Compile Data Set for Download or QSAR
maximum 50k data
Found 119 of ec50 data for polymerid = 49000249
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337291(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419652(MILVETEROL)
Affinity DataEC50:  0.0501nMAssay Description:Agonist activity at beta2 receptor in guinea pig trachea assessed as fast onset of inhibition of electrically stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337299(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50295573(BR-AEA | CHEMBL552398)
Affinity DataEC50:  0.0720nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring assessed as bronchorelaxation activity against histamine-induced co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337301(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50365058(CHEMBL1951067)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50151720(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Affinity DataEC50:  0.126nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50151720(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Affinity DataEC50:  0.126nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337302(3-((3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihy...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50151720(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419675(CHEMBL1945032)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig trachea assessed as reduction in methacholine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419008(CHEMBL1814277 | CHEMBL1814278)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig trachea assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337300(1-benzyl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337294(1-(2,6-dichlorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337293(1-(4-fluorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337292(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337295(1-benzhydryl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419687(CHEMBL1947151)
Affinity DataEC50:  0.251nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig trachea assessed as reduction in methacholine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419670(CHEMBL1944691)
Affinity DataEC50:  0.251nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig trachea assessed as reduction in methacholine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419310(CHEMBL1835859)
Affinity DataEC50:  0.251nMAssay Description:Agonist activity at beta2 adrenergic receptor in guinea pig tracheal strip assessed as inhibition of electrically-induced bronchocontractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419689(CHEMBL1945033)
Affinity DataEC50:  0.316nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig trachea assessed as reduction in methacholine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50151720(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Affinity DataEC50:  0.316nMAssay Description:Agonist activity at beta2 adrenergic receptor in guinea pig tracheal strip assessed as inhibition of electrically-induced bronchocontractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50151720(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Affinity DataEC50:  0.316nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig trachea assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM25769(4-[2-(tert-butylamino)-1-hydroxyethyl]-2-(hydroxym...)
Affinity DataEC50:  0.454nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring assessed as bronchorelaxation activity against histamine-induced co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50365057(CHEMBL1951066)
Affinity DataEC50:  0.501nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419688(CHEMBL1947152)
Affinity DataEC50:  0.501nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig trachea assessed as reduction in methacholine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419680(CHEMBL1945039)
Affinity DataEC50:  0.501nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig trachea assessed as reduction in methacholine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337296(1-(biphenyl-2-yl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy-...)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419011(CHEMBL1814268)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig trachea assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337303(1-(4-tert-butylbenzyl)-3-(3-(2-(2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419010(CHEMBL1814279 | CHEMBL1814280)
Affinity DataEC50:  1nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig trachea assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444835(CHEMBL3099249)
Affinity DataEC50:  1nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50318159(8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-diethylindan-2-y...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337298(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444835(CHEMBL3099249)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419317(CHEMBL1835854)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at beta2 adrenergic receptor in guinea pig tracheal strip assessed as inhibition of electrically-induced bronchocontractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM86453(CAS_73573-87-2 | Formoterol | NSC_3083544)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at beta2 receptor in guinea pig trachea assessed as fast onset of inhibition of electrically stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419312(CHEMBL1835862)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at beta2 adrenergic receptor in guinea pig tracheal strip assessed as inhibition of electrically-induced bronchocontractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50018589(CHEMBL3290999)
Affinity DataEC50:  2nMAssay Description:Agonist activity at beta2 receptor in guinea pig trachea assessed as slow onset of inhibition of electrically stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50018587(CHEMBL3290997)
Affinity DataEC50:  2nMAssay Description:Agonist activity at beta2 receptor in guinea pig trachea assessed as slow onset of inhibition of electrically stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50343153(CHEMBL1773197 | N-(3-(3-((R)-3-(diisopropylamino)-...)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig trachea assessed as bronchorelaxation activity against histamine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50295573(BR-AEA | CHEMBL552398)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring assessed as bronchorelaxation activity against carbachol-induced co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419309(CHEMBL1835853)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at beta2 adrenergic receptor in guinea pig tracheal strip assessed as inhibition of electrically-induced bronchocontractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419015(CHEMBL1814272)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig trachea assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM25771(1-hydroxy-2-naphthoic acid;4-[1-hydroxy-2-[6-(4-ph...)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig trachea assessed as inhibition of histamine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
Affinity DataEC50:  3nMAssay Description:Activity for Beta-2 adrenergic receptor was assessed from effect on relaxation of guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50419660(CHEMBL1945292)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig trachea assessed as reduction in methacholine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337297(1-Adamantan-1-ylmethyl-3-(3-{2-[2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50343161(5-((R)-2-(4-(4-(3-((R)-3-(diisopropylamino)-1-phen...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig trachea assessed as bronchorelaxation activity against histamine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444836(CHEMBL3099248)
Affinity DataEC50:  5nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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