TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.0347nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.0759nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.0832nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.100nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.100nMAssay Description:Binding affinity against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.204nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.234nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.302nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.310nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.230nM Kd: 0.315nM Koff: 8.17E+5s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.400nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.400nMAssay Description:Binding affinity against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 2.80nM Kd: 0.484nM Koff: 6.76E+6s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.589nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.600nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.590nM Kd: 0.608nM Koff: 3.92E+6s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.640nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.550nM Kd: 0.643nM Koff: 4.77E+5s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.708nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.900nMAssay Description:Binding affinity against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 0.977nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.310nM Kd: 1.07nM Koff: 1.53E+6s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 1.07nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 1.10nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.230nM Kd: 1.13nM Koff: 4.43E+6s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.610nM Kd: 1.18nM Koff: 3.23E+5s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 1.18nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 660nM Kd: 1.30nM Koff: 3.48E+5s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.540nM Kd: 1.64nM Koff: 6.63E+5s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 1.64nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.0900nM Kd: 1.95nM Koff: 2.04E+5s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 1.95nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 40nM Kd: 2.99nM Koff: 9.20E+3s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 1.20nM Kd: 3nM Koff: 3.48E+5s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 3.04nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.270nM Kd: 3.83nM Koff: 2.52E+10s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 3.90nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.0540nM Kd: 4.42nM Koff: 5.97E+6s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 4.42nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 700nM Kd: 5nM Koff: 4.36E+4s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.230nM Kd: 7nM Koff: 7.06E+9s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 7.90nMAssay Description:Affinity for HIV ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 10.8nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.400nM Kd: 11nM Koff: 3.55E+5s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 13.9nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.600nM Kd: 14nM Koff: 6.39E+6s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 17.5nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.300nM Kd: 18nM Koff: 2.93E+4s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 1.40nM Kd: 18nM Koff: 1.81E+5s-1Assay Description:Association rate constant for the interaction between inhibitor and HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKd: 18.2nMAssay Description:Binding affinity for human immunodeficiency virus type 1 proteaseMore data for this Ligand-Target Pair