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Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101509(CHEMBL306947 | N*1*-(2-Cyclohexyl-1-{2-[2-(morphol...)
Affinity DataKi:  0.0100nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101508(2-[3-(4-Chloro-phenyl)-propyl]-N*1*-(2-cyclohexyl-...)
Affinity DataKi:  0.0100nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101512(CHEMBL306033 | N*1*-{2-Cyclohexyl-1-[2-(2-morpholi...)
Affinity DataKi:  0.0100nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101499(CHEMBL74040 | N*1*-(2-Cyclohexyl-1-{2-[2-(4-sulfam...)
Affinity DataKi:  0.0100nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283704((R)-N*1*-[(S)-2-Cyclohexyl-1-(2-morpholin-4-yl-eth...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283715((R)-N*1*-{(S)-2-Cyclohexyl-1-[2-(morpholine-4-sulf...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283705((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-{(S)-2-cyc...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283701(3-{(S)-2-[(R)-5-(4-Chloro-phenyl)-2-hydroxycarbamo...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283703((R)-N*1*-{(S)-2-Cyclohexyl-1-[2-(4-sulfamoyl-pheny...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283708(3-{(S)-2-[(R)-5-(4-Chloro-phenyl)-2-hydroxycarbamo...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101516(3-(3-{2-[5-(4-Chloro-phenyl)-2-hydroxycarbamoylmet...)
Affinity DataKi:  0.0100nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101505(3-(3-{2-[5-(4-Chloro-phenyl)-2-hydroxycarbamoylmet...)
Affinity DataKi:  0.0100nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283713((R)-N*1*-[(S)-2-Cyclohexyl-1-(4-dimethylamino-buty...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283711((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-[(S)-2-cyc...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101518(2-[3-(4-Chloro-phenyl)-propyl]-N*1*-{2-cyclohexyl-...)
Affinity DataKi:  0.0200nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101504(CHEMBL77057 | N*1*-{2-Cyclohexyl-1-[2-(4-dimethyla...)
Affinity DataKi:  0.0200nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283710((R)-N*1*-[(S)-2-Cyclohexyl-1-(4-morpholin-4-yl-but...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101520(CHEMBL77663 | N*1*-{2-Cyclohexyl-1-[2-(4-morpholin...)
Affinity DataKi:  0.0200nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101511(2-[3-(4-Chloro-phenyl)-propyl]-N*1*-(2-cyclohexyl-...)
Affinity DataKi:  0.0300nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101495((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-((S)-2-cyc...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283702((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-{(S)-2-cyc...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101495((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-((S)-2-cyc...)
Affinity DataKi:  0.0300nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283707((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-[(S)-2-cyc...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101503(2-[3-(4-Chloro-phenyl)-propyl]-N*1*-{2-cyclohexyl-...)
Affinity DataKi:  0.0300nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50563343(CHEMBL4746390)
Affinity DataKi:  0.0440nMAssay Description:Inhibition of MMP2 (unknown origin) using Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate incubated for 5 min followed by substrate addition and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101497(2-[3-(4-Chloro-phenyl)-propyl]-N*1*-{2-cyclohexyl-...)
Affinity DataKi:  0.0500nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50283714((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-[(S)-2-cyc...)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50082556((S)-2,2-Dimethyl-4-[4-(pyridin-4-yloxy)-benzenesul...)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50082556((S)-2,2-Dimethyl-4-[4-(pyridin-4-yloxy)-benzenesul...)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of human MMP-2 assessed as inhibition constant using MCA-Pro-Leu-Gly-Leu-DPA-Ala-Arg-NH2 substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101526((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101530((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0600nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101526((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0600nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101492((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101530((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101492((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0620nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101492((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0620nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101513((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101513((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0800nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50082556((S)-2,2-Dimethyl-4-[4-(pyridin-4-yloxy)-benzenesul...)
Affinity DataKi:  0.0830nMAssay Description:Inhibition of matrix metalloprotease-2 (MMP-2).Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50082556((S)-2,2-Dimethyl-4-[4-(pyridin-4-yloxy)-benzenesul...)
Affinity DataKi:  0.0830nMAssay Description:Inhibition of gelatinase-A (Matrix metalloprotease-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50563342(CHEMBL4797032)
Affinity DataKi:  0.0870nMAssay Description:Inhibition of MMP2 (unknown origin) using Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate incubated for 5 min followed by substrate addition and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM11873(N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}-...)
Affinity DataKi: <0.100nMAssay Description:Inhibitors were assayed against purified hMMP-1, hMMP-2, hMMP-3, hMMP-8, hMMP-9, and hMMP-13 using an enzyme assay based on cleavage of the quenched ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM11874(N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]...)
Affinity DataKi:  0.100nMAssay Description:Inhibitors were assayed against purified hMMP-1, hMMP-2, hMMP-3, hMMP-8, hMMP-9, and hMMP-13 using an enzyme assay based on cleavage of the quenched ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM11876(1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxypheny...)
Affinity DataKi: <0.100nMAssay Description:Inhibitors were assayed against purified hMMP-1, hMMP-2, hMMP-3, hMMP-8, hMMP-9, and hMMP-13 using an enzyme assay based on cleavage of the quenched ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM11878(1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-...)
Affinity DataKi: <0.100nMAssay Description:Inhibitors were assayed against purified hMMP-1, hMMP-2, hMMP-3, hMMP-8, hMMP-9, and hMMP-13 using an enzyme assay based on cleavage of the quenched ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM11883(1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]-...)
Affinity DataKi:  0.100nMAssay Description:Inhibitors were assayed against purified hMMP-1, hMMP-2, hMMP-3, hMMP-8, hMMP-9, and hMMP-13 using an enzyme assay based on cleavage of the quenched ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM11889(N-Hydroxy-2-methyl-2-[(4-phenoxyphenyl)sulfonyl]-p...)
Affinity DataKi:  0.100nMAssay Description:Inhibitors were assayed against purified hMMP-1, hMMP-2, hMMP-3, hMMP-8, hMMP-9, and hMMP-13 using an enzyme assay based on cleavage of the quenched ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM11870(4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxy ...)
Affinity DataKi: <0.100nMAssay Description:Inhibitors were assayed against purified hMMP-1, hMMP-2, hMMP-3, hMMP-8, hMMP-9, and hMMP-13 using an enzyme assay based on cleavage of the quenched ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101494((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Human)
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50101494((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.100nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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