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Report error Found 6459 with Last Name = 'yu' and Initial = 'k'
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31918(carbohydrazide derivative, 3a)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31919(carbohydrazide derivative, 3b)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31920(carbohydrazide derivative, 3c)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31921(carbohydrazide derivative, 3d)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31922(carbohydrazide derivative, 3e)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31923(carbohydrazide derivative, 3f)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31924(carbohydrazide derivative, 3g)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31929(carbohydrazide derivative, 3l)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31932(carbohydrazide derivative, 3o)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31933(carbohydrazide derivative, 3p)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31935(carbohydrazide derivative, 3r)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31936(1,3-thiazolidin-5-ylidene derivative, 2)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31937(1,3-thiazolidin-5-ylidene derivative, 4a)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31938(1,3-thiazolidin-5-ylidene derivative, 4b)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31939(1,3-thiazolidin-5-ylidene derivative, 4c)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31940(1,3-thiazolidin-5-ylidene derivative, 4d)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31941(1,3-thiazolidin-5-ylidene derivative, 4e)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31942(1,3-thiazolidin-5-ylidene derivative, 4f)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31943(1,3-thiazolidin-5-ylidene derivative, 4g)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31944(1,3-thiazolidin-5-ylidene derivative, 4h)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31945(1,3-thiazolidin-5-ylidene derivative, 4i)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31946(1,3-thiazolidin-5-ylidene derivative, 4j)
Affinity DatapH: 8.0 T: 2°CAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31947(1,3-thiazolidin-5-ylidene derivative, 4k)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31948(1,3-thiazolidin-5-ylidene derivative, 4l)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31949(1,3-thiazolidin-5-ylidene derivative, 4m)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31950(1,3-thiazolidin-5-ylidene derivative, 4n)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31951(1,3-thiazolidin-5-ylidene derivative, 4o)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31952(1,3-thiazolidin-5-ylidene derivative, 4p)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31953(1,3-thiazolidin-5-ylidene derivative, 4q)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31954(1,3-thiazolidin-5-ylidene derivative, 4r)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31955(1,3-thiazolidin-5-ylidene derivative, 4s)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31956(1,3-thiazolidin-5-ylidene derivative, 4t)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31957(1,3-thiazolidin-5-ylidene derivative, 4u)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31958(carbohydrazide derivative, 5a)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31962(carbohydrazide derivative, 5e)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31968(trimethoxybenzyl thiourea, 5k)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Shanghai Institute of Materia Medica

LigandPNGBDBM31969(trimethoxyphenyl prop-2-enamide, 5l)
Affinity DataAssay Description:The enzymatic inhibition assay of HpFabZ was monitored by the spectrophotometric method. The activity of HpFabZ was measured by detection of the decr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2009
Entry Details Article
PubMed
TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM614150(US11744839, Compound Phloxine B)
Affinity DataKd:  1.36E+3nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent

TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM79514(sodium;2-(2,4,5,7-tetraiodo-3-oxido-6-oxo-9-xanthe...)
Affinity DataKd:  160nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent

TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM50061625(4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)
Affinity DataKd:  1.38E+3nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM50103596(CHEBI:9334 | Azulfidine | Azulfidine EN | Azulfidi...)
Affinity DataKd:  440nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM50548283(Olsalazine | C. i. mordant yellow 5 | Dipentum | U...)
Affinity DataKd:  70nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent

TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM50320491(CHEMBL1164729 | 2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-M...)
Affinity DataKd:  1.63E+3nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent

TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM50582214(ATALUREN | Ataluren | Translarna | PTC-124 | PTC12...)
Affinity DataKd:  200nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent

TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM50088376(CHEBI:49005 | Deferasirox | Exjade | ICL670A | US1...)
Affinity DataKd:  1.71E+3nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent

TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM50201618(CHEBI:76138 | Flunixin | SCH-14714 | US11744839, C...)
Affinity DataKd:  270nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetFlavin reductase (NADPH)(Human)
Korea Basic Science Institute

US Patent
LigandPNGBDBM38549(MLS000028605 | cid_25096 | CHEMBL170358 | SMR00005...)
Affinity DataKd:  1.80E+3nMAssay Description:An enzyme activity assay for BLVRB was conducted. Since BLVRB catalyzes the NAD(P)H dependent readuction of FMN, changes in the NAD(P)H concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2023
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245586(CHEMBL4077123)
Affinity DataEC50: <30nMAssay Description:Inhibition of BTK auto-phosphorylation at Y223 in human U2932 cells measured after 4 hrs by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245586(CHEMBL4077123)
Affinity DataEC50:  4.70nMAssay Description:Irreversible inhibition of recombinant full length wild-type 3'-FLAG-tagged BTK (unknown origin) expressed in HEK293T cells assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandPNGBDBM50245586(CHEMBL4077123)
Affinity DataEC50: <30nMAssay Description:Inhibition of BTK auto-phosphorylation at Y223 in human Pfeiffer cells measured after 4 hrs by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
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