Affinity DataIC50: 2.20nMAssay Description:In vitro antagonist potency in transactivation assay in NIH3T3 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:In vitro antagonist potency in transactivation assay in NIH3T3 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Agonist activity at GR in mouse RAW cells assessed as suppression of TNF-alpha-induced IL-6 productionMore data for this Ligand-Target Pair