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Report error Found 675 of ic50 for UniProtKB: P08588
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378919(CHEMBL2011218)
Affinity DataIC50: 0.0400nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378927(CHEMBL2011226)
Affinity DataIC50: 0.0500nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378913(CHEMBL2011227)
Affinity DataIC50: 0.0500nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378917(CHEMBL2011216)
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378925(CHEMBL2011224)
Affinity DataIC50: 0.100nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378916(CHEMBL2011215)
Affinity DataIC50: 0.100nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378914(CHEMBL2011213)
Affinity DataIC50: 0.110nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378935(CHEMBL2011235)
Affinity DataIC50: 0.140nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378915(CHEMBL2011214)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378918(CHEMBL2011217)
Affinity DataIC50: 0.25nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378926(CHEMBL2011225)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378928(CHEMBL2011228)
Affinity DataIC50: 0.350nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378923(CHEMBL2011222)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378920(CHEMBL2011219)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378922(CHEMBL2011221)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378924(CHEMBL2011223)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50419677(CHEMBL1945035)
Affinity DataIC50: 2nMAssay Description:Displacement of radiolabeled iodocyanopindolol from beta1 adrenoceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataIC50: 2.30nMAssay Description:Compound was evaluated for its Beta adrenergic receptor blocking actionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378934(CHEMBL2011234)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50418942(CHEMBL1807822)
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50418943(CHEMBL1807821)
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataIC50: 4nMAssay Description:Concentration effective against displacing [3H]dihydroalprenolol from beta adrenergic receptor from canine ventricular tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50418944(CHEMBL1807819)
Affinity DataIC50: 4nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50218691(CHEMBL51667)
Affinity DataIC50: 4.30nMAssay Description:Compound was evaluated for its Beta adrenergic receptor blocking actionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50518969(CHEMBL4514723)
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataIC50: 4.90nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-1 adrenergic receptor in dog heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378936(CHEMBL2011236)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50518985(CHEMBL4465278)
Affinity DataIC50: 5.60nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50518977(CHEMBL1160734)
Affinity DataIC50: 5.90nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataIC50: 6.10nMAssay Description:Compound was evaluated for its inhibitory activity against CHO cells expressing the cloned human beta-1 adrenergic receptor (AR) in the presence of [...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50419703(CHEMBL1945042)
Affinity DataIC50: 6.30nMAssay Description:Displacement of radiolabeled iodocyanopindolol from beta1 adrenoceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070125(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataIC50: 6.70nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50419706(CHEMBL1945296)
Affinity DataIC50: 7.90nMAssay Description:Displacement of radiolabeled iodocyanopindolol from beta1 adrenoceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50418945(CHEMBL1807818)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50418946(CHEMBL1807817)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50418958(CHEMBL1807820)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50419704(CHEMBL1945289)
Affinity DataIC50: 10nMAssay Description:Displacement of radiolabeled iodocyanopindolol from beta1 adrenoceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070138(4-{(S)-2-Hydroxy-3-[(S)-3-(4-methoxy-phenyl)-1-met...)
Affinity DataIC50: 10nMAssay Description:Compound was tested for binding affinity against cloned human beta-1 adrenergic receptor from CHO cells using [125I]-iodocyanopindolol as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378930(CHEMBL2011230)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50419682(CHEMBL1945041)
Affinity DataIC50: 10nMAssay Description:Displacement of radiolabeled iodocyanopindolol from beta1 adrenoceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50378933(CHEMBL2011233)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50518979(CHEMBL4434772)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataIC50: 12nMAssay Description:Tested for Beta Adrenergic receptor binding inhibition from canine ventricular tissue, using [3H]dihydroalprenolol as the radioligand in anesthetized...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50419668(CHEMBL1947157)
Affinity DataIC50: 13nMAssay Description:Displacement of radiolabeled iodocyanopindolol from beta1 adrenoceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50518968(CHEMBL4441975)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50518984(CHEMBL4564189)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070142(4-{(S)-2-Hydroxy-3-[3-(4-methoxy-phenyl)-propylami...)
Affinity DataIC50: 15nMAssay Description:Compound was tested for agonist activity against cloned human beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070149(4-((3S)-3-{[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)pro...)
Affinity DataIC50: 15nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50096772(Cyanoguanidine derivative | CHEMBL123745)
Affinity DataIC50: 16nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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