Compile Data Set for Download or QSAR
Report error Found 245 of ec50 for UniProtKB: Q00987
LigandPNGBDBM43381(SMR000159660 | MLS000544543 | N'-[3-(2,3-dihydro-1...)
Affinity DataEC50:  2.10nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43398(MLS000569046 | cid_5749438 | (E)-4-(2-sulfanyliden...)
Affinity DataEC50:  10nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43393(cid_1348398 | (5Z)-5-[[5-(3-chlorophenyl)-2-furany...)
Affinity DataEC50:  10nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43437(SMR000324732 | MLS000680115 | cid_7150639 | (6-met...)
Affinity DataEC50:  10nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43492(1-(3,5-dichlorophenyl)-4-[(pyridin-3-ylmethylene)a...)
Affinity DataEC50:  10nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43428(cid_1229743 | 3-[(4-propan-2-ylphenoxy)methyl]-N-(...)
Affinity DataEC50:  20nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43377(cid_2107414 | 2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)...)
Affinity DataEC50:  30nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43343(N-cyclohexyl-2-[(4-cyclohexyl-5-pyridin-3-yl-1,2,4...)
Affinity DataEC50:  40nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43428(cid_1229743 | 3-[(4-propan-2-ylphenoxy)methyl]-N-(...)
Affinity DataEC50:  40nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43395(2-[1-(4-Diethylamino-phenyl)-meth-(E)-ylidene]-1,3...)
Affinity DataEC50:  50nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43399((2Z)-2-[[4-(diethylamino)phenyl]methylidene]-1,3-d...)
Affinity DataEC50:  60nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43399((2Z)-2-[[4-(diethylamino)phenyl]methylidene]-1,3-d...)
Affinity DataEC50:  70nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43362(TETRAMETHYLTHIURAM DISULFIDE | SMR000059023 | MLS0...)
Affinity DataEC50:  80nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43394(MLS000580916 | 4-Methyl-N-{5-[1-(1-methyl-1H-pyrro...)
Affinity DataEC50:  90nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43391(3-[[2,4-bis(chloranyl)phenoxy]methyl]-N-methyl-N-p...)
Affinity DataEC50:  90nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43395(2-[1-(4-Diethylamino-phenyl)-meth-(E)-ylidene]-1,3...)
Affinity DataEC50:  100nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43478(5-(furan-2-ylmethylimino)-N,N-dimethyl-1,2,4-dithi...)
Affinity DataEC50:  100nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43447(MLS000677107 | (5Z)-1-[2-(4-fluorophenyl)ethyl]-5-...)
Affinity DataEC50:  130nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43391(3-[[2,4-bis(chloranyl)phenoxy]methyl]-N-methyl-N-p...)
Affinity DataEC50:  160nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43351(SMR000065944 | 5-methyl-2-pyrazinecarboxylic acid ...)
Affinity DataEC50:  170nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43484(SMR000445626 | (3aR,5R,5aR,8aR,9S,9aS)-9-hydroxy-5...)
Affinity DataEC50:  180nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43362(TETRAMETHYLTHIURAM DISULFIDE | SMR000059023 | MLS0...)
Affinity DataEC50:  180nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43410(MLS000720375 | N-(1,3-benzodioxol-5-yl)-2-[[3-(4-m...)
Affinity DataEC50:  190nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43478(5-(furan-2-ylmethylimino)-N,N-dimethyl-1,2,4-dithi...)
Affinity DataEC50:  200nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43491(MLS000860258 | 3,5-di(3,4,5-trimethoxybenzylidene)...)
Affinity DataEC50:  220nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43443(N5-(isoquinolin-5-ylmethyl)-N6-(2-methoxyethyl)-N5...)
Affinity DataEC50:  220nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43383((Z)-3-(3,4-dimethoxyphenyl)-1-(2-ethylsulfanylbenz...)
Affinity DataEC50:  240nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43478(5-(furan-2-ylmethylimino)-N,N-dimethyl-1,2,4-dithi...)
Affinity DataEC50:  260nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43386((E)-1-(2-prop-2-enylsulfanylbenzimidazol-1-yl)-3-(...)
Affinity DataEC50:  270nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43451(cid_3100036 | MLS000693671 | SMR000285418 | ethyl ...)
Affinity DataEC50:  290nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43477(MLS000766145 | 1,4-Pentadien-3-one, 1,5-di-3-pyrid...)
Affinity DataEC50:  290nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43474((3Z,5E)-1-ethyl-3,5-bis[(4-methoxy-3-oxidanyl-phen...)
Affinity DataEC50:  380nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43464(N'-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-4-me...)
Affinity DataEC50:  380nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM39392(3-[2-(acetylamino)ethyl]-5-methoxy-1H-indole-2-car...)
Affinity DataEC50:  390nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43362(TETRAMETHYLTHIURAM DISULFIDE | SMR000059023 | MLS0...)
Affinity DataEC50:  400nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43383((Z)-3-(3,4-dimethoxyphenyl)-1-(2-ethylsulfanylbenz...)
Affinity DataEC50:  410nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43484(SMR000445626 | (3aR,5R,5aR,8aR,9S,9aS)-9-hydroxy-5...)
Affinity DataEC50:  420nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43366(5'-phenyl-5-propan-2-yl-spiro[1H-indole-3,2'-3H-1,...)
Affinity DataEC50:  430nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43465(SMR000334340 | (Z)-2,3-dichloro-3-[(4-chlorophenyl...)
Affinity DataEC50:  460nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43474((3Z,5E)-1-ethyl-3,5-bis[(4-methoxy-3-oxidanyl-phen...)
Affinity DataEC50:  480nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43392(N-(4-fluorophenyl)-2-(2-nitrophenyl)sulfonylbenzam...)
Affinity DataEC50:  530nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43463((Z)-2,3-bis(chloranyl)-3-[(4-methoxyphenyl)methyls...)
Affinity DataEC50:  540nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43348(SMR000040429 | MLS000039260 | cid_659383 | 6-(meth...)
Affinity DataEC50:  560nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43463((Z)-2,3-bis(chloranyl)-3-[(4-methoxyphenyl)methyls...)
Affinity DataEC50:  560nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43390(1-[3-(3,4-dimethoxyphenyl)acryloyl]-2-(ethylthio)-...)
Affinity DataEC50:  580nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43477(MLS000766145 | 1,4-Pentadien-3-one, 1,5-di-3-pyrid...)
Affinity DataEC50:  580nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43483(cid_282529 | Aromaticin | SMR000445634 | (3aS,5R,5...)
Affinity DataEC50:  590nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43368(Dimethyl-dithiocarbamic acid 1-acetylamino-2,2,2-t...)
Affinity DataEC50:  600nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
LigandPNGBDBM43479(1-Piperidinecarboxylic acid, 4-oxo-3,5-bis(phenyl-...)
Affinity DataEC50:  610nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
LigandPNGBDBM43465(SMR000334340 | (Z)-2,3-dichloro-3-[(4-chlorophenyl...)
Affinity DataEC50:  620nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
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