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TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0350nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha3-beta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50143314((+)-Epibatidine | (-)-epibatidine | (1R,2R,4S)-2-(...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK243 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK cell membranes after 4 hrs by liquid scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to human alpha3beta4 nAChRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50162983(6-[5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-3-yl]...)
Affinity DataKi:  0.230nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha3-beta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.457nMAssay Description:Binding affinity of the compound was determined against Nicotinic acetylcholine receptor using [3H]-(-)-nicotine radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406472(CHEMBL4163848)
Affinity DataKi:  0.684nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406641(CHEMBL4170527)
Affinity DataKi:  0.799nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406541(CHEMBL4163257)
Affinity DataKi:  0.818nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406792(CHEMBL4174509)
Affinity DataKi:  0.988nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406686(CHEMBL4167298)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406544(CHEMBL4174940)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406500(CHEMBL4166573)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406685(CHEMBL4164252)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406539(CHEMBL4175573)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534298(CHEMBL4438684)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534286(CHEMBL4453542)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534287(CHEMBL4519018)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to alpha3beta4 nAChR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50500410(CHEMBL3745799)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534288(CHEMBL4472617)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50140291(CHEMBL3758455)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]-epibatidine from human alpha3beta4 nACh receptor expressed in HEK293 cells preincubated for 5 mins followed by radioligand addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406704(CHEMBL4160411)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
Affinity DataKi:  5nMAssay Description:Binding affinity to human alpha3beta4 nAChRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534291(CHEMBL4559236)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50135594((+/-)-2-(6-chloropyridin-3-yl)-9-aza-bicyclo[4.2.1...)
Affinity DataKi:  6.5nMAssay Description:Binding affinity towards alpha3-beta4 subtype of neuronal nicotinic acetylcholine receptor (nAChR) using [3H]-epibatidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534299(CHEMBL4450133)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50162988(3-[5-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-pyridin...)
Affinity DataKi:  7.10nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha3-beta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534300(CHEMBL4442125)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534284(CHEMBL4468804)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50049756(3-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-pyridine |...)
Affinity DataKi:  7.70nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha3-beta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50162986(3-Ethynyl-5-((S)-1-methyl-pyrrolidin-2-ylmethoxy)-...)
Affinity DataKi:  8.20nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha3-beta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50538046(CHEMBL4647198)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in IMR32 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534292(CHEMBL4437323)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50097613(3-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-5-phenylet...)
Affinity DataKi:  8.60nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha3-beta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406687(CHEMBL4164706)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50465459(CHEMBL4290888)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK cell membranes after 4 hrs by liquid scintillation counting ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50465456(CHEMBL4283703)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK cell membranes after 4 hrs by liquid scintillation counting ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM604954(US11667638, Example 160)
Affinity DataKi:  11.9nMAssay Description:The binding of a group of compounds mentioned above were tested for their affinity at different nAChR subtypes, specifically the α4β2, the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534297(CHEMBL4443082)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50162987(6-[5-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-pyridin...)
Affinity DataKi:  13nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha3-beta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50406540(CHEMBL4177240)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50498034(CHEMBL3329543)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534296(CHEMBL4557590)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50162984(3-(6-Fluoro-hex-1-ynyl)-5-((S)-1-methyl-pyrrolidin...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha3-beta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50549596(CHEMBL4785648)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-epibatidine from human alpha3beta4 transfected in HEK293 cell membranes preincubated for 5 mins followed by [3H]-epibatidine add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534283(CHEMBL4440403)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50534282(CHEMBL4437189)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50515321(CHEMBL4543232)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK243 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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