Compile Data Set for Download or QSAR
Report error Found 155 with Last Name = 'zhang' and Initial = 'xk'
TargetCellular retinoic acid-binding protein 1(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataKd: >200nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataKd: >200nMAssay Description:Binding affinity for human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 2(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataKd: >200nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataKd:  3nMAssay Description:Binding affinity for human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 1(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataKd:  210nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 2(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  2nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataKd:  16nMAssay Description:Binding affinity for human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 2(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataKd:  1.40nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataKd: >200nMAssay Description:Binding affinity for human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 2(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031459((2Z,4E6E,8E)-3,7-dimethyl-9-(2,6,6-trimethylcycloh...)
Affinity DataKd: >200nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd: >200nMAssay Description:Inhibition of binding to human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 1(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  0.400nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 2(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataKd:  190nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 1(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataKd:  0.300nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 1(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataKd: >200nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 1(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031459((2Z,4E6E,8E)-3,7-dimethyl-9-(2,6,6-trimethylcycloh...)
Affinity DataKd: >200nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 2(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataKd: >200nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 2(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataKd: >200nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataKd: >200nMAssay Description:Binding affinity for human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCellular retinoic acid-binding protein 1(Mouse)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataKd: >200nMAssay Description:Binding affinity for mouse Cytoplasmic retinoic acid binding protein type 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50497864(CHEMBL3319093)
Affinity DataKd:  488nMAssay Description:Binding affinity to RXRalpha ligand binding domain (unknown origin) expressed in human HEK293T cells by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524686(CHEMBL4470378)
Affinity DataKd:  2.94E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50071058(CHEMBL301982 | cid_4274774 | (2R,4aS,6aS,12bR,14aS...)
Affinity DataKd:  320nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50481947(CHEBI:8416 | GNF-Pf-476 | Pristimerine | PRISTIMER...)
Affinity DataKd:  960nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50079524(CHEMBL3417313)
Affinity DataKd:  220nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524687(CHEMBL3928971)
Affinity DataKd:  830nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524688(CHEMBL3980631)
Affinity DataKd:  270nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524689(CHEMBL4451088)
Affinity DataKd:  4.13E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524690(CHEMBL4463133)
Affinity DataKd:  5.56E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50071058(CHEMBL301982 | cid_4274774 | (2R,4aS,6aS,12bR,14aS...)
Affinity DataKd:  290nMAssay Description:Binding affinity to purified Nur77 LBD (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50481949(Dihydrocelastrol | acs.jmedchem.1c00409_ST.616)
Affinity DataKd:  870nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524691(CHEMBL4207143)
Affinity DataKd:  2.69E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524692(CHEMBL4470497)
Affinity DataKd:  3.80E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524693(CHEMBL4459092)
Affinity DataKd:  720nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524694(CHEMBL3892041)
Affinity DataKd:  520nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524695(CHEMBL4446742)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50079525(CHEMBL3417314)
Affinity DataKd:  800nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50103504(Sulindac | CHEBI:9352 | Clinoril)
Affinity DataEC50:  2.27E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50430575(CHEMBL2337794)
Affinity DataEC50:  2.78E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50572732(CHEMBL4870772)
Affinity DataEC50:  1.17E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50572733(CHEMBL4853469)
Affinity DataEC50:  1.84E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50430574(CHEMBL2337793)
Affinity DataEC50: >5.00E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50572734(CHEMBL4870096)
Affinity DataEC50:  6.41E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50572735(CHEMBL4846764)
Affinity DataEC50: >5.00E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50572736(CHEMBL4867346)
Affinity DataEC50:  1.18E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50572737(CHEMBL4865825)
Affinity DataEC50: >5.00E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM84514(Sulindac analogue, 11)
Affinity DataEC50:  930nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50572738(CHEMBL4861380)
Affinity DataEC50:  4.61E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50572739(CHEMBL4864627)
Affinity DataEC50:  1.74E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50572740(CHEMBL4863504)
Affinity DataEC50:  6.29E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 155 total ) | Next | Last >>
Jump to: