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TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM22543(2-[4-(1H-imidazol-4-ylmethyl)phenyl]-4,4-dimethyl-...)
Affinity DatapH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH4R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;perchlorate | 2-...)
Affinity DataKd:  458nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKd:  40.7nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM50143314(CHEMBL298826 | (+)-Epibatidine | 2-(6-Chloro-pyrid...)
Affinity DataKd:  0.0835nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;perchlorate | 2-...)
Affinity DataKd:  3.85E+3nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKd:  310nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM50143314(CHEMBL298826 | (+)-Epibatidine | 2-(6-Chloro-pyrid...)
Affinity DataKd:  2.67nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM50119572(Quinuclidine analogue, 1 | CHEMBL142049 | Dimethyl...)
Affinity DataKd:  4.25E+3nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM92875(Quinuclidine analogue, 2)
Affinity DataKd:  345nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM92876(Quinuclidine analogue, 3)
Affinity DataKd:  141nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM92877(Quinuclidine analogue, 4)
Affinity DataKd:  53.5nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Beactica

LigandPNGBDBM92878(Quinuclidine analogue, 5)
Affinity DataKd:  12.8nMpH: 7.4 T: 2°CAssay Description:Interaction assay using AChBP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50150944(CHEMBL153207)
Affinity DataEC50:  513nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50121205(CHEBI:18295 | Histamine)
Affinity DataEC50:  55nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474422(CHEMBL358028)
Affinity DataEC50:  1.82E+3nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474423(CHEMBL153284)
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474424(CHEMBL153051)
Affinity DataEC50:  1.02E+3nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50407522(CHEMBL554031)
Affinity DataEC50:  33nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474425(CHEMBL356666)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474426(Impentamine)
Affinity DataEC50:  2.30nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474428(CHEMBL152936)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50150943(CHEMBL154529)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50150945(CHEBI:81390 | Immepip)
Affinity DataEC50:  0.132nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474425(CHEMBL356666)
Affinity DataEC50:  3.20nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474422(CHEMBL358028)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50127605(VUF-5297 | (1S,2S)-2-(1H-Imidazol-4-yl)-cyclopropy...)
Affinity DataEC50:  5.90nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474429(CHEMBL150243)
Affinity DataEC50:  1.51E+3nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50407522(CHEMBL554031)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50127607(VUF-5296 | 2-(1H-Imidazol-4-yl)-cyclopropylamine |...)
Affinity DataEC50:  58nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474431(CHEMBL150512)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474432(CHEMBL345954)
Affinity DataEC50:  2.75E+3nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50127605(VUF-5297 | (1S,2S)-2-(1H-Imidazol-4-yl)-cyclopropy...)
Affinity DataEC50:  7.08E+3nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474434(CHEMBL150703)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50170164(Imbutamine)
Affinity DataEC50:  7.40nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50150943(CHEMBL154529)
Affinity DataEC50:  513nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50409817(VUF-5681 | CHEMBL78498)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474430(CHEMBL152948)
Affinity DataEC50:  324nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474433(CHEMBL440730)
Affinity DataEC50:  2.10nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474428(CHEMBL152936)
Affinity DataEC50:  2.30nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474430(CHEMBL152948)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50121205(CHEBI:18295 | Histamine)
Affinity DataEC50:  9.80nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474433(CHEMBL440730)
Affinity DataEC50:  417nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474431(CHEMBL150512)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474435(Homohistamine)
Affinity DataEC50:  43nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474427(CHEMBL153061)
Affinity DataEC50:  741nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50474424(CHEMBL153051)
Affinity DataEC50:  0.389nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474432(CHEMBL345954)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50127607(VUF-5296 | 2-(1H-Imidazol-4-yl)-cyclopropylamine |...)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

LigandPNGBDBM50474426(Impentamine)
Affinity DataEC50: <1.00E+4nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H3 receptor(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50409817(VUF-5681 | CHEMBL78498)
Affinity DataEC50:  8.30nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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