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TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-pu...)
Affinity DataKi:  0.00483nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214981((2R,3R,4S)-2-(2-chloro-6-(3-chlorobenzylamino)-9H-...)
Affinity DataKi:  0.0102nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataKi:  0.0480nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50180197((2S,3S,4R,5R)-5-(2-chloro-6-(3-iodobenzylamino)-9H...)
Affinity DataKi:  0.160nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM33283((3-{4-[(3-phenyl-7-propyl-1,2-benzisoxazol-6-yl)ox...)
Affinity DataKi:  0.300nMAssay Description:Agonistic activity was determined in COS1 cells transfected with GAL 4-PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  0.430nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29882(alkynyl ether, 24)
Affinity DataKi:  0.600nM EC50:  2.00E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214980((2R,3R,4S)-2-(2-chloro-6-(2-chlorobenzylamino)-9H-...)
Affinity DataKi:  0.620nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataKi:  0.820nMAssay Description:Binding affinity to PPARdelta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataKi:  1nMAssay Description:Binding affinity to PPARdelta (unknown origin) assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124377(3-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-ylox...)
Affinity DataKi:  2nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29881(alkynyl ether, 23)
Affinity DataKi:  2nM EC50:  220nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304639(9-(5'-Cyclopropylmethylaminocarbonyl-4'-thio-beta-...)
Affinity DataKi:  2.40nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50252829((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-9H-purin-9-...)
Affinity DataKi:  2.5nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304633(9-(5'-Cyclobutylaminocarbonyl-4'-thio-beta-D-ribof...)
Affinity DataKi:  2.60nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304637(9-(5'-Cyclopropylaminocarbonyl-4'-thio-beta-D-ribo...)
Affinity DataKi:  3nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304635(9-(5'-Ethylaminocarbonyl-4-thio-beta-D-ribofuranos...)
Affinity DataKi:  3.20nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124369(CHEMBL367019 | {3-Chloro-4-[3-(3-phenyl-7-propyl-b...)
Affinity DataKi:  3.70nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124384(CHEMBL173494 | {4-[3-(3-Phenyl-7-propyl-benzo[d]is...)
Affinity DataKi:  3.70nMAssay Description:Agonistic activity was determined in COS1 cells transfected with GAL 4-PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29885(alkynyl ether, 27)
Affinity DataKi:  4nM EC50:  470nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29868(alkynyl ether, 10)
Affinity DataKi:  4nM EC50:  54nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124378(2-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-ylox...)
Affinity DataKi:  4.60nMAssay Description:Agonistic activity was determined in COS1 cells transfected with GAL 4-PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50383373(CHEMBL592652 | GSK0660)
Affinity DataKi:  4.60nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124379(2-(4-(3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataKi:  5nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29879(alkynyl ether, 21)
Affinity DataKi:  5nM EC50:  44nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29883(alkynyl ether, 25)
Affinity DataKi:  6nM EC50:  1.20E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29878(alkynyl ether, 20)
Affinity DataKi:  6nM EC50:  43nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataKi:  6.10nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29877(alkynyl ether, 19)
Affinity DataKi:  7nM EC50:  52nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29867(phenoxyacetic acid-ether, 9)
Affinity DataKi:  8nM EC50:  1.90E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29884(alkynyl ether, 26)
Affinity DataKi:  9nM EC50:  340nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29891(alkynyl ether, 33)
Affinity DataKi:  11nM EC50:  1.20E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-pu...)
Affinity DataKi:  11nMAssay Description:Binding affinity to PPAR-delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124383(3-{4-[2-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-ylox...)
Affinity DataKi:  11nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29869(phenoxyacetic acid-ether, 11)
Affinity DataKi:  11nM EC50:  1.70E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29870(phenoxyacetic acid-ether, 12)
Affinity DataKi:  16nM EC50:  1.10E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29886(alkynyl ether, 28)
Affinity DataKi:  16nM EC50:  680nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124371((E)-3-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124388(3-{3-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-ylox...)
Affinity DataKi:  21nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29880(alkynyl ether, 22)
Affinity DataKi:  22nM EC50:  1.40E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124394(2-Methyl-2-{4-[4-(3-phenyl-7-propyl-benzo[d]isoxaz...)
Affinity DataKi:  23nMAssay Description:Agonistic activity was determined in COS1 cells transfected with GAL 4-PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124381(CHEMBL172718 | {3-[3-(3-Phenyl-7-propyl-benzo[d]is...)
Affinity DataKi:  26nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29890(alkynyl ether, 32)
Affinity DataKi:  28nM EC50:  370nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29871(phenoxyacetic acid-ether, 13)
Affinity DataKi:  35nM EC50:  2.20E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29887(alkynyl ether, 29)
Affinity DataKi:  35nM EC50:  420nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29872(phenoxyacetic acid-ether, 14)
Affinity DataKi:  36nM EC50:  2.90E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM29889(alkynyl ether, 31)
Affinity DataKi:  36nM EC50:  350nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124374(3-{4-[4-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-ylox...)
Affinity DataKi:  38nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124376(4-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-ylox...)
Affinity DataKi:  38nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50124391(CHEMBL176421 | {2-[4-(3-Phenyl-7-propyl-benzo[d]is...)
Affinity DataKi:  47nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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