Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 573 with Last Name = 'zlotos' and Initial = 'dp'
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266433(CHEMBL445427 | N-(2-{5-Methoxy-2-[(2,3-dihydro-1H-...)
Affinity DataKi:  0.00100nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50114716(CHEMBL329263 | N-[2-(2-Benzyl-5-methoxy-benzofuran...)
Affinity DataKi:  0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50086013(CHEMBL10009 | N-[2-(2-Methoxy-6H-isoindolo[2,1-a]i...)
Affinity DataKi:  0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0680nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50114701(But-3-enoic acid {2-[5-methoxy-2-(3-methoxy-benzyl...)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266405(CHEMBL457128 | N-(3-(3-methoxyphenyl)-3-(naphthale...)
Affinity DataKi:  0.110nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50240952((4-Methoxy-6,7-dihydro-5H-dibenzo[a,c]cyclohepten-...)
Affinity DataKi:  0.160nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011344(CHEMBL3260982)
Affinity DataKi:  0.180nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.220nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50114704(CHEMBL33549 | N-(2-(5-methoxy-2-(3-methoxybenzyl)b...)
Affinity DataKi:  0.25nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM85066(Luzindole,5-Methoxy)
Affinity DataKi:  0.25nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50011344(CHEMBL3260982)
Affinity DataKi:  0.290nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50114704(CHEMBL33549 | N-(2-(5-methoxy-2-(3-methoxybenzyl)b...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50240440(4-P-PDOT | CHEMBL285718 | N-(4-Phenyl-1,2,3,4-tetr...)
Affinity DataKi:  0.460nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50086001(CHEMBL274438 | N-[2-(11-Methoxy-6,7-dihydro-5H-ben...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50086001(CHEMBL274438 | N-[2-(11-Methoxy-6,7-dihydro-5H-ben...)
Affinity DataKi:  0.5nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50340325(CHEMBL1760945 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  0.600nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in HEK293 cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125757(CHEMBL14453 | N,N'-(2,2'-(7,7'-(butane-1,4-diylbis...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50149181(CHEMBL334079 | Cyclopropanecarboxylic acid {3-[2-(...)
Affinity DataKi:  0.630nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM85054(1-[3-(5-Methoxy-1H-indol-3-yl)piperidino]ethanone ...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266354(CHEMBL514280 | N-(2-((1R,3R)-7-methoxy-3-phenyl-1,...)
Affinity DataKi:  0.900nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50366779(METHYLLYCACONITINE)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]methyllycaconitine from human alpha-7 in tsA201 cells coexpressed with 5HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266430(CHEMBL514415 | N-(2-{5-Methoxy-2-[(2,3-dihydro-1H-...)
Affinity DataKi:  1.10nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011356(CHEMBL3260984)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011353(CHEMBL3260987)
Affinity DataKi:  1.20nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50114716(CHEMBL329263 | N-[2-(2-Benzyl-5-methoxy-benzofuran...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]2-iodomelatonin from MT1 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011338(CHEMBL3260979)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50011349(CHEMBL189449)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50340325(CHEMBL1760945 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  1.40nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in HEK293 cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50240952((4-Methoxy-6,7-dihydro-5H-dibenzo[a,c]cyclohepten-...)
Affinity DataKi:  1.40nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50240440(4-P-PDOT | CHEMBL285718 | N-(4-Phenyl-1,2,3,4-tetr...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50011338(CHEMBL3260979)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50241105((E)-N-[3-(3-methoxyphenyl)-3-phenyl-2-propenyl]ace...)
Affinity DataKi:  2.5nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125757(CHEMBL14453 | N,N'-(2,2'-(7,7'-(butane-1,4-diylbis...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011356(CHEMBL3260984)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM82556(melatonin, 6-Methoxy)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011354(CHEMBL3260985)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]GR65630 from human 5HT3A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50086013(CHEMBL10009 | N-[2-(2-Methoxy-6H-isoindolo[2,1-a]i...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011351(CHEMBL1097525)
Affinity DataKi:  5.20nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50266434(CHEMBL515856 | N-(2-{5-Methoxy-2-[(5-methoxy-2,3-d...)
Affinity DataKi:  5.80nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50366779(METHYLLYCACONITINE)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]methyllycaconitine from alpha7 nAChR in tsA201 cells co-expressed with Ric3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266434(CHEMBL515856 | N-(2-{5-Methoxy-2-[(5-methoxy-2,3-d...)
Affinity DataKi:  7.10nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011355(CHEMBL3260986)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50295871(CHEMBL552002 | N-[2-(5-Methoxy-2-{[(4-methoxypheny...)
Affinity DataKi:  8nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50266431(CHEMBL457138 | N-(2-{5-Methoxy-2-[(2,3-dihydro-1H-...)
Affinity DataKi:  8nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 573 total ) | Next | Last >>
Jump to: