Compile Data Set for Download or QSAR
Report error Found 10 of ki for UniProtKB: Q99500
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 22202BDBM22202({[(4Z)-2-amino-3-hydroxyoctadec-4-en-1-yl]oxy}phos...)
Affinity DataKi:  5.40nM ΔG°:  -10.5kcal/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 23165BDBM23165(CHEMBL366208 | [(2S)-2-amino-3-hydroxy-2-[2-(4-oct...)
Affinity DataKi:  5.90nM ΔG°:  -10.4kcal/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 23163BDBM23163({2-amino-3-hydroxy-2-[2-(4-octylphenyl)ethyl]propo...)
Affinity DataKi:  13nM ΔG°:  -9.99kcal/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 50198836BDBM50198836([3-amino-3-(3-octylphenylcarbamoyl)propyl]-phospho...)
Affinity DataKi:  300nMAssay Description:Displacement of [32P]S1P from human S1P3 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 50133425BDBM50133425(CHEMBL227371 | CHEMBL422074 | Phosphoric acid mono...)
Affinity DataKi:  300nMAssay Description:Displacement of [32P]S1P from human S1P3 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 23164BDBM23164(CHEMBL190006 | [(2R)-2-amino-3-hydroxy-2-[2-(4-oct...)
Affinity DataKi:  586nM ΔG°:  -7.90kcal/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 50248369BDBM50248369(CHEMBL4076530)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [33P]-S1P from S1P3 receptor (unknown origin) expressed in CHOK1 cells after 60 mins by microbeta scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2019
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 50248368BDBM50248368(CHEMBL4085783)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [33P]-S1P from S1P3 receptor (unknown origin) expressed in CHOK1 cells after 60 mins by microbeta scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2019
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 50494302BDBM50494302(CHEMBL3086532)
Affinity DataKi:  4.88E+3nMAssay Description:Inhibition of S1P3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Mitsubishi Pharma

LigandChemical structure of BindingDB Monomer ID 50250631BDBM50250631(CHEMBL4093489)
Affinity DataKi: >5.63E+3nMAssay Description:Displacement of [33P]-S1P from human S1P3 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2019
Entry Details Article
PubMed