Compile Data Set for Download or QSAR
Report error Found 125 of ki for UniProtKB: Q9Y271
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227363(CHEMBL299837)
Affinity DataKi:  0.100nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227366(CHEMBL48927)
Affinity DataKi:  0.200nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50009075(CHEMBL22033 | ICI 198615 | [1-(4-Benzenesulfonylam...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227364(CHEMBL299093)
Affinity DataKi:  0.25nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227361(CHEMBL51585)
Affinity DataKi:  0.25nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM50009073(cyclopentyl 3-(2-methoxy-4-((o-tolylsulfonyl)carba...)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227365(CHEMBL300096)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227358(CHEMBL412056)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227356(CHEMBL49944)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227355(CHEMBL296821)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227642(CHEMBL50562)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227640(CHEMBL297952)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227390(CHEMBL301616)
Affinity DataKi:  0.5nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM50292408(5S-hydroxy-6R-(S-cysteinylglycinyl)-7E,9E,11E,14Z-...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]LTD4 from LTD4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227389(CHEMBL51580)
Affinity DataKi:  0.700nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227367(CHEMBL48435)
Affinity DataKi:  0.800nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50023198(CHEMBL21333 | N-(4-oxo-2-(1H-tetrazol-5-yl)-4H-chr...)
Affinity DataKi:  0.800nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227638(CHEMBL49566)
Affinity DataKi:  1.40nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50070919(C,C,C-Trifluoro-N-{3-[(2R,3S,4R)-6-(5-fluoro-benzo...)
Affinity DataKi:  2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50070919(C,C,C-Trifluoro-N-{3-[(2R,3S,4R)-6-(5-fluoro-benzo...)
Affinity DataKi:  2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50009073(cyclopentyl 3-(2-methoxy-4-((o-tolylsulfonyl)carba...)
Affinity DataKi:  2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCysteinyl leukotriene receptor 1(Human)
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM85673(NSC_5311297 | CAS_5311297 | Montelukast)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50215874(CHEMBL52102)
Affinity DataKi:  3nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227354(CHEMBL51289)
Affinity DataKi:  5.60nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227353(CHEMBL51239)
Affinity DataKi:  6.80nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228527(CHEMBL93991)
Affinity DataKi:  8nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227359(CHEMBL51061)
Affinity DataKi:  10nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM50009070(CHEMBL22776 | 3-(2-Carboxy-ethylsulfanyl)-2-hydrox...)
Affinity DataKi:  10nMAssay Description:Binding affinity against Cysteinyl leukotriene D4 receptor in human lung membranes using [3H]LTD4 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM50001285(3-(((3-(2-(7-chloroquinoline-2-yl)ethenyl)phenyl)(...)
Affinity DataKi:  10.4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of California Irvine

Curated by PDSP Ki Database
LigandPNGBDBM50013901(CHEMBL97356 | 2-(4-{2-[2-(1H-Tetrazol-5-yl)-ethyl]...)
Affinity DataKi:  11nMAssay Description:In vitro binding affinity against Cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228524(CHEMBL317945)
Affinity DataKi:  11nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228506(CHEMBL97656)
Affinity DataKi:  12nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50070921(3-[6-(5-Fluoro-benzothiazol-2-ylmethoxy)-4-hydroxy...)
Affinity DataKi:  14nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228530(CHEMBL97400)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228517(CHEMBL328815)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228525(CHEMBL98232)
Affinity DataKi:  17nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50013536(2-{4-[4-(2H-Tetrazol-5-yl)-butyl]-phenoxymethyl}-q...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50215871(CHEMBL415954)
Affinity DataKi:  19nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228512(CHEMBL264799)
Affinity DataKi:  20nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228519(CHEMBL97713)
Affinity DataKi:  21nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228511(CHEMBL421750)
Affinity DataKi:  22nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228523(CHEMBL97693)
Affinity DataKi:  24nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228526(CHEMBL96592)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228529(CHEMBL420082)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50215875(CHEMBL299779)
Affinity DataKi:  27nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228531(CHEMBL97401)
Affinity DataKi:  31nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228510(CHEMBL98517)
Affinity DataKi:  31nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228508(CHEMBL329753)
Affinity DataKi:  34nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50013534(CHEMBL418551 | 2-{3-[3-(1H-Tetrazol-5-yl)-propoxy]...)
Affinity DataKi:  42nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50228520(CHEMBL97701)
Affinity DataKi:  43nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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