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Report error Found 1521 of ki for UniProtKB: P15823
LigandPNGBDBM50122243(4-Chloro-5-[4-(furan-2-carbonyl)-piperazin-1-yl]-2...)
Affinity DataKi:  0.0520nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230846(CHEMBL2114071)
Affinity DataKi:  0.0680nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230859(CHEMBL309150)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226239(CHEMBL50451)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
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LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226814(CHEMBL6424)
Affinity DataKi:  0.100nMAssay Description:In vitro binding affinity determined for alpha-1 adrenergic receptor by the displacement of [3H]- prazosin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50328498(1-Methyl-4-[8-(2-methyl-2H-tetrazol-5-ylmethyl)-10...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]prozosin from alpha1b receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230848(CHEMBL70872)
Affinity DataKi:  0.110nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50227376(CHEMBL8689)
Affinity DataKi:  0.140nMAssay Description:Binding affinity towards alpha-1 adrenergic receptor from rat brain homogenate preparation by displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50328499(1-Methyl-4-[8-(1-methyl-1H-tetrazol-5-ylmethyl)-10...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]prozosin from alpha1b receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50328478(1-Methyl-4-(8-(2-methyl-2H-tetrazol-5-yl)-10,11-di...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]prozosin from alpha1b receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50227298(CHEMBL147255)
Affinity DataKi:  0.150nMAssay Description:Binding affinity for alpha-1 adrenergic receptor by displacement of [3H]-prazosin from rat brain homogenate preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50227290(CHEMBL148457)
Affinity DataKi:  0.150nMAssay Description:Binding affinity for alpha-1 adrenergic receptor by displacement of [3H]-prazosin from rat brain homogenate preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity for alpha-1 adrenergic receptor by displacement of [3H]-prazosin from rat brain homogenate preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of [3H]- prazosin binding against Alpha-1B adrenergic receptor from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226234(CHEMBL50979)
Affinity DataKi:  0.160nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.160nMAssay Description:Compound was tested for the inhibition of [3H]prazosin binding Alpha-1 adrenergic receptor of crude rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226235(CHEMBL54288)
Affinity DataKi:  0.180nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226227(CHEMBL52155)
Affinity DataKi:  0.180nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.190nMAssay Description:In vitro binding affinity determined for alpha-1 adrenergic receptor by the displacement of [3H]- prazosin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109058(1H-4-indolyl 2-[4-(1H-3-indolyl)-1,2,3,6-tetrahydr...)
Affinity DataKi:  0.190nMAssay Description:In vitro binding affinity towards Alpha-1 adrenergic receptor was determined by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity to Alpha-1 adrenergic receptor by displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226233(CHEMBL275524)
Affinity DataKi:  0.190nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity against alpha-1-adrenoceptor was determined by displacement of [3H]-prazosin in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity towards alpha-1 adrenergic receptor from rat brain homogenate preparation by displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.190nMAssay Description:Compound was tested for its binding affinity for alpha-1 adrenergic receptor site by displacement of [3H]clonidine at 10e-6 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226844(CHEMBL415288)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity determined for alpha-1 adrenergic receptor by the displacement of [3H]- prazosin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.200nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
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Curated by ChEMBL
LigandPNGBDBM50487287((+)-CYCLAZOSIN)
Affinity DataKi:  0.209nMAssay Description:Binding affinity to alpha1B adrenoreceptor in Rattus norvegicus (rat) liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50006952(2-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-...)
Affinity DataKi:  0.210nMAssay Description:Alpha-1-adrenergic receptor binding affinity of the compound, value taken from literatureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50066109(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-2,6-...)
Affinity DataKi:  0.210nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226846(CHEMBL6474)
Affinity DataKi:  0.220nMAssay Description:In vitro binding affinity determined for alpha-1 adrenergic receptor by the displacement of [3H]- prazosin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity by its ability to displace [3H]prazosin radioligand from Alpha-1 adrenergic receptor on rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity towards alpha-1 adrenergic receptor in rat cortex membrane using [3H]-prazosin radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226237(CHEMBL299584)
Affinity DataKi:  0.240nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in rat cerebral cortex membranes after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50040253(3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50122239(4-Chloro-5-{4-[2-(2-ethoxy-phenoxy)-ethyl]-piperaz...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226229(CHEMBL52439)
Affinity DataKi:  0.260nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226228(CHEMBL50137)
Affinity DataKi:  0.270nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226225(CHEMBL50746)
Affinity DataKi:  0.270nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50227379(CHEMBL267428)
Affinity DataKi:  0.290nMAssay Description:Binding affinity towards alpha-1 adrenergic receptor from rat brain homogenate preparation by displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226238(CHEMBL301614)
Affinity DataKi:  0.290nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.300nMAssay Description:Alpha-1 adrenergic receptor binding affinity was evaluated by its ability to displace [3H]prazosin in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50226241(CHEMBL301749)
Affinity DataKi:  0.310nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226230(CHEMBL50084)
Affinity DataKi:  0.320nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.320nMAssay Description:Evaluated for binding affinity against alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230870(CHEMBL70498)
Affinity DataKi:  0.340nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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