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Found 93 of ec50 for UniProtKB: P51449
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106285(CHEMBL3596279 | US9550771, Example 91)
Affinity DataEC50:  2nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268455(4-[8-chloro-3-(2-chloro-6- cyclopropyl- benzoyl)im...)
Affinity DataEC50:  2nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106287(CHEMBL3598148 | US9550771, Example 17)
Affinity DataEC50:  2nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268417(4-[3-(2,6- dichlorobenzoyl)imidazo[1,5 a]pyridin-1...)
Affinity DataEC50:  3nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268454(4-[3-(2-chloro-6-morpholino- benzoyl)imidazo[1,5-a...)
Affinity DataEC50:  3nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268449(4-[6-(azetidine-1-carbonyl)-3-(2- chloro-6-cyclopr...)
Affinity DataEC50:  3nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268425(4-[3-[2-chloro-6- (trifluoromethyl)benzoyl]-5,6,7,...)
Affinity DataEC50:  3nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268439(4-[3-(2- cyclopropylbenzoyl)imidazo[1,5- a]pyridin...)
Affinity DataEC50:  3nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268413(2-hydroxy-4-[3-[2- (trifluoromethyl)benzoyl]imidaz...)
Affinity DataEC50:  3nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268479(4-[3-[2-chloro-6- (trifluoromethyl)benzoyl]-5,6,7,...)
Affinity DataEC50:  4nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268483(4-[3-[2-chloro-6- (trifluoromethyl)benzoyl]-5,6,7,...)
Affinity DataEC50:  4nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268481(4-[3-[2-chloro-6- (trifluoromethyl)benzoyl]-5,6,7,...)
Affinity DataEC50:  6nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268474(4-[3-[2-bromo-6- (trifluoromethyl)benzoyl]-5,6,7,8...)
Affinity DataEC50:  6nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268444(4-[3-(2-chloro-6-cyclopropyl- benzoyl)-6- (dimethy...)
Affinity DataEC50:  6nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268475(4-[3-(2-bromo-6-chloro-benzoyl)- 5,6,7,8-tetrahydr...)
Affinity DataEC50:  7nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268427(2-acetoxy-4-[3-[2-chloro-6- (trifluoromethyl)benzo...)
Affinity DataEC50:  7nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268469(4-[3-(2,6-dichlorobenzoyl)- 5,6,7,8-tetrahydroimid...)
Affinity DataEC50:  8nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268404(4-(3-(2-(Trifluoromethyl)benzoyl)imidazo[1,5-a]pyr...)
Affinity DataEC50:  8nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268435(4-[3-(2-chloro-6-cyclopropyl- benzoyl)imidazo[1,5-...)
Affinity DataEC50:  9nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106288(CHEMBL3598149 | US9550771, Example 28)
Affinity DataEC50:  9nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268491(4-[3-(2-chloro-6-cyclopropyl- benzoyl)-5,6,7,8- te...)
Affinity DataEC50:  9nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106286(CHEMBL3598141 | US9550771, Example 27)
Affinity DataEC50:  10nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268482(4-[3-[2-chloro-6- (trifluoromethyl)benzoyl]-5,6,7,...)
Affinity DataEC50:  12nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268461((3S,4R)-1-[8-chloro-3-(2-chloro- 6-cyclopropyl- be...)
Affinity DataEC50:  13nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268478(2-hydroxy-4-[3-[2-methyl-6- (trifluoromethyl)benzo...)
Affinity DataEC50:  14nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268457((3S,4R)-1-[3-(2-chloro-6- cyclopropyl-benzoyl)-6- ...)
Affinity DataEC50:  19nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268445(4-[3-(2-chloro-6-cyclopropyl- benzoyl)-6- (dimethy...)
Affinity DataEC50:  22nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268402(4-(3-(2,6-Dichlorobenzoyl)imidazo[1,5-a]pyridin-1-...)
Affinity DataEC50:  26nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106290(CHEMBL3596276 | US9550771, Example 89)
Affinity DataEC50:  27nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268450((3S,4R)-1-[3-(2-chloro-6- cyclopropyl- benzoyl)imi...)
Affinity DataEC50:  29nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106289(CHEMBL3596270 | US9550771, Example 21)
Affinity DataEC50:  32nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268436(4-[3-(2-chloro-6-cyclopropyl- benzoyl)imidazo[1,5-...)
Affinity DataEC50:  45nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268463(2-hydroxy-4-[3-[2- (trifluoromethyl)benzoyl]-5,6,7...)
Affinity DataEC50:  49nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268448(2-hydroxy-4-[3-(2- morpholinobenzoyl)imidazo[1,5- ...)
Affinity DataEC50:  50nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268456(1-[6-(azetidine-1-carbonyl)-3-(2- chloro-6-cyclopr...)
Affinity DataEC50:  50nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106302(CHEMBL3598142 | US9550771, Example 22)
Affinity DataEC50:  58nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268450((3S,4R)-1-[3-(2-chloro-6- cyclopropyl- benzoyl)imi...)
Affinity DataEC50:  63nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268459(1-[3-(2-chloro-6-cyclopropyl- benzoyl)-6-(3-methox...)
Affinity DataEC50:  70nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268438(1-[3-[2-chloro-6- (trifluoromethyl)benzoyl]imidazo...)
Affinity DataEC50:  72nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106296(CHEMBL3596273 | US9550771, Example 69)
Affinity DataEC50:  77nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268406(1-(3-(2-chloro-6-(trifluoromethyl)benzoyl)imidazo[...)
Affinity DataEC50:  77nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268419(4-[6-(2,6- dichlorobenzoyl)imidazo[1,5- a]pyrimidi...)
Affinity DataEC50:  84nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106293(CHEMBL3596269 | US9550771, Example 41)
Affinity DataEC50:  97nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50106325(CHEMBL3598150 | US9550771, Example 29)
Affinity DataEC50:  103nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268447(4-[3-(2-chloro-6-cyclopropyl- benzoyl)imidazo[1,5-...)
Affinity DataEC50:  109nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268440(6-[3-[2-chloro-6- (trifluoromethyl)benzoyl]imidazo...)
Affinity DataEC50:  111nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268446(1-[3-(2-chloro-6-cyclopropyl- benzoyl)imidazo[1,5-...)
Affinity DataEC50:  139nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268426(3-chloro-4-[3-[2-chloro-6- (trifluoromethyl)benzoy...)
Affinity DataEC50:  171nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268407(4-[3-[2- (trifluoromethyl)benzoyl]imidazo [1,5-a]p...)
Affinity DataEC50:  179nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [262-507](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268416(3,5-difluoro-4-[3-[2- (trifluoromethyl)benzoyl]imi...)
Affinity DataEC50:  189nMT: 2°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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