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Found 19 of ic50 for UniProtKB: A2RTI3
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364367(CHEMBL1950283)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364353(CHEMBL1950109)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364366(CHEMBL1950282)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM228618(BDBM50364365 | US9345789, LI-2)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364368(CHEMBL1950284)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364356(CHEMBL1950112)
Affinity DataIC50:  9.30nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM36332(LI-1 | Legumain Inhibitor -1)
Affinity DataIC50:  9.30nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM36332(LI-1 | Legumain Inhibitor -1)
Affinity DataIC50:  11.5nMpH: 5.8 T: 2°CAssay Description:IC50 measurements and enzyme kinetics assays were performed on a Spectramax M5 fluorescent plate reader (Molecular Devices).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364358(CHEMBL1950273)
Affinity DataIC50:  17nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364354(CHEMBL1950110)
Affinity DataIC50:  141nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364355(CHEMBL1950111)
Affinity DataIC50:  148nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364360(CHEMBL1950275)
Affinity DataIC50:  167nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364357(CHEMBL1950272)
Affinity DataIC50:  198nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364363(CHEMBL1950278)
Affinity DataIC50:  267nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364359(CHEMBL1950274)
Affinity DataIC50:  638nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM36333(LI-0 | Legumain Inhibitor -0)
Affinity DataIC50:  704nMpH: 5.8 T: 2°CAssay Description:IC50 measurements and enzyme kinetics assays were performed on a Spectramax M5 fluorescent plate reader (Molecular Devices).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364364(CHEMBL1950279)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364361(CHEMBL1950276)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Mus musculus)
Stanford University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50364362(CHEMBL1950277)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed