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TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50241166(N6-benzylado | CHEMBL388757 | (2R,3R,4S,5R)-2-(6-(...)
Affinity DataEC50:  384nMAssay Description:Effective concentration for stimulation of [35S]GTP-gamma-S, binding to human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataEC50:  89nMAssay Description:Effective concentration for stimulation of [35S]GTP-gamma-S, binding to human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataEC50:  40nMAssay Description:G-protein activation in human Adenosine A2A receptor expressing CHO cells using cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369514(CHEMBL605266)
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369512(CHEMBL605054)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50207816(N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1,3-dipropyl-2,3...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067081(9-Fluoro-2-furan-2-yl-5,6-dihydro-[1,2,4]triazolo[...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50088475(VUF-5574 | 1-(2-Methoxy-phenyl)-3-(2-pyridin-3-yl-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]DPCPX from rat cortical membranes Adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataKi:  7.14nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50370152(CHEMBL610150)
Affinity DataKi:  7.20nMAssay Description:Binding affinity at human Adenosine A3 receptor expressed in HEK 293 cells by [125I]-AB MECA displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097451(4-Hydroxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369503(CHEMBL606312)
Affinity DataKi:  7.80nMAssay Description:Binding affinity at human Adenosine A3 receptor expressed in HEK 293 cells by [125I]AB-MECA displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataKi:  9.47nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369509(CHEMBL605885)
Affinity DataKi:  9.70nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKi:  11nMAssay Description:Binding affinity at human Adenosine A3 receptor expressed in HEK 293 cells by [125I]-AB MECA displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards rat Adenosine A1 receptor using [3H]-DPCPXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM35804(3-(4-{2-[6-Amino-9-((2R,3R,4S,5S)-5-ethylcarbamoyl...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]NECA from Adenosine A2A receptor in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A2a(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKi:  16nMAssay Description:Binding affinity at Adenosine A2A receptor in rat striatal membrane by [3H]ZM-241385 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50067116(4-Methoxy-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benz...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101787(4-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067081(9-Fluoro-2-furan-2-yl-5,6-dihydro-[1,2,4]triazolo[...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101782(4-Nitro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097441(4-Methoxy-N-(2-phenyl-quinazolin-4-yl)-benzamide |...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097436(4-Methyl-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benza...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369515(CHEMBL604636)
Affinity DataKi:  31nMAssay Description:Binding affinity at human Adenosine A3 receptor expressed in HEK 293 cells by [125I]AB-MECA displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097440(N-(3-Phenyl-[1,2,4]thiadiazol-5-yl)-benzamide | CH...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097423(LUF-5417 | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097423(LUF-5417 | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097432((Cis)-4-Methoxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097432((Cis)-4-Methoxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101783(4-Bromo-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101781(4-Methyl-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101790(N-(4-Phenyl-thiazol-2-yl)-benzamide | CHEMBL60334)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369511(CHEMBL605468)
Affinity DataKi:  41nMAssay Description:Binding affinity at human Adenosine A3 receptor expressed in HEK 293 cells by [125I]AB-MECA displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097442(4-Chloro-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benza...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097426(4-Hydroxy-cyclohexanecarboxylic acid (3-phenyl-[1,...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097426(4-Hydroxy-cyclohexanecarboxylic acid (3-phenyl-[1,...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101786(2,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101784(3,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50207816(N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1,3-dipropyl-2,3...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKi:  63nMAssay Description:Ability to displace [3H]DPCPX from Adenosine A1 receptor in rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50088465(1-Phenyl-3-(3-pyridin-2-yl-isoquinolin-1-yl)-urea ...)
Affinity DataKi:  76nMAssay Description:Binding affinity by its ability to displace [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(LUF-5417 | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(LUF-5417 | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101789(3-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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