46.8kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35700(5H-1-benzazepin-5-ylidene acetamide, 10g)
Affinity DataKi:  6nM ΔG°:  -46.6kJ/mole EC50: >1.00E+4nMpH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  6.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35681(5H-1-benzazepin-5-ylidene acetamide, 1i)
Affinity DataKi:  7.40nM ΔG°:  -46.1kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85094(CAS_62357-86-2 | NSC_64759 | dDAVP)
Affinity DataKi:  7.94nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35699(5H-1-benzazepin-5-ylidene acetamide, 10f)
Affinity DataKi:  9.10nM ΔG°:  -45.6kJ/mole EC50: >1.00E+4nMpH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35695(5H-1-benzazepin-5-ylidene acetamide, 10b)
Affinity DataKi:  9.20nM ΔG°:  -45.6kJ/mole EC50:  61.9nMpH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35666(BMC173130 Compound 1t | benzazepinelidene acetamid...)
Affinity DataKi:  9.70nM ΔG°:  -45.4kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35666(BMC173130 Compound 1t | benzazepinelidene acetamid...)
Affinity DataKi:  9.70nM ΔG°:  -45.4kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35679(5H-1-benzazepin-5-ylidene acetamide, 1g)
Affinity DataKi:  10nM ΔG°:  -45.4kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35706(5H-1-benzazepin-5-ylidene acetamide, 10m)
Affinity DataKi:  11nM ΔG°:  -45.1kJ/mole EC50:  646nMpH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35684(5H-1-benzazepin-5-ylidene acetamide, 1l)
Affinity DataKi:  11nM ΔG°:  -45.1kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35694(5H-1-benzazepin-5-ylidene acetamide, 1w)
Affinity DataKi:  11nM ΔG°:  -45.1kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35680(5H-1-benzazepin-5-ylidene acetamide, 1h)
Affinity DataKi:  11nM ΔG°:  -45.1kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35686(5H-1-benzazepin-5-ylidene acetamide, 1n)
Affinity DataKi:  11nM ΔG°:  -45.1kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35698(5H-1-benzazepin-5-ylidene acetamide, 10e)
Affinity DataKi:  11nM ΔG°:  -45.1kJ/mole EC50: >1.00E+4nMpH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35685(5H-1-benzazepin-5-ylidene acetamide, 1m)
Affinity DataKi:  11nM ΔG°:  -45.1kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35687(5H-1-benzazepin-5-ylidene acetamide, 1o)
Affinity DataKi:  12nM ΔG°:  -44.9kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Astellas Pharma

LigandPNGBDBM35669(benzazepinelidene acetamide derivative, 1d)
Affinity DataKi:  13nM ΔG°:  -44.7kJ/molepH: 7.4 T: 23°CAssay Description:Chinese hamster ovary (CHO) cells stably expressing human V1a receptors. Cells were washed with phosphate buffered saline, and then collected in ice-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35669(benzazepinelidene acetamide derivative, 1d)
Affinity DataKi:  13nM ΔG°:  -44.7kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Astellas Pharma

LigandPNGBDBM35691(5H-1-benzazepin-5-ylidene acetamide, 1s)
Affinity DataKi:  13nM ΔG°:  -45.0kJ/moleT: 25°CAssay Description:Chinese hamster ovary (CHO) cells stably expressing human V1a receptors. Cells were washed with phosphate buffered saline, and then collected in ice-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35703(5H-1-benzazepin-5-ylidene acetamide, 10j | racemat...)
Affinity DataKi:  14nM ΔG°:  -44.5kJ/mole EC50:  1.25nMpH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35705(5H-1-benzazepin-5-ylidene acetamide, 10l)
Affinity DataKi:  14nM ΔG°:  -44.5kJ/mole EC50:  104nMpH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35672(benzazepinelidene acetamide derivative, 1g)
Affinity DataKi:  14nM ΔG°:  -44.5kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35671(benzazepinelidene acetamide derivative, 1f)
Affinity DataKi:  14nM ΔG°:  -44.5kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35682(5H-1-benzazepin-5-ylidene acetamide, 1j)
Affinity DataKi:  14nM ΔG°:  -44.5kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50029644(CHEMBL296908 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinol...)
Affinity DataKi:  14.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Human)
Astellas Pharma

LigandPNGBDBM35675(5H-1-benzazepin-5-ylidene acetamide, 1c)
Affinity DataKi:  15nM ΔG°:  -44.7kJ/moleT: 25°CAssay Description:Chinese hamster ovary (CHO) cells stably expressing human V1a receptors. Cells were washed with phosphate buffered saline, and then collected in ice-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35704(5H-1-benzazepin-5-ylidene acetamide, 10k)
Affinity DataKi:  16nM ΔG°:  -44.2kJ/mole EC50:  1.10E+3nMpH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35670(benzazepinelidene acetamide derivative, 1e)
Affinity DataKi:  16nM ΔG°:  -44.2kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35678(5H-1-benzazepin-5-ylidene acetamide, 1f)
Affinity DataKi:  16nM ΔG°:  -44.2kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Astellas Pharma

LigandPNGBDBM35671(benzazepinelidene acetamide derivative, 1f)
Affinity DataKi:  17nM ΔG°:  -44.0kJ/molepH: 7.4 T: 23°CAssay Description:Chinese hamster ovary (CHO) cells stably expressing human V1a receptors. Cells were washed with phosphate buffered saline, and then collected in ice-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Astellas Pharma

LigandPNGBDBM35691(5H-1-benzazepin-5-ylidene acetamide, 1s)
Affinity DataKi:  18nM ΔG°:  -43.9kJ/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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