Compile Data Set for Download or QSAR
Report error Found 8 of kd for UniProtKB: P97287
LigandPNGBDBM21447(4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity for GST-tagged mouse MCL1 expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM21400(N-[(4-{[(2R)-4-(dimethylamino)-1-(phenylsulfanyl)b...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity for GST-tagged mouse MCL1 expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50262597([(2S,3R,4S)-1-(Biphenyl-4-carbonyl)-4-[(biphenyl-4...)
Affinity DataKd:  2.50E+4nMAssay Description:Binding affinity to mouse Mcl-1 expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262594((2S,3R,4S)-4-[(Biphenyl-4-carbonyl)-amino]-2-carbo...)
Affinity DataKd:  1.00E+5nMAssay Description:Binding affinity to mouse Mcl-1 expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262593(2-((2S,3R,4S)-4-(2-naphthamido)-3-hydroxy-6-((2-me...)
Affinity DataKd:  2.00E+5nMAssay Description:Binding affinity to mouse Mcl-1 expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262591([(2S,3R,4S)-4-Allyloxycarbonylamino-1-(biphenyl-4-...)
Affinity DataKd:  3.00E+5nMAssay Description:Binding affinity to mouse Mcl-1 expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262596(2-((2S,3R,4S)-4-(2-naphthamido)-1-(2-naphthoyl)-3-...)
Affinity DataKd:  3.00E+5nMAssay Description:Binding affinity to mouse Mcl-1 expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50262590(2-((2S,3R,4S)-1-(2-naphthoyl)-4-(allyloxycarbonyl)...)
Affinity DataKd:  5.00E+5nMAssay Description:Binding affinity to mouse Mcl-1 expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed