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TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080540(CHEMBL57997 | CHEMBL203347 | (2-amino-4,5,6,7-tetr...)
Affinity DataEC50:  6.80E+3nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080539([2-Amino-6-(3-chloro-benzyl)-4,5,6,7-tetrahydro-th...)
Affinity DataEC50:  1.51E+4nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080551((2-Amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)...)
Affinity DataEC50:  1.64E+4nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080548((2-Amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)...)
Affinity DataEC50:  6.00E+3nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080549([2-Amino-6-(3,4-dichloro-benzyl)-4,5,6,7-tetrahydr...)
Affinity DataEC50:  3.20E+4nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080550((2-amino-4,5-dimethylthien-3-yl)-[3-(trifluorometh...)
Affinity DataEC50:  1.47E+4nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080547((2-Amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)...)
Affinity DataEC50:  6.20E+3nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080545((2-amino-6-benzyl-4,5,6,7-tetrahydrothieno[2,3-c]p...)
Affinity DataEC50:  1.13E+4nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080544((2-Amino-6-benzyl-4,5,6,7-tetrahydro-thieno[2,3-c]...)
Affinity DataEC50:  9.20E+3nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080543((2-Amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)...)
Affinity DataEC50:  1.05E+4nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080542((2-Amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)...)
Affinity DataEC50:  3.49E+4nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080541((2-Amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)...)
Affinity DataEC50:  4.50E+3nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080546((2-Amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)...)
Affinity DataEC50:  4.70E+3nMAssay Description:Enhanced 0.5 nM [3H]CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataKi:  7.14nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataKi:  9.47nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101787(4-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101782(4-Nitro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(LUF-5417 | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM23515(pyridine-3-carboxylic acid | CHEMBL573 | [5, 6-3H]...)
Affinity DataKi:  33nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101783(4-Bromo-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101781(4-Methyl-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101790(N-(4-Phenyl-thiazol-2-yl)-benzamide | CHEMBL60334)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101786(2,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101784(3,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50220842(3-butyl-1H-pyrazole-5-carboxylic acid | 5-butyl-1H...)
Affinity DataKi:  72nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(LUF-5417 | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101789(3-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50220850(3-propyl-1H-pyrazole-5-carboxylic acid | 5-propyl-...)
Affinity DataKi:  143nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132140(1,4,5,6-Tetrahydro-cyclopentapyrazole-3-carboxylic...)
Affinity DataKi:  156nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101788(N-(4-Phenyl-thiazol-2-yl)-4-trifluoromethyl-benzam...)
Affinity DataKi:  165nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataKi:  204nMAssay Description:Affinity towards Adenosine A3 receptor expressed in HEK 293 cells using [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataKi:  281nMAssay Description:Affinity towards Adenosine A3 receptor expressed in HEK 293 cells using [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50216550(5-(3-Chloro-benzyl)-1H-pyrazole-3-carboxylic acid ...)
Affinity DataKi:  504nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132132(1H-pyrazole-3-carboxylic acid | CHEMBL128679)
Affinity DataKi:  594nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  670nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50211363(5-isopropyl-3-carboxyl-pyrazole | 5-Isopropyl-1H-p...)
Affinity DataKi:  683nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50216537(3-benzyl-1H-pyrazole-5-carboxylic acid | 5-Benzyl-...)
Affinity DataKi:  1.25E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50101785(4-tert-Butyl-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132146(5-Phenethyl-1H-pyrazole-3-carboxylic acid | CHEMBL...)
Affinity DataKi:  1.57E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]ZM-241385 from A2A receptor in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132142(4,5,6,7-Tetrahydro-1H-indazole-3-carboxylic acid |...)
Affinity DataKi:  3.54E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132144(5-(4-Chloro-benzyl)-1H-pyrazole-3-carboxylic acid ...)
Affinity DataKi:  3.61E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132139(5-(3-Phenyl-propyl)-1H-pyrazole-3-carboxylic acid ...)
Affinity DataKi:  6.30E+3nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132150(5-(4-Methyl-benzyl)-1H-pyrazole-3-carboxylic acid ...)
Affinity DataKi:  2.03E+4nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132136(5-Undecyl-1H-pyrazole-3-carboxylic acid | CHEMBL12...)
Affinity DataKi:  2.14E+4nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132133(cid_818267 | CHEMBL341154 | 5-p-Tolyl-1H-pyrazole-...)
Affinity DataKi:  3.79E+4nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50132149(5-(3-Chloro-phenyl)-1H-pyrazole-3-carboxylic acid ...)
Affinity DataKi:  6.37E+4nMAssay Description:Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
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