Compile Data Set for Download or QSAR
maximum 50k data
Found 24 of kd for UniProtKB: Q13936
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50318494(3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...)
Affinity DataKd:  0.260nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataKd:  0.400nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50227245(CHEMBL3392281)
Affinity DataKd:  2.60nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035794(4-Methyl-2-methylsulfanyl-13-nitro-3,8,9,10,11,16b...)
Affinity DataKd:  5nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50226760(CHEMBL2398396)
Affinity DataKd:  12nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035795(4-Methyl-2-methylsulfanyl-3,8,9,10,11,16b-hexahydr...)
Affinity DataKd:  18nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035800((S)-2,6-Dimethyl-5-nitro-4-(2-trifluoromethyl-phen...)
Affinity DataKd:  18nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50015432(6-Methyl-2-methylsulfanyl-4-(3-nitro-phenyl)-1,4-d...)
Affinity DataKd:  23nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035790(6-Methyl-2-methylsulfanyl-4-(2-methylsulfanyl-3-ni...)
Affinity DataKd:  30nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50226761(CHEMBL3392285)
Affinity DataKd:  35nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50226804(CHEMBL88149)
Affinity DataKd:  105nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50226978(CHEMBL282279)
Affinity DataKd:  120nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50016385(4-Methyl-2-(3-nitro-phenyl)-2,5-dihydro-benzo[b][1...)
Affinity DataKd:  360nMAssay Description:Inhibition of [3H]-nitrendipine binding to calcium channels of guinea pig myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035789(6-Methyl-2-methylsulfanyl-4-(3-nitro-phenyl)-1,4-d...)
Affinity DataKd:  480nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50016388(5-(2-Dimethylamino-ethyl)-4-methyl-2-(3-nitro-phen...)
Affinity DataKd:  488nMAssay Description:Inhibition of [3H]-nitrendipine binding to calcium channels of guinea pig myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035797(4-Methyl-2-methylsulfanyl-15-nitro-3,8,9,10,11,16b...)
Affinity DataKd:  873nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035793(6-Methyl-2-methylsulfanyl-4-(2-methylsulfanyl-phen...)
Affinity DataKd:  1.52E+3nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035802(6-Methyl-2-methylsulfanyl-4-(2-methylsulfanyl-5-ni...)
Affinity DataKd:  2.70E+3nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50226808(CHEMBL3392278)
Affinity DataKd:  3.40E+3nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035799(2-Methylsulfanyl-4-(2-methylsulfanyl-3-nitro-pheny...)
Affinity DataKd:  1.37E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035796(2-Methylsulfanyl-4-(3-nitro-phenyl)-4,7-dihydro-1H...)
Affinity DataKd:  3.69E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035791(2-Methylsulfanyl-4-(2-methylsulfanyl-phenyl)-4,7-d...)
Affinity DataKd:  4.52E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035801(2-Methylsulfanyl-4-(2-methylsulfanyl-5-nitro-pheny...)
Affinity DataKd: >5.00E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Squibb Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50035798(4-(2-Butylsulfanyl-phenyl)-2-methylsulfanyl-4,7-di...)
Affinity DataKd: >5.00E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed